PT100035A - 23-oxa-derivados da serie da vitamina d processo para a sua preparacao composicoes farmaceuticas contendo esses derivados bem como a sua utilizacao como medicamentos - Google Patents

23-oxa-derivados da serie da vitamina d processo para a sua preparacao composicoes farmaceuticas contendo esses derivados bem como a sua utilizacao como medicamentos

Info

Publication number
PT100035A
PT100035A PT100035A PT10003592A PT100035A PT 100035 A PT100035 A PT 100035A PT 100035 A PT100035 A PT 100035A PT 10003592 A PT10003592 A PT 10003592A PT 100035 A PT100035 A PT 100035A
Authority
PT
Portugal
Prior art keywords
derivatives
pct
oxa
vitamin
medicines
Prior art date
Application number
PT100035A
Other languages
English (en)
Other versions
PT100035B (pt
Inventor
Gerald Kirsch
Katica Schwarz
Ruth Thieroff-Ekerdt
Petra Rach
Andreas Steinmeyer
Gunter Neel
Martin Haberey
Original Assignee
Schering Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Schering Ag filed Critical Schering Ag
Publication of PT100035A publication Critical patent/PT100035A/pt
Publication of PT100035B publication Critical patent/PT100035B/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C401/00Irradiation products of cholesterol or its derivatives; Vitamin D derivatives, 9,10-seco cyclopenta[a]phenanthrene or analogues obtained by chemical preparation without irradiation
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Dermatology (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
PT100035A 1991-01-19 1992-01-17 23-oxa-derivados da serie da vitamina d processo para a sua preparacao composicoes farmaceuticas contendo esses derivados bem como a sua utilizacao como medicamentos PT100035B (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE4101953A DE4101953A1 (de) 1991-01-19 1991-01-19 23-oxa-derivate in der vitamin-d-reihe, verfahren zu ihrer herstellung diese derivate enthaltende pharmazeutische praeparate sowie deren verwendung als arzneimittel

Publications (2)

Publication Number Publication Date
PT100035A true PT100035A (pt) 1993-05-31
PT100035B PT100035B (pt) 1999-08-31

Family

ID=6423566

Family Applications (1)

Application Number Title Priority Date Filing Date
PT100035A PT100035B (pt) 1991-01-19 1992-01-17 23-oxa-derivados da serie da vitamina d processo para a sua preparacao composicoes farmaceuticas contendo esses derivados bem como a sua utilizacao como medicamentos

Country Status (11)

Country Link
US (1) US5411949A (pt)
EP (1) EP0639179B1 (pt)
JP (1) JP3207423B2 (pt)
AT (1) ATE138647T1 (pt)
DE (2) DE4101953A1 (pt)
DK (1) DK0639179T3 (pt)
ES (1) ES2089497T3 (pt)
GR (1) GR3020083T3 (pt)
IE (1) IE74251B1 (pt)
PT (1) PT100035B (pt)
WO (1) WO1992012963A1 (pt)

Families Citing this family (24)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ATE189887T1 (de) * 1992-10-16 2000-03-15 Chugai Pharmaceutical Co Ltd Vitamin-d-derivat und verfahren zu seiner herstellung
TW267161B (pt) * 1992-11-20 1996-01-01 Hoffmann La Roche
US20040167106A1 (en) * 1993-06-04 2004-08-26 Rodriguez Gustavo C. Prevention of ovarian cancer by administration of a Vitamin D compound
US6407082B1 (en) * 1996-09-13 2002-06-18 New Life Pharmaceuticals Inc. Prevention of ovarian cancer by administration of a vitamin D compound
WO1997024127A1 (en) * 1995-12-29 1997-07-10 A And D Assay, Incorporated Labeled vitamin d compounds and the use thereof
US6034074A (en) 1996-09-13 2000-03-07 New Life Pharmaceuticals Inc. Prevention of ovarian cancer by administration of a Vitamin D compound
US6765002B2 (en) 2000-03-21 2004-07-20 Gustavo Rodriguez Prevention of ovarian cancer by administration of products that induce transforming growth factor-β and/or apoptosis in the ovarian epithelium
US6511970B1 (en) 1996-09-13 2003-01-28 New Life Pharmaceuticals Inc. Prevention of ovarian cancer by administration of products that induce transforming growth factor-beta and/or apoptosis in the ovarian epithelium
US6028064A (en) 1996-09-13 2000-02-22 New Life Pharmaceuticals Inc. Prevention of ovarian cancer by administration of progestin products
US6087350A (en) * 1997-08-29 2000-07-11 University Of Pittsburgh Of The Commonwealth System Of Higher Education Use of pretreatment chemicals to enhance efficacy of cytotoxic agents
AU762481C (en) 1998-03-27 2004-08-19 Oregon Health Sciences University Vitamin D and its analogs in the treatment of tumors and other hyperproliferative disorders
KR20010109357A (ko) * 1999-04-23 2001-12-08 룬딩 에른스트 비타민 d 동족체 및 이의 약제학적 용도
US20010044431A1 (en) * 2000-03-21 2001-11-22 Rodriguez Gustavo C. Prevention of ovarian cancer by administration of products that induce biologic effects in the ovarian epithelium
WO2004054968A2 (en) * 2002-12-18 2004-07-01 Johns Hopkins University 25-so2-substituted analogs of 1alpha, 25-dihydroxyvitamin d3 (calcitriol)
NZ563270A (en) 2005-05-10 2010-11-26 Dermipsor Ltd Calcipotriol, polyethylene oxide topical compositions for the treatment of hyperproliferative epidermal diseases
WO2008024485A2 (en) 2006-08-25 2008-02-28 Cougar Biotechnology, Inc. Methods for treating cancer comprising the administration of a vitamin d compound and an additional therapeutic agent
US20080051380A1 (en) 2006-08-25 2008-02-28 Auerbach Alan H Methods and compositions for treating cancer
US20080051375A1 (en) * 2006-08-25 2008-02-28 Auerbach Alan H Methods for treating cancer comprising the administration of a vitamin d compound and an additional therapeutic agent, and compositions containing the same
WO2009009132A1 (en) * 2007-07-12 2009-01-15 Cougar Biotechnology, Inc. Use of 17alpha-hydroxylase/c17, 20-lyase inhibitors for the treatment of cancer
KR20170096238A (ko) * 2009-01-27 2017-08-23 베르그 엘엘씨 화학요법과 연관된 부작용을 경감시키기 위한 비타민 d3 및 이의 유사물
JP5978130B2 (ja) 2009-08-14 2016-08-24 バーグ エルエルシー 脱毛症を治療するためのビタミンd3およびその類似体
FI124171B (en) 2012-05-29 2014-04-15 Matti Mällinen Biofilter
WO2017209934A1 (en) 2016-05-13 2017-12-07 Case Western Reserve University Autophagy activators for treating or preventing skin injury
US11903952B2 (en) 2020-05-27 2024-02-20 Northwestern University Vitamin D as an immune modulator to prevent immune-related complication from COVID-19 infection

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0078704B1 (en) * 1981-11-02 1987-04-29 Research Institute For Medicine And Chemistry Inc. Intermediates in the synthesis of vitamin d derivatives
EP0184112B1 (en) * 1984-11-27 1990-05-09 Chugai Seiyaku Kabushiki Kaisha Novel vitamin d derivatives and process for producing the same
GB8904153D0 (en) * 1989-02-23 1989-04-05 Leo Pharm Prod Ltd Chemical compounds
GB9007236D0 (en) * 1990-03-30 1990-05-30 Leo Pharm Prod Ltd Chemical compounds

Also Published As

Publication number Publication date
US5411949A (en) 1995-05-02
DE4101953A1 (de) 1992-07-23
ES2089497T3 (es) 1996-10-01
DE59206439D1 (de) 1996-07-04
DK0639179T3 (da) 1996-10-14
EP0639179B1 (de) 1996-05-29
IE920156A1 (en) 1992-07-29
PT100035B (pt) 1999-08-31
EP0639179A1 (de) 1995-02-22
GR3020083T3 (en) 1996-08-31
JPH06506915A (ja) 1994-08-04
EP0639179A4 (de) 1993-09-17
ATE138647T1 (de) 1996-06-15
JP3207423B2 (ja) 2001-09-10
IE74251B1 (en) 1997-07-16
WO1992012963A1 (de) 1992-08-06

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Legal Events

Date Code Title Description
BB1A Laying open of patent application

Effective date: 19930121

FG3A Patent granted, date of granting

Effective date: 19990526

MM4A Annulment/lapse due to non-payment of fees, searched and examined patent

Free format text: LAPSE DUE TO NON-PAYMENT OF FEES

Effective date: 20071126