DK0697019T3 - Risperidon pamoater - Google Patents

Risperidon pamoater

Info

Publication number
DK0697019T3
DK0697019T3 DK94915538T DK94915538T DK0697019T3 DK 0697019 T3 DK0697019 T3 DK 0697019T3 DK 94915538 T DK94915538 T DK 94915538T DK 94915538 T DK94915538 T DK 94915538T DK 0697019 T3 DK0697019 T3 DK 0697019T3
Authority
DK
Denmark
Prior art keywords
pct
risperidone
pamoater
sec
compositions
Prior art date
Application number
DK94915538T
Other languages
English (en)
Inventor
Jean Louis Mesens
Jozef Peeters
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Application granted granted Critical
Publication of DK0697019T3 publication Critical patent/DK0697019T3/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C65/00Compounds having carboxyl groups bound to carbon atoms of six—membered aromatic rings and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups
    • C07C65/01Compounds having carboxyl groups bound to carbon atoms of six—membered aromatic rings and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups containing hydroxy or O-metal groups
    • C07C65/105Compounds having carboxyl groups bound to carbon atoms of six—membered aromatic rings and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups containing hydroxy or O-metal groups polycyclic
    • C07C65/11Compounds having carboxyl groups bound to carbon atoms of six—membered aromatic rings and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups containing hydroxy or O-metal groups polycyclic with carboxyl groups on a condensed ring system containing two rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
DK94915538T 1993-04-28 1994-04-22 Risperidon pamoater DK0697019T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP93201216 1993-04-28
PCT/EP1994/001296 WO1994025460A1 (en) 1993-04-28 1994-04-22 Risperidone pamoate

Publications (1)

Publication Number Publication Date
DK0697019T3 true DK0697019T3 (da) 1998-09-28

Family

ID=8213799

Family Applications (1)

Application Number Title Priority Date Filing Date
DK94915538T DK0697019T3 (da) 1993-04-28 1994-04-22 Risperidon pamoater

Country Status (32)

Country Link
US (2) US5612346A (da)
EP (1) EP0697019B1 (da)
JP (1) JP3478397B2 (da)
KR (1) KR100307101B1 (da)
CN (1) CN1041727C (da)
AT (1) ATE163418T1 (da)
AU (1) AU675136B2 (da)
BG (1) BG62004B1 (da)
CA (1) CA2160366C (da)
CY (1) CY2107B1 (da)
CZ (1) CZ286688B6 (da)
DE (1) DE69408666T2 (da)
DK (1) DK0697019T3 (da)
ES (1) ES2113652T3 (da)
FI (1) FI109125B (da)
GR (1) GR3026028T3 (da)
HK (1) HK1006059A1 (da)
HU (1) HU218212B (da)
IL (1) IL109448A (da)
LV (1) LV12315B (da)
NO (1) NO305083B1 (da)
NZ (1) NZ266143A (da)
PH (1) PH30476A (da)
PL (1) PL182466B1 (da)
RO (1) RO115955B1 (da)
RU (1) RU2131428C1 (da)
SG (1) SG47046A1 (da)
SI (1) SI9420031B (da)
SK (1) SK280589B6 (da)
TW (1) TW376319B (da)
WO (1) WO1994025460A1 (da)
ZA (1) ZA942909B (da)

Families Citing this family (42)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2236700T3 (es) 1993-11-19 2005-07-16 Janssen Pharmaceutica N.V. 1,2-benzazoles microencapsulados.
US5453425A (en) * 1994-07-11 1995-09-26 Janssen Pharmaceutica N.V. Risperidone oral formulation
TW487572B (en) * 1996-05-20 2002-05-21 Janssen Pharmaceutica Nv Aqueous suspensions of 9-hydroxyrisperidone fatty acid esters
US6617321B2 (en) 1997-09-30 2003-09-09 Eli Lilly And Company 2-methyl-thieno-benzodiazepine formulation
IL135295A0 (en) * 1997-09-30 2001-05-20 Lilly Co Eli 2-methyl-thieno-benzodiazepine formulation
UA72189C2 (uk) * 1997-11-17 2005-02-15 Янссен Фармацевтика Н.В. Фармацевтична композиція, що містить водну суспензію субмікронних ефірів 9-гідроксирисперидон жирних кислот
DK1119359T3 (da) * 1998-09-30 2004-08-16 Lilly Co Eli 2-methyl-thieno-benzodiazepinformulering
JP2002529468A (ja) * 1998-11-12 2002-09-10 メルク エンド カムパニー インコーポレーテッド GABA−Aα−5逆活性薬の治療性多形およびそのパモエート組成物
FR2802101B1 (fr) 1999-12-10 2003-02-28 Aventis Pharma Sa Association de cymemazine et d'un neuroleptique atypique
US6770478B2 (en) * 2000-02-10 2004-08-03 The Regents Of The University Of California Erythrocytic cells and method for preserving cells
US6495164B1 (en) 2000-05-25 2002-12-17 Alkermes Controlled Therapeutics, Inc. I Preparation of injectable suspensions having improved injectability
WO2002043766A1 (fr) * 2000-11-29 2002-06-06 Takeda Chemical Industries, Ltd. Compositions medicinales et leur procede de preparation
US20050232995A1 (en) 2002-07-29 2005-10-20 Yam Nyomi V Methods and dosage forms for controlled delivery of paliperidone and risperidone
US20060148826A1 (en) * 2002-08-23 2006-07-06 Ashish Gogia Stable aqueous solutions of risperidone and methods for their preparation
KR20040034996A (ko) * 2002-10-18 2004-04-29 한미약품 주식회사 리스페리돈의 개선된 제조방법
WO2004094414A1 (en) * 2003-04-22 2004-11-04 Synthon B.V. Water soluble salts of risperidone
US6987111B2 (en) * 2003-08-06 2006-01-17 Alkermes Controlled Therapeutics, Ii Aripiprazole, olanzapine and haloperidol pamoate salts
PT1675573E (pt) * 2003-10-23 2008-12-30 Otsuka Pharma Co Ltd Formulação de iripiprazole injectável estéril de libertação controlada e um processo para a sua preparação
US7884096B2 (en) * 2003-12-02 2011-02-08 Pharmaneuroboost N.V. Method of treating mental disorders using of D4 and 5-HT2A antagonists, inverse agonists or partial agonists
CA2547639A1 (en) * 2003-12-02 2005-06-16 B&B Beheer Nv Use of d4 and 5-ht2a antagonists, inverse agonists or partial agonists
CA2554959A1 (en) * 2004-01-29 2005-08-11 Neuromolecular, Inc. Combination of a nmda receptor antagonist and a mao-inhibitor or a gadpf-inhibitor for the treatment of central nervous system-related conditions
PL1838716T3 (pl) * 2005-01-05 2011-09-30 Lilly Co Eli Dihydrat embonianu olanzapiny
EP1695973A1 (en) * 2005-02-24 2006-08-30 Neuro3D Ocaperidone salt and pharmaceutical compositions containing the same
AR055099A1 (es) * 2005-07-28 2007-08-08 Alza Corp Formulaciones liquidas para la administracion controlada de derivados de bencisoxazol
EP2279727A3 (en) * 2005-09-15 2011-10-05 Elan Pharma International Limited Nanoparticulate aripiprazole formulations
US8852638B2 (en) 2005-09-30 2014-10-07 Durect Corporation Sustained release small molecule drug formulation
CN101801415B (zh) 2007-05-25 2015-09-23 Rb医药品有限公司 利培酮化合物的持续递送制剂
RU2483711C2 (ru) * 2007-07-31 2013-06-10 Оцука Фармасьютикал Ко., Лтд. Способы получения суспензии арипипразола и лиофилизированного состава
KR20100099292A (ko) * 2007-12-19 2010-09-10 얀센 파마슈티카 엔.브이. 장기 작용성 주사가능 팔리페리돈 에스테르와 관련된 투여 요법
CA2830511C (en) 2011-03-18 2021-09-14 Alkermes Pharma Ireland Limited Pharmaceutical compositions comprising aripiprazole lauroxil and sorbitan laurate
PL2702060T3 (pl) 2011-04-26 2016-06-30 Torrent Pharmaceuticals Ltd Kwasowe addycyjne sole risperidonu i ich kompozycje farmaceutyczne
CA2867121C (en) 2012-03-19 2021-05-25 Alkermes Pharma Ireland Limited Pharmaceutical compositions comprising fatty acid esters
US9999670B2 (en) 2012-03-19 2018-06-19 Alkermes Pharma Ireland Limited Pharmaceutical compositions comprising benzyl alcohol
US9993556B2 (en) 2012-03-19 2018-06-12 Alkermes Pharma Ireland Limited Pharmaceutical compositions comprising fatty glycerol esters
CN109010296A (zh) 2012-04-04 2018-12-18 英特维特国际股份有限公司 异噁唑啉化合物的固体口服药物组合物
CN102659577B (zh) * 2012-04-07 2014-07-02 安徽绩溪县徽煌化工有限公司 一种亚甲基双羟基萘酸的制备方法
EP3718536A1 (en) 2012-09-19 2020-10-07 Alkermes Pharma Ireland Limited Pharmaceutical compositions having improved storage stability
WO2014049071A1 (en) 2012-09-26 2014-04-03 Tangent Reprofiling Limited Modulators of androgen synthesis
US9375433B2 (en) 2012-09-26 2016-06-28 Tangent Reprofiling Limited Modulators of androgen synthesis
MA39495A (fr) 2014-03-20 2015-09-24 Alkermes Pharma Ireland Ltd Formulations d'aripiprazole présentant des vitesses d'injection plus élevées
CN106831594B (zh) * 2017-01-18 2018-02-02 力赛生物医药科技(厦门)有限公司 可乐定双羟萘酸盐及其制备方法
EP3761983A1 (en) 2018-03-05 2021-01-13 Alkermes Pharma Ireland Limited Aripiprazole dosing strategy

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4804663A (en) * 1985-03-27 1989-02-14 Janssen Pharmaceutica N.V. 3-piperidinyl-substituted 1,2-benzisoxazoles and 1,2-benzisothiazoles

Also Published As

Publication number Publication date
CA2160366A1 (en) 1994-11-10
FI955166A (fi) 1995-10-27
CN1121719A (zh) 1996-05-01
CZ286688B6 (en) 2000-06-14
HUT72970A (en) 1996-06-28
NO305083B1 (no) 1999-03-29
SK131395A3 (en) 1996-06-05
HU9501934D0 (en) 1995-09-28
CN1041727C (zh) 1999-01-20
EP0697019A1 (en) 1996-02-21
IL109448A (en) 1997-03-18
BG62004B1 (bg) 1998-12-30
AU6721694A (en) 1994-11-21
SK280589B6 (sk) 2000-04-10
LV12315B (en) 2000-03-20
US5723467A (en) 1998-03-03
NO954275L (no) 1995-10-26
IL109448A0 (en) 1994-07-31
CA2160366C (en) 2006-06-06
FI955166A0 (fi) 1995-10-27
ZA942909B (en) 1995-10-26
HU218212B (hu) 2000-06-28
EP0697019B1 (en) 1998-02-25
DE69408666T2 (de) 1998-06-18
KR100307101B1 (ko) 2001-11-30
SI9420031A (en) 1996-08-31
PL311282A1 (en) 1996-02-05
FI109125B (fi) 2002-05-31
ES2113652T3 (es) 1998-05-01
JP3478397B2 (ja) 2003-12-15
CZ270695A3 (en) 1996-01-17
SI9420031B (sl) 2002-08-31
LV12315A (lv) 1999-07-20
WO1994025460A1 (en) 1994-11-10
BG100094A (bg) 1996-05-31
RO115955B1 (ro) 2000-08-30
AU675136B2 (en) 1997-01-23
GR3026028T3 (en) 1998-04-30
RU2131428C1 (ru) 1999-06-10
PH30476A (en) 1997-05-28
NZ266143A (en) 1996-07-26
JPH08509482A (ja) 1996-10-08
SG47046A1 (en) 1998-03-20
TW376319B (en) 1999-12-11
NO954275D0 (no) 1995-10-26
ATE163418T1 (de) 1998-03-15
CY2107B1 (en) 2002-04-26
DE69408666D1 (de) 1998-04-02
PL182466B1 (pl) 2002-01-31
US5612346A (en) 1997-03-18
HK1006059A1 (en) 1999-02-05

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