DK1458386T3 - Aroylpyrrolheteroaryl- og methanolforbindelser til behandling af en lidelse i centralnervesystemet - Google Patents

Aroylpyrrolheteroaryl- og methanolforbindelser til behandling af en lidelse i centralnervesystemet

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Publication number
DK1458386T3
DK1458386T3 DK02799923T DK02799923T DK1458386T3 DK 1458386 T3 DK1458386 T3 DK 1458386T3 DK 02799923 T DK02799923 T DK 02799923T DK 02799923 T DK02799923 T DK 02799923T DK 1458386 T3 DK1458386 T3 DK 1458386T3
Authority
DK
Denmark
Prior art keywords
aroylpyrrole
heteroaryl
treatment
nervous system
central nervous
Prior art date
Application number
DK02799923T
Other languages
Danish (da)
English (en)
Inventor
John R Carson
Ellen E Codd
Philip M Pitis
Original Assignee
Ortho Mcneil Pharm Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ortho Mcneil Pharm Inc filed Critical Ortho Mcneil Pharm Inc
Application granted granted Critical
Publication of DK1458386T3 publication Critical patent/DK1458386T3/da

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • A—HUMAN NECESSITIES
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    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/06—Anti-spasmodics, e.g. drugs for colics, esophagic dyskinesia
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    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
    • A—HUMAN NECESSITIES
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    • A—HUMAN NECESSITIES
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings

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  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
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  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Cardiology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Diabetes (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Psychiatry (AREA)
  • Hospice & Palliative Care (AREA)
  • Ophthalmology & Optometry (AREA)
  • Urology & Nephrology (AREA)
  • Endocrinology (AREA)
  • Virology (AREA)
  • Dermatology (AREA)
  • Hematology (AREA)
  • Communicable Diseases (AREA)
  • Obesity (AREA)
  • Emergency Medicine (AREA)
  • Vascular Medicine (AREA)
  • Oncology (AREA)
  • Molecular Biology (AREA)
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DK02799923T 2001-12-27 2002-12-10 Aroylpyrrolheteroaryl- og methanolforbindelser til behandling af en lidelse i centralnervesystemet DK1458386T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US34376801P 2001-12-27 2001-12-27
PCT/US2002/039487 WO2003057219A1 (en) 2001-12-27 2002-12-10 Aroyl pyrrole heteroeryl and methanols useful for treating a central nervous system disorder

Publications (1)

Publication Number Publication Date
DK1458386T3 true DK1458386T3 (da) 2007-08-13

Family

ID=23347573

Family Applications (1)

Application Number Title Priority Date Filing Date
DK02799923T DK1458386T3 (da) 2001-12-27 2002-12-10 Aroylpyrrolheteroaryl- og methanolforbindelser til behandling af en lidelse i centralnervesystemet

Country Status (14)

Country Link
US (3) US6897319B2 (de)
EP (1) EP1458386B1 (de)
JP (1) JP2005514412A (de)
AR (1) AR038664A1 (de)
AT (1) ATE359783T1 (de)
AU (2) AU2002364545A1 (de)
CY (1) CY1106658T1 (de)
DE (1) DE60219687T2 (de)
DK (1) DK1458386T3 (de)
ES (1) ES2286328T3 (de)
PT (1) PT1458386E (de)
SI (1) SI1458386T1 (de)
TW (1) TWI282277B (de)
WO (2) WO2003057219A1 (de)

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EP1533295A1 (de) * 2003-11-24 2005-05-25 Newron Pharmaceuticals S.p.A. Cyclopentylderivate
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US7598380B2 (en) * 2005-08-03 2009-10-06 Bristol-Myers Squibb Company Method of preparation of azaindole derivatives
EP1963280B1 (de) 2005-12-22 2015-10-28 Newron Pharmaceuticals S.p.A. 2-phenylethylaminoderivate als calcium- und/oder natrium-kanalmodulatoren
AU2008261325B2 (en) 2007-06-15 2012-12-06 Newron Pharmaceuticals S.P.A. Substituted 2- [2- (phenyl) ethylamino] alkaneamide derivatives and their use as sodium and/or calcium channel modulators
GB0804755D0 (en) * 2008-03-14 2008-04-16 Angeletti P Ist Richerche Bio Therapeutic compounds
GB0813873D0 (en) * 2008-07-30 2008-09-03 Univ Dundee Compounds
CN102548964B (zh) * 2009-07-10 2014-09-24 通用医疗公司 不抑制肾上腺皮质类固醇合成的依托咪酯类似物
WO2013000651A1 (en) 2011-06-27 2013-01-03 Newron Pharmaceuticals S.P.A. Fluorinated arylalkylaminocarboxamide derivatives
WO2013106717A1 (en) 2012-01-13 2013-07-18 The General Hospital Corporation Anesthetic compounds and related methods of use
WO2022159980A1 (en) * 2021-01-25 2022-07-28 Athos Therapeutics, Inc. Pharmaceutical compounds and methods of making and using the same

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WO2003057219A1 (en) 2003-07-17
JP2005514412A (ja) 2005-05-19
TWI282277B (en) 2007-06-11
AU2002359856A1 (en) 2003-07-24
US20030181481A1 (en) 2003-09-25
CY1106658T1 (el) 2012-01-25
AU2002359856A8 (en) 2003-07-24
EP1458386A1 (de) 2004-09-22
US6897319B2 (en) 2005-05-24
SI1458386T1 (sl) 2007-08-31
DE60219687D1 (de) 2007-05-31
DE60219687T2 (de) 2007-12-27
EP1458386B1 (de) 2007-04-18
AU2002364545A1 (en) 2003-07-24
ES2286328T3 (es) 2007-12-01
TW200400030A (en) 2004-01-01
PT1458386E (pt) 2007-06-04
WO2003057147A2 (en) 2003-07-17
AR038664A1 (es) 2005-01-26
ATE359783T1 (de) 2007-05-15
WO2003057147A3 (en) 2003-10-23
US20040058980A1 (en) 2004-03-25
US20050148636A1 (en) 2005-07-07

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