DE60309739T2 - Pyridinderivate als modulatoren des cb2-rezeptors - Google Patents

Pyridinderivate als modulatoren des cb2-rezeptors Download PDF

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Publication number
DE60309739T2
DE60309739T2 DE60309739T DE60309739T DE60309739T2 DE 60309739 T2 DE60309739 T2 DE 60309739T2 DE 60309739 T DE60309739 T DE 60309739T DE 60309739 T DE60309739 T DE 60309739T DE 60309739 T2 DE60309739 T2 DE 60309739T2
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Prior art keywords
fluorobenzyl
isopropylnicotinamide
chlorophenylamino
trifluoromethylnicotinamide
alkyl
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Expired - Fee Related
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DE60309739T
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German (de)
English (en)
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DE60309739D1 (de
Inventor
Andrew John Harlow EATHERTON
Gerard Martin Paul Harlow GIBLIN
Howard deceased Howard Harlow GREEN
Karamjit Singh Harlow JANDU
William Leonard Harlow MITCHELL
Alan Harlow NAYLOR
C/o NiKem Research S.r.L. Giovanni PALOMBI
Derek Anthony Harlow RAWLINGS
Brian Peter Harlow SLINGSBY
Andrew Richard Stevenage WHITTINGTON
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Glaxo Group Ltd
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Glaxo Group Ltd
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    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
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DE60309739T 2002-09-27 2003-09-25 Pyridinderivate als modulatoren des cb2-rezeptors Expired - Fee Related DE60309739T2 (de)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB0222495 2002-09-27
GBGB0222495.4A GB0222495D0 (en) 2002-09-27 2002-09-27 Compounds
PCT/EP2003/010935 WO2004029027A1 (en) 2002-09-27 2003-09-25 Pyridine derivatives as cb2 receptor modulators

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Publication Number Publication Date
DE60309739D1 DE60309739D1 (de) 2006-12-28
DE60309739T2 true DE60309739T2 (de) 2007-10-31

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US (1) US20070129367A1 (enExample)
EP (1) EP1562907B1 (enExample)
JP (1) JP2006508065A (enExample)
AT (1) ATE345329T1 (enExample)
AU (1) AU2003276028A1 (enExample)
DE (1) DE60309739T2 (enExample)
ES (1) ES2277149T3 (enExample)
GB (1) GB0222495D0 (enExample)
WO (1) WO2004029027A1 (enExample)

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WO2003082191A2 (en) 2002-03-28 2003-10-09 Merck & Co., Inc. Substituted 2,3-diphenyl pyridines
UY27939A1 (es) 2002-08-21 2004-03-31 Glaxo Group Ltd Compuestos
TW200505902A (en) 2003-03-20 2005-02-16 Schering Corp Cannabinoid receptor ligands
EP1669348A4 (en) 2003-09-30 2009-03-11 Eisai R&D Man Co Ltd NEW ANTIPILIC AGENT CONTAINING A HETEROCYCLIC COMPOUND
GB0402356D0 (en) * 2004-02-03 2004-03-10 Glaxo Group Ltd Novel compounds
GB0402357D0 (en) * 2004-02-03 2004-03-10 Glaxo Group Ltd Novel compounds
GB0402355D0 (en) * 2004-02-03 2004-03-10 Glaxo Group Ltd Novel compounds
JP4874958B2 (ja) 2005-03-30 2012-02-15 エーザイ・アール・アンド・ディー・マネジメント株式会社 ピリジン誘導体を含有する抗真菌剤
JPWO2006129609A1 (ja) * 2005-05-30 2009-01-08 塩野義製薬株式会社 ２−ナフチルイミノ−５，５−ジ置換−１，３−チアジン誘導体
TWI385169B (zh) 2005-10-31 2013-02-11 Eisai R&D Man Co Ltd 經雜環取代之吡啶衍生物及含有彼之抗真菌劑
WO2007118041A1 (en) * 2006-04-07 2007-10-18 Boehringer Ingelheim International Gmbh Compounds which modulate the cb2 receptor
EP2081905B1 (en) 2006-07-28 2012-09-12 Boehringer Ingelheim International GmbH Sulfonyl compounds which modulate the cb2 receptor
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AU2003276028A1 (en) 2004-04-19
ES2277149T3 (es) 2007-07-01
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ATE345329T1 (de) 2006-12-15
GB0222495D0 (en) 2002-11-06

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