DK0972762T3 - Hidtil ukendte strukturelle analoger af vitamin D - Google Patents

Hidtil ukendte strukturelle analoger af vitamin D

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Publication number
DK0972762T3
DK0972762T3 DK99203513T DK99203513T DK0972762T3 DK 0972762 T3 DK0972762 T3 DK 0972762T3 DK 99203513 T DK99203513 T DK 99203513T DK 99203513 T DK99203513 T DK 99203513T DK 0972762 T3 DK0972762 T3 DK 0972762T3
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DK
Denmark
Prior art keywords
vitamin
ring
hitherto unknown
structural analogues
analogue
Prior art date
Application number
DK99203513T
Other languages
Danish (da)
English (en)
Inventor
Roger Bouillon
Maurits Vandewalle
Clercq Pierre Jean De
Original Assignee
Theramex
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Theramex filed Critical Theramex
Application granted granted Critical
Publication of DK0972762T3 publication Critical patent/DK0972762T3/da

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    • C07C47/00—Compounds having —CHO groups
    • C07C47/02—Saturated compounds having —CHO groups bound to acyclic carbon atoms or to hydrogen
    • C07C47/198—Saturated compounds having —CHO groups bound to acyclic carbon atoms or to hydrogen containing ether groups, groups, groups, or groups
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    • A61P13/00—Drugs for disorders of the urinary system
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    • C07C35/00—Compounds having at least one hydroxy or O-metal group bound to a carbon atom of a ring other than a six-membered aromatic ring
    • C07C35/22—Compounds having at least one hydroxy or O-metal group bound to a carbon atom of a ring other than a six-membered aromatic ring polycyclic, at least one hydroxy group bound to a condensed ring system
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    • C07C35/22—Compounds having at least one hydroxy or O-metal group bound to a carbon atom of a ring other than a six-membered aromatic ring polycyclic, at least one hydroxy group bound to a condensed ring system
    • C07C35/23—Compounds having at least one hydroxy or O-metal group bound to a carbon atom of a ring other than a six-membered aromatic ring polycyclic, at least one hydroxy group bound to a condensed ring system with hydroxy on a condensed ring system having two rings
    • C07C35/27—Compounds having at least one hydroxy or O-metal group bound to a carbon atom of a ring other than a six-membered aromatic ring polycyclic, at least one hydroxy group bound to a condensed ring system with hydroxy on a condensed ring system having two rings the condensed ring system containing six carbon atoms
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    • C07C47/19—Saturated compounds having —CHO groups bound to acyclic carbon atoms or to hydrogen containing hydroxy groups
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    • C07C47/37—Saturated compounds having —CHO groups bound to carbon atoms of rings other than six—membered aromatic rings containing ether groups, groups, groups, or groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C49/00—Ketones; Ketenes; Dimeric ketenes; Ketonic chelates
    • C07C49/20—Unsaturated compounds containing keto groups bound to acyclic carbon atoms
    • C07C49/24—Unsaturated compounds containing keto groups bound to acyclic carbon atoms containing hydroxy groups
    • C07C49/242—Unsaturated compounds containing keto groups bound to acyclic carbon atoms containing hydroxy groups containing rings other than six-membered aromatic rings
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    • C07C49/00—Ketones; Ketenes; Dimeric ketenes; Ketonic chelates
    • C07C49/385—Saturated compounds containing a keto group being part of a ring
    • C07C49/517—Saturated compounds containing a keto group being part of a ring containing ether groups, groups, groups, or groups
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    • C07C49/587—Unsaturated compounds containing a keto groups being part of a ring
    • C07C49/687—Unsaturated compounds containing a keto groups being part of a ring containing halogen
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    • C07C49/587—Unsaturated compounds containing a keto groups being part of a ring
    • C07C49/703—Unsaturated compounds containing a keto groups being part of a ring containing hydroxy groups
    • C07C49/743—Unsaturated compounds containing a keto groups being part of a ring containing hydroxy groups having unsaturation outside the rings, e.g. humulones, lupulones
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    • C07C49/753—Unsaturated compounds containing a keto groups being part of a ring containing ether groups, groups, groups, or groups
    • C07C49/755—Unsaturated compounds containing a keto groups being part of a ring containing ether groups, groups, groups, or groups a keto group being part of a condensed ring system with two or three rings, at least one ring being a six-membered aromatic ring
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    • C07C59/01—Saturated compounds having only one carboxyl group and containing hydroxy or O-metal groups

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  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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  • Diabetes (AREA)
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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
DK99203513T 1993-07-09 1994-07-07 Hidtil ukendte strukturelle analoger af vitamin D DK0972762T3 (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP93202037 1993-07-09

Publications (1)

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DK0972762T3 true DK0972762T3 (da) 2004-02-09

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ID=8213977

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DK94924749T DK0707566T3 (da) 1993-07-09 1994-07-07 Hidtil ukendte strukturelle analoger til vitamin D
DK99203513T DK0972762T3 (da) 1993-07-09 1994-07-07 Hidtil ukendte strukturelle analoger af vitamin D

Family Applications Before (1)

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Country Status (16)

Country Link
US (2) US6017907A (el)
EP (2) EP0707566B1 (el)
JP (2) JP4235256B2 (el)
CN (1) CN1103755C (el)
AT (2) ATE251133T1 (el)
AU (1) AU699200B2 (el)
CA (1) CA2166898C (el)
DE (2) DE69433220T2 (el)
DK (2) DK0707566T3 (el)
ES (2) ES2209327T3 (el)
GR (1) GR3033856T3 (el)
NO (1) NO314142B1 (el)
NZ (1) NZ271332A (el)
PT (2) PT707566E (el)
RU (1) RU2153491C2 (el)
WO (1) WO1995001960A1 (el)

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US5919986A (en) * 1997-10-17 1999-07-06 Hoffmann-La Roche Inc. D-homo vitamin D3 derivatives
DE69939106D1 (de) * 1998-02-24 2008-08-28 Chugai Pharmaceutical Co Ltd Verfahren zur Herstellung von ED-71
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ES2147238T3 (es) 2000-09-01
CA2166898C (en) 2004-09-07
EP0707566A1 (en) 1996-04-24
ATE191712T1 (de) 2000-04-15
NO960099L (no) 1996-03-08
PT707566E (pt) 2000-09-29
DE69423966D1 (de) 2000-05-18
RU2153491C2 (ru) 2000-07-27
GR3033856T3 (en) 2000-10-31
JP4312183B2 (ja) 2009-08-12
AU7492794A (en) 1995-02-06
CN1130899A (zh) 1996-09-11
WO1995001960A1 (en) 1995-01-19
JP4235256B2 (ja) 2009-03-11
PT972762E (pt) 2004-02-27
US6548715B1 (en) 2003-04-15
DE69423966T2 (de) 2000-11-16
NO314142B1 (no) 2003-02-03
NO960099D0 (no) 1996-01-09
EP0972762A2 (en) 2000-01-19
EP0707566B1 (en) 2000-04-12
DE69433220D1 (de) 2003-11-06
EP0972762A3 (en) 2000-02-23
DE69433220T2 (de) 2004-08-19
DK0707566T3 (da) 2000-09-04
CA2166898A1 (en) 1995-01-19
AU699200B2 (en) 1998-11-26
JPH09500117A (ja) 1997-01-07
ATE251133T1 (de) 2003-10-15
CN1103755C (zh) 2003-03-26
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US6017907A (en) 2000-01-25
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