DK0639179T3 - 23-oxaderivater i D-vitaminserien, fremgangsmåde til fremstilling heraf, farmaceutiske præparater indeholdende disse derivater samt deres anvendelse som lægemidler - Google Patents

23-oxaderivater i D-vitaminserien, fremgangsmåde til fremstilling heraf, farmaceutiske præparater indeholdende disse derivater samt deres anvendelse som lægemidler

Info

Publication number
DK0639179T3
DK0639179T3 DK92903336.3T DK92903336T DK0639179T3 DK 0639179 T3 DK0639179 T3 DK 0639179T3 DK 92903336 T DK92903336 T DK 92903336T DK 0639179 T3 DK0639179 T3 DK 0639179T3
Authority
DK
Denmark
Prior art keywords
derivatives
pct
vitamin
series
drugs
Prior art date
Application number
DK92903336.3T
Other languages
Danish (da)
English (en)
Inventor
Martin Haberey
Petra Rach
Ruth Thieroff-Ekerdt
Guenter Neef
Katica Schwarz
Andreas Steinmeyer
Gerald Kirsch
Original Assignee
Schering Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Schering Ag filed Critical Schering Ag
Application granted granted Critical
Publication of DK0639179T3 publication Critical patent/DK0639179T3/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C401/00Irradiation products of cholesterol or its derivatives; Vitamin D derivatives, 9,10-seco cyclopenta[a]phenanthrene or analogues obtained by chemical preparation without irradiation
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Dermatology (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
DK92903336.3T 1991-01-19 1992-01-20 23-oxaderivater i D-vitaminserien, fremgangsmåde til fremstilling heraf, farmaceutiske præparater indeholdende disse derivater samt deres anvendelse som lægemidler DK0639179T3 (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE4101953A DE4101953A1 (de) 1991-01-19 1991-01-19 23-oxa-derivate in der vitamin-d-reihe, verfahren zu ihrer herstellung diese derivate enthaltende pharmazeutische praeparate sowie deren verwendung als arzneimittel

Publications (1)

Publication Number Publication Date
DK0639179T3 true DK0639179T3 (da) 1996-10-14

Family

ID=6423566

Family Applications (1)

Application Number Title Priority Date Filing Date
DK92903336.3T DK0639179T3 (da) 1991-01-19 1992-01-20 23-oxaderivater i D-vitaminserien, fremgangsmåde til fremstilling heraf, farmaceutiske præparater indeholdende disse derivater samt deres anvendelse som lægemidler

Country Status (11)

Country Link
US (1) US5411949A (pt)
EP (1) EP0639179B1 (pt)
JP (1) JP3207423B2 (pt)
AT (1) ATE138647T1 (pt)
DE (2) DE4101953A1 (pt)
DK (1) DK0639179T3 (pt)
ES (1) ES2089497T3 (pt)
GR (1) GR3020083T3 (pt)
IE (1) IE74251B1 (pt)
PT (1) PT100035B (pt)
WO (1) WO1992012963A1 (pt)

Families Citing this family (25)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PT665221E (pt) * 1992-10-16 2000-06-30 Chugai Pharmaceutical Co Ltd Derivado da vitamina d e processo para a sua producao
TW267161B (pt) * 1992-11-20 1996-01-01 Hoffmann La Roche
US6407082B1 (en) * 1996-09-13 2002-06-18 New Life Pharmaceuticals Inc. Prevention of ovarian cancer by administration of a vitamin D compound
US20040167106A1 (en) * 1993-06-04 2004-08-26 Rodriguez Gustavo C. Prevention of ovarian cancer by administration of a Vitamin D compound
EP0873126A4 (en) 1995-12-29 2000-04-19 A And D Assay Inc BRANDED VITAMIN COMPOUNDS AND THEIR USE
US6028064A (en) 1996-09-13 2000-02-22 New Life Pharmaceuticals Inc. Prevention of ovarian cancer by administration of progestin products
US6511970B1 (en) 1996-09-13 2003-01-28 New Life Pharmaceuticals Inc. Prevention of ovarian cancer by administration of products that induce transforming growth factor-beta and/or apoptosis in the ovarian epithelium
US6034074A (en) * 1996-09-13 2000-03-07 New Life Pharmaceuticals Inc. Prevention of ovarian cancer by administration of a Vitamin D compound
US6765002B2 (en) 2000-03-21 2004-07-20 Gustavo Rodriguez Prevention of ovarian cancer by administration of products that induce transforming growth factor-β and/or apoptosis in the ovarian epithelium
US6087350A (en) * 1997-08-29 2000-07-11 University Of Pittsburgh Of The Commonwealth System Of Higher Education Use of pretreatment chemicals to enhance efficacy of cytotoxic agents
EP1064000B1 (en) * 1998-03-27 2011-07-06 Oregon Health & Science University Vitamin d and its analogs in the treatment of tumors and other hyperproliferative disorders
ATE253555T1 (de) * 1999-04-23 2003-11-15 Leo Pharma As Vitamin d-analogen und ihre pharmazeutische verwendung
US20010044431A1 (en) * 2000-03-21 2001-11-22 Rodriguez Gustavo C. Prevention of ovarian cancer by administration of products that induce biologic effects in the ovarian epithelium
CA2510228C (en) * 2002-12-18 2012-10-30 Johns Hopkins University 25-so2-substituted analogs of 1.alpha.,25-dihydroxyvitamin d3
US9173835B2 (en) 2005-05-10 2015-11-03 Dermipsor Ltd. Compositions and methods for treating hyperproliferative epidermal diseases
US20080051375A1 (en) * 2006-08-25 2008-02-28 Auerbach Alan H Methods for treating cancer comprising the administration of a vitamin d compound and an additional therapeutic agent, and compositions containing the same
KR20090060306A (ko) 2006-08-25 2009-06-11 코우가 바이오테크놀로지, 인크. 비타민 d 화합물 및 추가 치료제, 및 그를 함유하는 조성물을 투여하는 것을 포함하는, 암을 치료하는 방법
US20080051380A1 (en) 2006-08-25 2008-02-28 Auerbach Alan H Methods and compositions for treating cancer
US20090124587A1 (en) * 2007-07-12 2009-05-14 Auerbach Alan H METHODS FOR TREATING CANCER USING 17alpha-HYDROXYLASE/C17,20-LYASE INHIBITORS
CN107019795A (zh) * 2009-01-27 2017-08-08 博格有限责任公司 用于减轻与化疗有关的副作用的维生素d3化合物
MX366076B (es) 2009-08-14 2019-06-27 Berg Llc Vitamina d3 y analogos de la misma para tratar alopecia.
FI124171B (en) 2012-05-29 2014-04-15 Matti Mällinen Biofilter
WO2017209934A1 (en) 2016-05-13 2017-12-07 Case Western Reserve University Autophagy activators for treating or preventing skin injury
WO2018023017A1 (en) 2016-07-29 2018-02-01 Janssen Pharmaceutica Nv Methods of treating prostate cancer
US11903952B2 (en) 2020-05-27 2024-02-20 Northwestern University Vitamin D as an immune modulator to prevent immune-related complication from COVID-19 infection

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0078704B1 (en) * 1981-11-02 1987-04-29 Research Institute For Medicine And Chemistry Inc. Intermediates in the synthesis of vitamin d derivatives
DE3577552D1 (de) * 1984-11-27 1990-06-13 Chugai Pharmaceutical Co Ltd Vitamin d-derivate und verfahren zu deren herstellung.
GB8904153D0 (en) * 1989-02-23 1989-04-05 Leo Pharm Prod Ltd Chemical compounds
GB9007236D0 (en) * 1990-03-30 1990-05-30 Leo Pharm Prod Ltd Chemical compounds

Also Published As

Publication number Publication date
IE920156A1 (en) 1992-07-29
DE4101953A1 (de) 1992-07-23
EP0639179B1 (de) 1996-05-29
PT100035B (pt) 1999-08-31
US5411949A (en) 1995-05-02
WO1992012963A1 (de) 1992-08-06
EP0639179A4 (de) 1993-09-17
DE59206439D1 (de) 1996-07-04
PT100035A (pt) 1993-05-31
ATE138647T1 (de) 1996-06-15
GR3020083T3 (en) 1996-08-31
EP0639179A1 (de) 1995-02-22
JPH06506915A (ja) 1994-08-04
IE74251B1 (en) 1997-07-16
JP3207423B2 (ja) 2001-09-10
ES2089497T3 (es) 1996-10-01

Similar Documents

Publication Publication Date Title
DK0639179T3 (da) 23-oxaderivater i D-vitaminserien, fremgangsmåde til fremstilling heraf, farmaceutiske præparater indeholdende disse derivater samt deres anvendelse som lægemidler
NO981944L (no) Lipopolyaminer som transfeksjonsmidler samt farmas÷ytisk anvendelse derav
ES2114931T3 (es) Nuevos esteres esteroidales.
AR024390A1 (es) Nuevos compuestos
ATE29255T1 (de) Succinimid-derivate und deren herstellung.
ES2051753T3 (es) N-(1-azabiciclo(2.2.2)octo-3-il) benzamidas y tiobenzamidas ansioliticas.
ES8403494A1 (es) "un procedimiento para la preparacion de derivados de s-adenosilmetionina".
FI894061A (fi) Menetelmä lääkeaineina käyttökelpoisten , -disubstituoitujen N-sykloalkyylialkyylibentsyyliamiinien valmistamiseksi ja niiden synteesivälituotteita
DK0649405T3 (da) 22-en-25-oxa-derivater i D-vitaminserien, fremgangsmåde til fremstilling heraf, farmaceutiske præparater indeholdende disse derivater samt anvendelse af sådanne præparater som lægemidler.
ES2063039T3 (es) Derivados de imidazo(1,2-b)piridazina.
FI922806A0 (fi) Substituerade 4-fenyl-4 -piperidinkarboxamider med baode lokalbedoevande och smaertstillande effekt samt foerfaranden foer deras framstaellning.
FR2631625B1 (fr) Derives de phenyl-6 piperazinylalkyl-3 1h,3h-pyrimidinedione-2,4, leur preparation et leur application en therapeutique
ES2091126T3 (es) Nuevos compuestos biciclicos de pirimidina, su procedimiento de preparacion y composiciones farmaceuticas que los contienen.
ES2164869T3 (es) Conjugados lipidos especificos de nucleosidos-difosfato y su uso como medicamentos.
PT97286A (pt) Processo para a preparacao de novos derivados do 3-aminocromano e de composicoes farmaceuticas que os contem
DK157489C (da) N-substituerede pyridiniumforbindelser og farmaceutiske praeparater indeholdende disse
DE3870167D1 (de) N-(vinblastinoyl-23)-derivate von 1-aminomethylposphonsaeure, verfahren zu ihrer herstellung und sie enthaltende arzneimittel.
AR012601A1 (es) Derivados de amidina, formulaciones farmaceuticas que los contiene, uso de dichos derivados en la preparacion de medicamentos y proceso para lapreparacion de dichos derivados
ES8402839A1 (es) Procedimiento para la obtencion de nuevos poliazaheterociclicos policiclicos.
DK601888D0 (da) Anvendelse af 2-pyrimidinyl-1-piperazinderivater
ES2149817T3 (es) Piridinas sustituidas, su preparacion y uso farmaceutico.
NO301760B1 (no) Farmakologisk aktive <alfa>-[tertiær-aminometyl]-benzenmetanolderivater, farmasöytiske preparater inneholdende disse samt anvendelse av forbindelsene for fremstilling av farmasöytiske preparater
DE69300011D1 (de) Diacylglycerol-Nicotinate, Verfahren zu ihrer Herstellung und diese enthaltende pharmazeutische Zubereitungen.
ES479440A1 (es) Un procedimiento para preparar compuestos con propiedades broncodilatadoras.
DK179389A (da) Trienderivater indeholdende en chromenstruktur, fremgangsmaade til fremstilling heraf samt farmaceutiske midler indeholdende disse derivater