JP2006508065A - Ｃｂ２受容体モジュレーターとしてのピリジン誘導体 - Google Patents

Ｃｂ２受容体モジュレーターとしてのピリジン誘導体 Download PDF

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JP2006508065A
JP2006508065A JP2004539059A JP2004539059A JP2006508065A JP 2006508065 A JP2006508065 A JP 2006508065A JP 2004539059 A JP2004539059 A JP 2004539059A JP 2004539059 A JP2004539059 A JP 2004539059A JP 2006508065 A JP2006508065 A JP 2006508065A
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alkyl
substituted
hydrogen
halo
compound
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JP2006508065A5 (enExample
Inventor
アンドリュー・ジョン・イーサートン
ジェラード・マーティン・ポール・ギブリン
リチャード・ハワード・グリーン
カラムジット・シン・ジャンドゥ
ウィリアム・レナード・ミッチェル
アラン・ネイラー
ジョヴァンニ・パロンビ
デレク・アンソニー・ローリングズ
ブライアン・ピーター・スリングズビー
アンドリュー・リチャード・ホイッティントン
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Glaxo Group Ltd
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Glaxo Group Ltd
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Publication of JP2006508065A publication Critical patent/JP2006508065A/ja
Publication of JP2006508065A5 publication Critical patent/JP2006508065A5/ja
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    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
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  • Diabetes (AREA)
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  • Dermatology (AREA)
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JP2004539059A 2002-09-27 2003-09-25 Ｃｂ２受容体モジュレーターとしてのピリジン誘導体 Withdrawn JP2006508065A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB0222495.4A GB0222495D0 (en) 2002-09-27 2002-09-27 Compounds
PCT/EP2003/010935 WO2004029027A1 (en) 2002-09-27 2003-09-25 Pyridine derivatives as cb2 receptor modulators

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JP2006508065A true JP2006508065A (ja) 2006-03-09
JP2006508065A5 JP2006508065A5 (enExample) 2006-05-18

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US (1) US20070129367A1 (enExample)
EP (1) EP1562907B1 (enExample)
JP (1) JP2006508065A (enExample)
AT (1) ATE345329T1 (enExample)
AU (1) AU2003276028A1 (enExample)
DE (1) DE60309739T2 (enExample)
ES (1) ES2277149T3 (enExample)
GB (1) GB0222495D0 (enExample)
WO (1) WO2004029027A1 (enExample)

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2013537173A (ja) * 2010-09-09 2013-09-30 エフ．ホフマン−ラ ロシュ アーゲー ヘテロアリールメチルアミド
JP2014510696A (ja) * 2010-10-20 2014-05-01 グリュネンタール・ゲゼルシャフト・ミト・ベシュレンクテル・ハフツング Ｋｃｎｑ２／３調節因子としての置換６−アミノ−ニコチンアミド

Families Citing this family (41)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2003082191A2 (en) 2002-03-28 2003-10-09 Merck & Co., Inc. Substituted 2,3-diphenyl pyridines
UY27939A1 (es) 2002-08-21 2004-03-31 Glaxo Group Ltd Compuestos
TW200505902A (en) 2003-03-20 2005-02-16 Schering Corp Cannabinoid receptor ligands
EP1669348A4 (en) 2003-09-30 2009-03-11 Eisai R&D Man Co Ltd NEW ANTIPILIC AGENT CONTAINING A HETEROCYCLIC COMPOUND
GB0402356D0 (en) * 2004-02-03 2004-03-10 Glaxo Group Ltd Novel compounds
GB0402357D0 (en) * 2004-02-03 2004-03-10 Glaxo Group Ltd Novel compounds
GB0402355D0 (en) * 2004-02-03 2004-03-10 Glaxo Group Ltd Novel compounds
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