DK126198B - Fremgangsmåde til fremstilling af pyrimidinnucleosider eller 6-azapyrimidinnucleosider. - Google Patents

Fremgangsmåde til fremstilling af pyrimidinnucleosider eller 6-azapyrimidinnucleosider.

Info

Publication number
DK126198B
DK126198B DK168870AA DK168870A DK126198B DK 126198 B DK126198 B DK 126198B DK 168870A A DK168870A A DK 168870AA DK 168870 A DK168870 A DK 168870A DK 126198 B DK126198 B DK 126198B
Authority
DK
Denmark
Prior art keywords
nucleosides
preparation
azapyrimidine
pyrimidine
pyrimidine nucleosides
Prior art date
Application number
DK168870AA
Other languages
Danish (da)
English (en)
Inventor
H Vorbrueggen
U Niedballa
Original Assignee
Schering Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from DE19691919307 external-priority patent/DE1919307C/de
Priority claimed from DE19691943428 external-priority patent/DE1943428C3/de
Application filed by Schering Ag filed Critical Schering Ag
Publication of DK126198B publication Critical patent/DK126198B/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/06—Pyrimidine radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/12—Triazine radicals
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
DK168870AA 1969-04-11 1970-04-03 Fremgangsmåde til fremstilling af pyrimidinnucleosider eller 6-azapyrimidinnucleosider. DK126198B (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE19691919307 DE1919307C (de) 1969-04-11 Verfahren zur Herstellung von Nucleo siden
DE19691943428 DE1943428C3 (de) 1969-08-23 1969-08-23 Verfahren zur Herstellung von Pyrimidin- und 6-Azauracilnueleosiden

Publications (1)

Publication Number Publication Date
DK126198B true DK126198B (da) 1973-06-18

Family

ID=25757275

Family Applications (1)

Application Number Title Priority Date Filing Date
DK168870AA DK126198B (da) 1969-04-11 1970-04-03 Fremgangsmåde til fremstilling af pyrimidinnucleosider eller 6-azapyrimidinnucleosider.

Country Status (18)

Country Link
US (1) US3748320A (fi)
JP (1) JPS52955B1 (fi)
AT (1) AT315384B (fi)
BE (1) BE748799A (fi)
CA (1) CA931948A (fi)
CH (1) CH541566A (fi)
DK (1) DK126198B (fi)
ES (1) ES378367A1 (fi)
FI (1) FI54314C (fi)
FR (1) FR2043174A5 (fi)
GB (1) GB1313411A (fi)
IE (1) IE33786B1 (fi)
IL (1) IL34301A (fi)
NL (1) NL166266B (fi)
NO (1) NO126322B (fi)
PL (1) PL93943B1 (fi)
SE (1) SE363830B (fi)
SU (1) SU452961A3 (fi)

Families Citing this family (23)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2066931A2 (en) * 1970-10-30 1971-08-13 Schering Ag 2-thio -6-aza-uridine derivs
JPS4924977A (fi) * 1972-06-30 1974-03-05
US3868361A (en) * 1973-03-12 1975-02-25 Richard L Tolman s-Triazolo{8 2,3-A{9 {0 pryimidine nucleosides
JPS5152183A (ja) * 1974-10-28 1976-05-08 Mitsui Seiyaku Kogyo Kk Nukureoshidoruinoseizoho
JPS5195082A (en) * 1975-02-14 1976-08-20 55 furuoroshichijinno seizoho
DE2508312A1 (de) * 1975-02-24 1976-09-02 Schering Ag Neues verfahren zur herstellung von nucleosiden
JPS51100087A (en) * 1975-02-26 1976-09-03 Mitsui Seiyaku Kogyo Kk 11 * beeta dd arabinofuranoshiru * 55 furuoroshitoshinno seizoho
DE2514275A1 (de) * 1975-03-27 1976-10-14 Schering Ag Verfahren zur herstellung von n- (polysaccharidyl)-stickstoffheterocyclen, insbesondere von pyrimidin- oder purinbasen
GB1531469A (en) * 1975-12-18 1978-11-08 Farmaceutici Italia Daunosamine nucleosides
US4171431A (en) * 1976-08-19 1979-10-16 The Upjohn Company Nucleosides and process
DE2721466A1 (de) * 1977-05-12 1978-11-16 Robugen Gmbh Verfahren zur herstellung von 2'-desoxyribofuranosylnucleosiden
DE2757365A1 (de) * 1977-12-20 1979-06-21 Schering Ag Neues verfahren zur herstellung von nucleosiden
GB1601020A (en) 1978-04-24 1981-10-21 Stichting Grega Vzw 2'-deoxy-5 (2-halogenovinyl)-uridines
US4423212A (en) * 1980-12-18 1983-12-27 The Upjohn Company Nucleosides and process
US4929723A (en) * 1987-07-21 1990-05-29 Ethyl Corporation Process for preparing 2-deoxynucleosides
CA1301166C (en) * 1987-07-21 1992-05-19 John Nicholas Freskos Process for preparing 2-deoxynucleosides
US4914233A (en) * 1988-03-01 1990-04-03 Ethyl Corporation Synthesis of beta-thymidine
JPH0217199A (ja) * 1988-07-05 1990-01-22 Japan Tobacco Inc ２’−デオキシ−β−アデノシンの製造方法
US5134066A (en) * 1989-08-29 1992-07-28 Monsanto Company Improved probes using nucleosides containing 3-dezauracil analogs
CA2091732C (en) * 1992-07-08 1998-07-21 Anica Markovac A process for the preparation of 2-fluoro-9-(2,3,5-tri-o-benzyl-beta-d-arabinofuranosyl) adenine
US5532349A (en) * 1993-07-20 1996-07-02 Mitsui Toatsu Chemicals, Inc. Process for producing 1-(2'-deoxy-β-D-erythro-pentofuranosyl)-5-trifluoromethyluracil derivatives
DE19513330A1 (de) * 1995-04-03 1996-10-10 Schering Ag Neues Verfahren zur Herstellung von Nucleosiden
CN101076535A (zh) * 2004-12-08 2007-11-21 西科尔公司 二氟核苷及其制备方法

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1795357A1 (de) * 1968-09-18 1972-01-05 Schering Ag 2-Thio-pyrimidin-nucleoside

Also Published As

Publication number Publication date
IL34301A (en) 1973-06-29
FI54314B (fi) 1978-07-31
IE33786B1 (en) 1974-10-30
AT315384B (de) 1974-05-27
NO126322B (fi) 1973-01-22
CA931948A (en) 1973-08-14
NL166266B (nl) 1981-02-16
US3748320A (en) 1973-07-24
SE363830B (fi) 1974-02-04
CH541566A (de) 1973-09-15
IE33786L (en) 1970-10-11
ES378367A1 (es) 1972-06-16
IL34301A0 (en) 1970-06-17
PL93943B1 (fi) 1977-07-30
NL7005235A (fi) 1970-10-13
GB1313411A (en) 1973-04-11
FR2043174A5 (fi) 1971-02-12
JPS52955B1 (fi) 1977-01-11
FI54314C (fi) 1978-11-10
BE748799A (fr) 1970-10-12
SU452961A3 (ru) 1974-12-05

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