DK0974598T3 - Hidtil ukendte erythromcinderivater, fremgangsmådetil fremstillingheraf og anvendelse heraf som lægemidler - Google Patents

Hidtil ukendte erythromcinderivater, fremgangsmådetil fremstillingheraf og anvendelse heraf som lægemidler

Info

Publication number
DK0974598T3
DK0974598T3 DK99401706.9T DK99401706T DK0974598T3 DK 0974598 T3 DK0974598 T3 DK 0974598T3 DK 99401706 T DK99401706 T DK 99401706T DK 0974598 T3 DK0974598 T3 DK 0974598T3
Authority
DK
Denmark
Prior art keywords
preparation
pharmaceuticals
erythromycin derivatives
hitherto unknown
erythromycin
Prior art date
Application number
DK99401706.9T
Other languages
Danish (da)
English (en)
Inventor
Giuseppe Gigliotti
Alexis Denis
Original Assignee
Aventis Pharma Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from FR9808795A external-priority patent/FR2780977B1/fr
Priority claimed from FR9905245A external-priority patent/FR2792637B1/fr
Application filed by Aventis Pharma Sa filed Critical Aventis Pharma Sa
Application granted granted Critical
Publication of DK0974598T3 publication Critical patent/DK0974598T3/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08Hetero rings containing eight or more ring members, e.g. erythromycins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Communicable Diseases (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
DK99401706.9T 1998-07-09 1999-07-08 Hidtil ukendte erythromcinderivater, fremgangsmådetil fremstillingheraf og anvendelse heraf som lægemidler DK0974598T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR9808795A FR2780977B1 (fr) 1998-07-09 1998-07-09 Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments
FR9905245A FR2792637B1 (fr) 1999-04-26 1999-04-26 Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments

Publications (1)

Publication Number Publication Date
DK0974598T3 true DK0974598T3 (da) 2011-12-19

Family

ID=26234434

Family Applications (1)

Application Number Title Priority Date Filing Date
DK99401706.9T DK0974598T3 (da) 1998-07-09 1999-07-08 Hidtil ukendte erythromcinderivater, fremgangsmådetil fremstillingheraf og anvendelse heraf som lægemidler

Country Status (8)

Country Link
US (1) US6433151B1 (https=)
EP (1) EP0974598B1 (https=)
JP (1) JP4573925B2 (https=)
AT (1) ATE521619T1 (https=)
CY (1) CY1112087T1 (https=)
DK (1) DK0974598T3 (https=)
ES (1) ES2372156T3 (https=)
PT (1) PT974598E (https=)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TR200102129T2 (tr) * 1998-12-10 2002-01-21 Pfizer Products Inc. Karbamat ve karbazat ketolid antibiyotikleri.
JP2008508322A (ja) * 2004-07-28 2008-03-21 ランバクシー ラボラトリーズ リミテッド 抗菌剤としてのケトライド誘導体
US20080318878A1 (en) * 2004-09-27 2008-12-25 Biswajit Das Antibacterial Agents
EP1807439A2 (en) * 2004-10-25 2007-07-18 Ranbaxy Laboratories Limited Ketolide derivatives as antibacterial agents
UA85937C2 (uk) * 2004-12-21 2009-03-10 Пфайзер Продактс Інк. Макроліди
WO2007054904A2 (en) * 2005-11-08 2007-05-18 Ranbaxy Laboratories Limited Macrolides as anti-inflammatory agents
US20090075916A1 (en) * 2005-11-23 2009-03-19 Upadhyay Dilip J Use of Macrolide Derivatives for Treating Acne
EP1960413A2 (en) * 2005-11-23 2008-08-27 Ranbaxy Laboratories Limited Macrolides derivatives as antibacterial agents
WO2007060518A2 (en) * 2005-11-23 2007-05-31 Ranbaxy Laboratories Limited Ketolide derivatives as antibacterial agents
EA017878B1 (ru) * 2006-12-12 2013-03-29 Замбон С.П.А. Макролидные соединения, обладающие противовоспалительной активностью
AU2019403048B2 (en) * 2018-12-17 2025-01-23 Lunella Biotech, Inc. Triple combination therapies for targeting mitochondria and killing cancer stem cells

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3725385A (en) * 1970-11-02 1973-04-03 Abbott Lab Process for the demethylation of 3-amino macrolides
IL114589A (en) * 1990-11-21 1999-12-22 Roussel Uclaf Intermediates for the preparation of erythromycin derivatives
US5527780A (en) * 1992-11-05 1996-06-18 Roussel Uclaf Erythromycin derivatives
FR2719587B1 (fr) * 1994-05-03 1996-07-12 Roussel Uclaf Nouveaux dérivés de l'érythromycine, leur procédé de préparation et leur application comme médicaments.
KR19990067492A (ko) * 1995-11-08 1999-08-25 스티븐 에프. 웨인스톡 트리사이클릭 에리트로마이신 유도체
FR2742757B1 (fr) * 1995-12-22 1998-01-30 Roussel Uclaf Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments
FR2745290B1 (fr) * 1996-02-28 1998-04-03 Roussel Uclaf Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments
DE69733723T2 (de) * 1996-09-04 2006-04-20 Abbott Laboratories, Abbott Park 6-o-Substituierte Ketoliden mit antibakteriellen Wirkung
DK1025114T3 (da) * 1997-09-30 2004-07-05 Abbott Lab 3'-N-modificerede 6-O-substituerede erythromycin-ketolidderivater med antibakteriel aktivitet

Also Published As

Publication number Publication date
EP0974598A2 (fr) 2000-01-26
CY1112087T1 (el) 2015-11-04
ES2372156T3 (es) 2012-01-16
PT974598E (pt) 2011-11-23
JP2000026494A (ja) 2000-01-25
US6433151B1 (en) 2002-08-13
JP4573925B2 (ja) 2010-11-04
ATE521619T1 (de) 2011-09-15
EP0974598A3 (fr) 2003-12-17
EP0974598B1 (fr) 2011-08-24

Similar Documents

Publication Publication Date Title
CY1112087T1 (el) Νεα παραγωγα της ερυθρομυκινης, η διαδικασια της παρασκευης τους και η εφαρμογη τους ως φαρμακευτικα προϊοντα
HUP9902576A1 (hu) Új eritromicinszármazékok, eljárás előállításukra és alkalmazásuk gyógyászati készítményekben
FR2518088B1 (fr) Nouveaux derives d'aminoacides, et leur application therapeutique
NO982606D0 (no) Naftylsubstituerte benzimidazolderivater som antikoagulanter
ES2085130T3 (es) Nuevos derivados de la eritromicina, su procedimiento de preparacion, y su aplicacion como medicamentos.
NO970512L (no) Nye heteroaryl-oksazolidinoner
NO970175L (no) Pyrido-annellerte tienyl- og furanyl-oksazolidinoner
TR199902593T2 (xx) �kame edilmi� fenil t�revleri, bunlar�n haz�rlanmas� ve kullan�m�.
TR199501253A2 (tr) Amino(tio) eter türevleri.
DE69813605D1 (de) Benzofuranderivate
TR200000586T2 (tr) Farmasötik maddelerin oral yoldan biyolojik kullanışlılığının arttırılması için bir yöntem, bileşimler ve kitler.
SE7704783L (sv) Medel for separationsendamal och forfarande for dess framstellning
TR199700206A2 (xx) Floralkil- ve floralkoksi ikame edilmi� heterosiklik bradikinin-antagonistleri, bunlar�n imal edilmesine mahsus usul ve bunlar�n kullan�lmalar�.
NO20001198L (no) Pyrrolopyrrolondervater som inhibitorer av nøytrofil elastase
BRPI0210746B8 (pt) derivados de 6-'2-(fosfonometóxi)alcóxi-pirimidina e seu método de preparação
IT1140209B (it) Reagenti per immunoluorescenza e metodo per la loro preparazione
ES528874A0 (es) Procedimiento para la preparacion de nuevos compuestos carboxamidicos de pirrol ortocondensado.
AU553927B2 (en) Oxazolo- thiazolo- imidazolo (5,4-b) pyridines
NO994104L (no) 5-hydroksymetyl-2-aminotetraliner i form av kardiovaskulaere midler
NO985685D0 (no) Dibenzo-oksazepin- og -dioksazepin-derivater og deres anvendelse som anti-tumormidler
ES2069669T3 (es) Compuestos biocidas.
PT78410A (fr) Procede de preparation de polymethylene imines disubstituees
ATE126799T1 (de) Derivate von methylpiperazinoazepin, verfahren zu ihrer herstellung und verwendung.
FR2555576B1 (fr) Derives de n-(methoxyphenacyl)-amine, utilisation notamment en therapeutique et procede de preparation
FI902764A7 (fi) N-(3-(((aryyli)amino)sulfonyyli)-1H-1,2,4,-triatsol-5-yyli)amiinien valmistus