DK0972762T3 - Hidtil ukendte strukturelle analoger af vitamin D - Google Patents

Hidtil ukendte strukturelle analoger af vitamin D

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Publication number
DK0972762T3
DK0972762T3 DK99203513T DK99203513T DK0972762T3 DK 0972762 T3 DK0972762 T3 DK 0972762T3 DK 99203513 T DK99203513 T DK 99203513T DK 99203513 T DK99203513 T DK 99203513T DK 0972762 T3 DK0972762 T3 DK 0972762T3
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DK
Denmark
Prior art keywords
vitamin
ring
hitherto unknown
structural analogues
analogue
Prior art date
Application number
DK99203513T
Other languages
English (en)
Inventor
Roger Bouillon
Maurits Vandewalle
Clercq Pierre Jean De
Original Assignee
Theramex
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Theramex filed Critical Theramex
Application granted granted Critical
Publication of DK0972762T3 publication Critical patent/DK0972762T3/da

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    • C07C47/02—Saturated compounds having —CHO groups bound to acyclic carbon atoms or to hydrogen
    • C07C47/198—Saturated compounds having —CHO groups bound to acyclic carbon atoms or to hydrogen containing ether groups, groups, groups, or groups
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    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/12—Drugs for disorders of the urinary system of the kidneys
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
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    • A61P17/00—Drugs for dermatological disorders
    • A61P17/02—Drugs for dermatological disorders for treating wounds, ulcers, burns, scars, keloids, or the like
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    • C07C35/00—Compounds having at least one hydroxy or O-metal group bound to a carbon atom of a ring other than a six-membered aromatic ring
    • C07C35/22—Compounds having at least one hydroxy or O-metal group bound to a carbon atom of a ring other than a six-membered aromatic ring polycyclic, at least one hydroxy group bound to a condensed ring system
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    • C07C35/00—Compounds having at least one hydroxy or O-metal group bound to a carbon atom of a ring other than a six-membered aromatic ring
    • C07C35/22—Compounds having at least one hydroxy or O-metal group bound to a carbon atom of a ring other than a six-membered aromatic ring polycyclic, at least one hydroxy group bound to a condensed ring system
    • C07C35/23—Compounds having at least one hydroxy or O-metal group bound to a carbon atom of a ring other than a six-membered aromatic ring polycyclic, at least one hydroxy group bound to a condensed ring system with hydroxy on a condensed ring system having two rings
    • C07C35/27—Compounds having at least one hydroxy or O-metal group bound to a carbon atom of a ring other than a six-membered aromatic ring polycyclic, at least one hydroxy group bound to a condensed ring system with hydroxy on a condensed ring system having two rings the condensed ring system containing six carbon atoms
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    • C07C401/00—Irradiation products of cholesterol or its derivatives; Vitamin D derivatives, 9,10-seco cyclopenta[a]phenanthrene or analogues obtained by chemical preparation without irradiation
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    • C07C47/02—Saturated compounds having —CHO groups bound to acyclic carbon atoms or to hydrogen
    • C07C47/19—Saturated compounds having —CHO groups bound to acyclic carbon atoms or to hydrogen containing hydroxy groups
    • C07C47/192—Saturated compounds having —CHO groups bound to acyclic carbon atoms or to hydrogen containing hydroxy groups containing rings
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    • C07C47/28—Saturated compounds having —CHO groups bound to carbon atoms of rings other than six—membered aromatic rings
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    • C07C47/00—Compounds having —CHO groups
    • C07C47/28—Saturated compounds having —CHO groups bound to carbon atoms of rings other than six—membered aromatic rings
    • C07C47/37—Saturated compounds having —CHO groups bound to carbon atoms of rings other than six—membered aromatic rings containing ether groups, groups, groups, or groups
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    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C49/00—Ketones; Ketenes; Dimeric ketenes; Ketonic chelates
    • C07C49/20—Unsaturated compounds containing keto groups bound to acyclic carbon atoms
    • C07C49/24—Unsaturated compounds containing keto groups bound to acyclic carbon atoms containing hydroxy groups
    • C07C49/242—Unsaturated compounds containing keto groups bound to acyclic carbon atoms containing hydroxy groups containing rings other than six-membered aromatic rings
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    • C07C49/00—Ketones; Ketenes; Dimeric ketenes; Ketonic chelates
    • C07C49/385—Saturated compounds containing a keto group being part of a ring
    • C07C49/517—Saturated compounds containing a keto group being part of a ring containing ether groups, groups, groups, or groups
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    • C07C49/587—Unsaturated compounds containing a keto groups being part of a ring
    • C07C49/703—Unsaturated compounds containing a keto groups being part of a ring containing hydroxy groups
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    • C07C49/587—Unsaturated compounds containing a keto groups being part of a ring
    • C07C49/753—Unsaturated compounds containing a keto groups being part of a ring containing ether groups, groups, groups, or groups
    • C07C49/755—Unsaturated compounds containing a keto groups being part of a ring containing ether groups, groups, groups, or groups a keto group being part of a condensed ring system with two or three rings, at least one ring being a six-membered aromatic ring
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    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C57/00—Unsaturated compounds having carboxyl groups bound to acyclic carbon atoms
    • C07C57/26—Unsaturated compounds having carboxyl groups bound to acyclic carbon atoms containing rings other than six-membered aromatic rings
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    • C07C59/00—Compounds having carboxyl groups bound to acyclic carbon atoms and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups
    • C07C59/01—Saturated compounds having only one carboxyl group and containing hydroxy or O-metal groups
DK99203513T 1993-07-09 1994-07-07 Hidtil ukendte strukturelle analoger af vitamin D DK0972762T3 (da)

Applications Claiming Priority (1)

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EP93202037 1993-07-09

Publications (1)

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DK0972762T3 true DK0972762T3 (da) 2004-02-09

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DK99203513T DK0972762T3 (da) 1993-07-09 1994-07-07 Hidtil ukendte strukturelle analoger af vitamin D
DK94924749T DK0707566T3 (da) 1993-07-09 1994-07-07 Hidtil ukendte strukturelle analoger til vitamin D

Family Applications After (1)

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Country Status (16)

Country Link
US (2) US6017907A (da)
EP (2) EP0707566B1 (da)
JP (2) JP4235256B2 (da)
CN (1) CN1103755C (da)
AT (2) ATE251133T1 (da)
AU (1) AU699200B2 (da)
CA (1) CA2166898C (da)
DE (2) DE69423966T2 (da)
DK (2) DK0972762T3 (da)
ES (2) ES2147238T3 (da)
GR (1) GR3033856T3 (da)
NO (1) NO314142B1 (da)
NZ (1) NZ271332A (da)
PT (2) PT972762E (da)
RU (1) RU2153491C2 (da)
WO (1) WO1995001960A1 (da)

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ATE191712T1 (de) 2000-04-15
JP2006001944A (ja) 2006-01-05
JP4312183B2 (ja) 2009-08-12
DK0707566T3 (da) 2000-09-04
EP0707566A1 (en) 1996-04-24
DE69433220T2 (de) 2004-08-19
CA2166898C (en) 2004-09-07
JPH09500117A (ja) 1997-01-07
CA2166898A1 (en) 1995-01-19
EP0972762B1 (en) 2003-10-01
CN1130899A (zh) 1996-09-11
ATE251133T1 (de) 2003-10-15
EP0972762A2 (en) 2000-01-19
WO1995001960A1 (en) 1995-01-19
PT972762E (pt) 2004-02-27
DE69423966D1 (de) 2000-05-18
NZ271332A (en) 2001-03-30
EP0707566B1 (en) 2000-04-12
NO960099L (no) 1996-03-08
AU699200B2 (en) 1998-11-26
NO314142B1 (no) 2003-02-03
US6548715B1 (en) 2003-04-15
EP0972762A3 (en) 2000-02-23
US6017907A (en) 2000-01-25
RU2153491C2 (ru) 2000-07-27
CN1103755C (zh) 2003-03-26
ES2209327T3 (es) 2004-06-16
DE69423966T2 (de) 2000-11-16
NO960099D0 (no) 1996-01-09
DE69433220D1 (de) 2003-11-06
AU7492794A (en) 1995-02-06
GR3033856T3 (en) 2000-10-31
PT707566E (pt) 2000-09-29
ES2147238T3 (es) 2000-09-01

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