DK0956287T3 - 3-Aryl-2-(1-substituerede-4-piperidinyl)-1(1-di)oxo-3H-benzo[D]-isothiazol-derivater, deres fremstilling og deres anvendelse som modulatorer af neurotransmitterfunktion - Google Patents
3-Aryl-2-(1-substituerede-4-piperidinyl)-1(1-di)oxo-3H-benzo[D]-isothiazol-derivater, deres fremstilling og deres anvendelse som modulatorer af neurotransmitterfunktionInfo
- Publication number
- DK0956287T3 DK0956287T3 DK97950636T DK97950636T DK0956287T3 DK 0956287 T3 DK0956287 T3 DK 0956287T3 DK 97950636 T DK97950636 T DK 97950636T DK 97950636 T DK97950636 T DK 97950636T DK 0956287 T3 DK0956287 T3 DK 0956287T3
- Authority
- DK
- Denmark
- Prior art keywords
- piperidinyl
- benzo
- modulators
- oxo
- aryl
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
- A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
- A61K31/454—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. pimozide, domperidone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Epidemiology (AREA)
- Pain & Pain Management (AREA)
- Psychiatry (AREA)
- Psychology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US77486696A | 1996-12-23 | 1996-12-23 | |
| PCT/US1997/021178 WO1998028295A1 (en) | 1996-12-23 | 1997-11-13 | 3-aryl-2-(1-substituted-4-piperidinyl)-1(1-di)oxo-3h-benzo[d]-isothiazole derivatives, their preparation and their use as modulators of neurotransmitter function |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DK0956287T3 true DK0956287T3 (da) | 2003-11-24 |
Family
ID=25102528
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK97950636T DK0956287T3 (da) | 1996-12-23 | 1997-11-13 | 3-Aryl-2-(1-substituerede-4-piperidinyl)-1(1-di)oxo-3H-benzo[D]-isothiazol-derivater, deres fremstilling og deres anvendelse som modulatorer af neurotransmitterfunktion |
Country Status (17)
| Country | Link |
|---|---|
| EP (1) | EP0956287B1 (de) |
| JP (1) | JP3282827B2 (de) |
| KR (1) | KR20000062283A (de) |
| AR (1) | AR009440A1 (de) |
| AT (1) | ATE247111T1 (de) |
| AU (1) | AU716689B2 (de) |
| BR (1) | BR9714432A (de) |
| CA (1) | CA2273181C (de) |
| DE (1) | DE69724148T2 (de) |
| DK (1) | DK0956287T3 (de) |
| ES (1) | ES2200205T3 (de) |
| HU (1) | HUP9904071A3 (de) |
| IL (1) | IL130605A0 (de) |
| NO (1) | NO993085L (de) |
| PT (1) | PT956287E (de) |
| WO (1) | WO1998028295A1 (de) |
| ZA (1) | ZA9711337B (de) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IT1393351B1 (it) * | 2009-03-16 | 2012-04-20 | Eos Ethical Oncology Science Spa In Forma Abbreviata Eos Spa | Procedimento per la preparazione della 6-(7-((1-amminociclopropil)metossi)-6-metossichinolin-4-ilossi)-n-metil-1-naftammide e suoi intermedi di sintesi |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE2509797C2 (de) * | 1975-03-06 | 1985-07-18 | Dr. Karl Thomae Gmbh, 7950 Biberach | Phthalimidine, deren physiologisch verträgliche Säureadditionssalze, Verfahren zu ihrer Herstellung und diese Verbindungen enthaltende Arzneimittel |
| AT345806B (de) * | 1975-03-06 | 1978-10-10 | Thomae Gmbh Dr K | Verfahren zur herstellung neuer substituierter arylalkylamine und deren salze |
| EP0429341A3 (en) * | 1989-11-20 | 1991-11-13 | Rhone-Poulenc Sante | Heterocyclic derivatives, their preparation and pharmaceuticals containing them |
| FR2662696A2 (fr) * | 1989-12-13 | 1991-12-06 | Rhone Poulenc Sante | Antagonistes de la serotonine, leur preparation et medicaments les contenant. |
| US5567718A (en) * | 1994-08-11 | 1996-10-22 | Hoechst Marion Roussel Inc. | 2,3-dihydro-1h-isoindole derivatives and their use as serotonin reuptake inhibitors |
-
1997
- 1997-11-13 AU AU53588/98A patent/AU716689B2/en not_active Ceased
- 1997-11-13 WO PCT/US1997/021178 patent/WO1998028295A1/en not_active Application Discontinuation
- 1997-11-13 CA CA002273181A patent/CA2273181C/en not_active Expired - Fee Related
- 1997-11-13 KR KR1019997005678A patent/KR20000062283A/ko not_active Application Discontinuation
- 1997-11-13 ES ES97950636T patent/ES2200205T3/es not_active Expired - Lifetime
- 1997-11-13 DK DK97950636T patent/DK0956287T3/da active
- 1997-11-13 EP EP97950636A patent/EP0956287B1/de not_active Expired - Lifetime
- 1997-11-13 IL IL13060597A patent/IL130605A0/xx unknown
- 1997-11-13 AT AT97950636T patent/ATE247111T1/de not_active IP Right Cessation
- 1997-11-13 PT PT97950636T patent/PT956287E/pt unknown
- 1997-11-13 JP JP52874198A patent/JP3282827B2/ja not_active Expired - Fee Related
- 1997-11-13 BR BR9714432-0A patent/BR9714432A/pt not_active Application Discontinuation
- 1997-11-13 DE DE69724148T patent/DE69724148T2/de not_active Expired - Fee Related
- 1997-11-13 HU HU9904071A patent/HUP9904071A3/hu unknown
- 1997-12-17 ZA ZA9711337A patent/ZA9711337B/xx unknown
- 1997-12-19 AR ARP970106005A patent/AR009440A1/es unknown
-
1999
- 1999-06-22 NO NO993085A patent/NO993085L/no not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| PT956287E (pt) | 2003-11-28 |
| DE69724148T2 (de) | 2004-06-09 |
| EP0956287B1 (de) | 2003-08-13 |
| HUP9904071A3 (en) | 2000-07-28 |
| AU716689B2 (en) | 2000-03-02 |
| AR009440A1 (es) | 2000-04-12 |
| CA2273181C (en) | 2004-01-20 |
| IL130605A0 (en) | 2000-06-01 |
| WO1998028295A1 (en) | 1998-07-02 |
| ATE247111T1 (de) | 2003-08-15 |
| KR20000062283A (ko) | 2000-10-25 |
| HUP9904071A2 (hu) | 2000-05-28 |
| EP0956287A1 (de) | 1999-11-17 |
| ZA9711337B (en) | 1998-06-23 |
| ES2200205T3 (es) | 2004-03-01 |
| NO993085L (no) | 1999-08-20 |
| AU5358898A (en) | 1998-07-17 |
| CA2273181A1 (en) | 1998-07-02 |
| JP2001520641A (ja) | 2001-10-30 |
| JP3282827B2 (ja) | 2002-05-20 |
| NO993085D0 (no) | 1999-06-22 |
| DE69724148D1 (de) | 2003-09-18 |
| BR9714432A (pt) | 2000-05-02 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| NO20001102D0 (no) | 2,3-diaryl-pyrazolo[1,5-B]pyridazinderivater, deres fremstilling og anvendelse som syklo-oksygenase 2 (COX-2) inhibitorer | |
| DK1006110T3 (da) | Derivater af acylpiperazinylpyrimidiner, fremstilling deraf og anvendelse som lægemidler | |
| DK0810218T3 (da) | 6-benzyl-2H-pyridazin-3-onderivater samt fremstilling og anvendelsen deraf som inhibitorer af prostaglandin-G/H-syntase I og II (COX I og COX II) | |
| NO993003D0 (no) | Sulfonamid-derivater, fremgangsmÕte for deres fremstilling og deres anvendelse som medikamenter | |
| NO20011503D0 (no) | Indeno-, nafto- og benzocyklohepta-dihydrotiazolderivater, deres fremstilling og anvendelse som anorektiske legemidler | |
| NO20011956D0 (no) | Substituerte fenylderivater, deres fremstilling og anvendelse | |
| EE200200138A (et) | Kinolüülpropüülpiperidiini derivaadid, nende valmistamine ja neid sisaldavad kompositsioonid | |
| DK0906292T3 (da) | Triazolylmercaptider og deres anvendelse som mikrobicider | |
| DK1206457T3 (da) | Biaryl-oxa(thia)zolderivater og deres anvendelse som modulatorer PPAP'ER | |
| DK1288206T3 (da) | Substituerede benzensulfonamidderivater som prolægemidler af COX-2-inhibitorer | |
| NO991815D0 (no) | Oksadiazoler, fremgangsmÕter for deres fremstilling og deres anvendelse som medikamenter | |
| DK0888297T3 (da) | N-arylsulfiliminforbindelser og deres anvendelse som katalysatorer ved fremstillingen af N-arylarylsulfonamidforbindelser | |
| NO20006138D0 (no) | Substituerte indolinoner, fremstilling og anvendelse derav som medikamenter | |
| NO20005146L (no) | Tienylazolylalkoksyetanaminer, deres fremstilling og deres anvendelse som medikamenter | |
| NO962952D0 (no) | 1,2,4-oksadiazolderivater og deres anvendelse som parasitticider for dyr | |
| NO20006460D0 (no) | 4, 5, 6 og 7-Indol og indolinderivater, deres fremstilling og anvendelse | |
| NO994510D0 (no) | Substituerte isokinolin-derivater og deres anvendelse som antikonvulsanter | |
| DK0879058T3 (da) | Blandinger hidrørende fra frø af Eugénia Jambolana Lamarck, fremstilling af disse blandinger og visse af deres bestanddele samt anvendelse af disse som lægemidler | |
| DK0911311T3 (da) | Fremstilling af lycopenmetabolitter | |
| NO955305L (no) | Optisk aktive benzotiepinderivater, deres fremstilling og anvendelse | |
| NO995513L (no) | N-triazolyl-2-indolkarboksamider og deres anvendelse som CCK- | |
| DK0795547T3 (da) | (Aminoalkyl- og acylaminoalkyl-oxy)benzyloxyquinoliner, fremgangsmåde til deres fremstilling og deres anvendelse som bradyk | |
| DK1015433T3 (da) | Substituerede 1,2,3,4,5,6-hexahydro-2,6-methano-3-benzazocin-10-oler, fremgangsmåder til fremstilling af disse og deres anvendelse som lægemidler | |
| NO20001934D0 (no) | 3-Substituerte tetrahydropyridopyrimidinon-derivater, deres fremstilling og anvendelse | |
| DK0951561T3 (da) | Enzymatiske fremgangsmåder til fremstilling af (S)-cyanhydriner |