DK0804417T3 - Fremgangsmåde til racemisering til brug ved fremstilling af levobupivacain og beslægtede piperidincarboxanilid bedøvelsesmidler - Google Patents

Fremgangsmåde til racemisering til brug ved fremstilling af levobupivacain og beslægtede piperidincarboxanilid bedøvelsesmidler

Info

Publication number
DK0804417T3
DK0804417T3 DK96900349T DK96900349T DK0804417T3 DK 0804417 T3 DK0804417 T3 DK 0804417T3 DK 96900349 T DK96900349 T DK 96900349T DK 96900349 T DK96900349 T DK 96900349T DK 0804417 T3 DK0804417 T3 DK 0804417T3
Authority
DK
Denmark
Prior art keywords
levobupivacaine
racemization
anesthetics
preparation
carboxanilide
Prior art date
Application number
DK96900349T
Other languages
Danish (da)
English (en)
Inventor
Ulrich Conrad Chiroscienc Dyer
Marianne Chiroscience Langston
Martin Chiroscience Limi Woods
Original Assignee
Darwin Discovery Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Darwin Discovery Ltd filed Critical Darwin Discovery Ltd
Application granted granted Critical
Publication of DK0804417T3 publication Critical patent/DK0804417T3/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D211/00Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/60Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Hydrogenated Pyridines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Rolling Contact Bearings (AREA)
  • Optical Head (AREA)
  • Beans For Foods Or Fodder (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Peptides Or Proteins (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
DK96900349T 1995-01-18 1996-01-12 Fremgangsmåde til racemisering til brug ved fremstilling af levobupivacain og beslægtede piperidincarboxanilid bedøvelsesmidler DK0804417T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB9501071.6A GB9501071D0 (en) 1995-01-18 1995-01-18 Racemisation
PCT/GB1996/000067 WO1996022281A1 (en) 1995-01-18 1996-01-12 Racemisation process for use in the manufacture of levobupivacaine and related piperidinecarboxanilide anaesthetic agents

Publications (1)

Publication Number Publication Date
DK0804417T3 true DK0804417T3 (da) 2003-10-06

Family

ID=10768271

Family Applications (1)

Application Number Title Priority Date Filing Date
DK96900349T DK0804417T3 (da) 1995-01-18 1996-01-12 Fremgangsmåde til racemisering til brug ved fremstilling af levobupivacain og beslægtede piperidincarboxanilid bedøvelsesmidler

Country Status (20)

Country Link
EP (1) EP0804417B1 (ja)
JP (1) JP4015696B2 (ja)
KR (1) KR100404390B1 (ja)
CN (1) CN1172912C (ja)
AT (1) ATE242214T1 (ja)
AU (1) AU701221B2 (ja)
BR (1) BR9606821A (ja)
CA (1) CA2208522C (ja)
DE (1) DE69628540T2 (ja)
DK (1) DK0804417T3 (ja)
ES (1) ES2201166T3 (ja)
FI (1) FI117437B (ja)
GB (1) GB9501071D0 (ja)
HU (1) HU227426B1 (ja)
MX (1) MX9705428A (ja)
NO (1) NO308843B1 (ja)
PL (1) PL184091B1 (ja)
PT (1) PT804417E (ja)
WO (1) WO1996022281A1 (ja)
ZA (1) ZA96403B (ja)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BR0002246A (pt) 2000-04-06 2003-04-15 Cristalia Prod Quimicos Farm Processo de obtenção dos enantiÈmeros da bupivacaìna racêmica, processo de obtenção de composições farmacêuticas a base de levobupivacaìna: composições farmacêuticas a base de levobupivacaìna formuladas nas formas básicas ou sais farmaceuticamente aceitáveis e utilização das composições farmacêuticas a base de levobupivacaìna formuladas nas formas básicas ou sais farmaceuticamente aceitáveis
US20040001889A1 (en) 2002-06-25 2004-01-01 Guohua Chen Short duration depot formulations
CN101797221B (zh) 2002-12-13 2013-06-12 杜雷科特公司 包含高粘度液体载体材料的口服递药系统
SI2767292T1 (sl) 2004-09-17 2017-01-31 Durect Corporation Pripravek, ki vsebuje lokalni anestetik SAIB, s podaljšanim sproščanjem
US20070027105A1 (en) 2005-07-26 2007-02-01 Alza Corporation Peroxide removal from drug delivery vehicle
ES2388355T3 (es) 2006-11-03 2012-10-11 Durect Corporation Sistemas de suministro transdémico que comprenden bupivacaína
AU2008347158B8 (en) 2007-12-06 2013-08-22 Durect Corporation Oral pharmaceutical dosage forms
US20100260844A1 (en) 2008-11-03 2010-10-14 Scicinski Jan J Oral pharmaceutical dosage forms
CN102093284B (zh) * 2010-12-29 2013-05-08 宜昌人福药业有限责任公司 富集哌啶-2-甲酰苯胺类旋光化合物的方法
WO2014144975A1 (en) 2013-03-15 2014-09-18 Durect Corporation Compositions with a rheological modifier to reduce dissolution variability
CN106187864B (zh) * 2016-07-11 2018-11-23 江苏天和制药有限公司 一种由盐酸布比卡因制备高纯度布比卡因碱的方法
CN115666621A (zh) 2020-01-13 2023-01-31 度勒科特公司 具有减少的杂质的持续释放药物递送系统及相关方法
WO2023158722A2 (en) * 2022-02-16 2023-08-24 Teva Pharmaceuticals International Gmbh Processes for preparation of avacopan and intermediates thereof

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2301498A1 (fr) * 1975-02-20 1976-09-17 Maggioni & C Spa Methode pour la racemisation d'une lysine optiquement active

Also Published As

Publication number Publication date
ATE242214T1 (de) 2003-06-15
DE69628540D1 (de) 2003-07-10
CN1172912C (zh) 2004-10-27
BR9606821A (pt) 1997-12-23
JP4015696B2 (ja) 2007-11-28
WO1996022281A1 (en) 1996-07-25
HU227426B1 (en) 2011-05-30
FI973040A0 (fi) 1997-07-17
FI973040A (fi) 1997-07-17
HUP9901418A3 (en) 2001-01-29
PL184091B1 (pl) 2002-08-30
ZA96403B (en) 1997-01-20
EP0804417B1 (en) 2003-06-04
CN1168134A (zh) 1997-12-17
FI117437B (fi) 2006-10-13
CA2208522A1 (en) 1996-07-25
CA2208522C (en) 2007-03-13
DE69628540T2 (de) 2004-01-08
EP0804417A1 (en) 1997-11-05
AU701221B2 (en) 1999-01-21
JPH11501905A (ja) 1999-02-16
ES2201166T3 (es) 2004-03-16
PT804417E (pt) 2003-09-30
GB9501071D0 (en) 1995-03-08
NO308843B1 (no) 2000-11-06
NO973312L (no) 1997-07-17
PL321378A1 (en) 1997-12-08
HUP9901418A2 (hu) 1999-08-30
KR19980701432A (ko) 1998-05-15
NO973312D0 (no) 1997-07-17
AU4394896A (en) 1996-08-07
KR100404390B1 (ko) 2004-01-31
MX9705428A (es) 1997-11-29

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