DE60309739D1 - Pyridinderivate als modulatoren des cb2-rezeptors - Google Patents

Pyridinderivate als modulatoren des cb2-rezeptors

Info

Publication number
DE60309739D1
DE60309739D1 DE60309739T DE60309739T DE60309739D1 DE 60309739 D1 DE60309739 D1 DE 60309739D1 DE 60309739 T DE60309739 T DE 60309739T DE 60309739 T DE60309739 T DE 60309739T DE 60309739 D1 DE60309739 D1 DE 60309739D1
Authority
DE
Germany
Prior art keywords
pyridine derivatives
receptor
modulators
diseases
indirectly
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
DE60309739T
Other languages
English (en)
Other versions
DE60309739T2 (de
Inventor
Andrew John Eatherton
Gerard Martin Paul Giblin
Howard Green
Karamjit Singh Jandu
William Leonard Mitchell
Alan Naylor
Giovanni Palombi
Derek Anthony Rawlings
Brian Peter Slingsby
Andrew Richard Whittington
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Glaxo Group Ltd
Original Assignee
Glaxo Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Application granted granted Critical
Publication of DE60309739D1 publication Critical patent/DE60309739D1/de
Publication of DE60309739T2 publication Critical patent/DE60309739T2/de
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

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    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D213/81—Amides; Imides
    • C07D213/82—Amides; Imides in position 3
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    • C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
DE60309739T 2002-09-27 2003-09-25 Pyridinderivate als modulatoren des cb2-rezeptors Expired - Fee Related DE60309739T2 (de)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GBGB0222495.4A GB0222495D0 (en) 2002-09-27 2002-09-27 Compounds
GB0222495 2002-09-27
PCT/EP2003/010935 WO2004029027A1 (en) 2002-09-27 2003-09-25 Pyridine derivatives as cb2 receptor modulators

Publications (2)

Publication Number Publication Date
DE60309739D1 true DE60309739D1 (de) 2006-12-28
DE60309739T2 DE60309739T2 (de) 2007-10-31

Family

ID=9944906

Family Applications (1)

Application Number Title Priority Date Filing Date
DE60309739T Expired - Fee Related DE60309739T2 (de) 2002-09-27 2003-09-25 Pyridinderivate als modulatoren des cb2-rezeptors

Country Status (9)

Country Link
US (1) US20070129367A1 (de)
EP (1) EP1562907B1 (de)
JP (1) JP2006508065A (de)
AT (1) ATE345329T1 (de)
AU (1) AU2003276028A1 (de)
DE (1) DE60309739T2 (de)
ES (1) ES2277149T3 (de)
GB (1) GB0222495D0 (de)
WO (1) WO2004029027A1 (de)

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TW200505902A (en) 2003-03-20 2005-02-16 Schering Corp Cannabinoid receptor ligands
EP1669348A4 (de) 2003-09-30 2009-03-11 Eisai R&D Man Co Ltd Neues antipilzmittel, das eine heterocyclische verbindung enthält
GB0402355D0 (en) * 2004-02-03 2004-03-10 Glaxo Group Ltd Novel compounds
GB0402357D0 (en) * 2004-02-03 2004-03-10 Glaxo Group Ltd Novel compounds
GB0402356D0 (en) * 2004-02-03 2004-03-10 Glaxo Group Ltd Novel compounds
US7829585B2 (en) 2005-03-30 2010-11-09 Eisai R&D Management Co., Ltd. Antifungal agent containing pyridine derivative
WO2006129609A1 (ja) * 2005-05-30 2006-12-07 Shionogi & Co., Ltd. ２－ナフチルイミノ－５，５－ジ置換－１，３－チアジン誘導体
TWI385169B (zh) 2005-10-31 2013-02-11 Eisai R&D Man Co Ltd 經雜環取代之吡啶衍生物及含有彼之抗真菌劑
WO2007118041A1 (en) * 2006-04-07 2007-10-18 Boehringer Ingelheim International Gmbh Compounds which modulate the cb2 receptor
CA2657247A1 (en) 2006-07-28 2008-01-31 Boehringer Ingelheim International Gmbh Compounds which modulate the cb2 receptor
WO2008035726A1 (fr) 2006-09-21 2008-03-27 Eisai R & D Management Co., Ltd. Dérivé de pyridine substitué par un cycle hétéroaryle, et agent antifongique le comprenant
WO2008039645A1 (en) 2006-09-25 2008-04-03 Boehringer Ingelheim International Gmbh Compounds which modulate the cb2 receptor
FR2907784B1 (fr) * 2006-10-27 2009-02-13 Sod Conseils Rech Applic Derives phenyliques et leur utilisation comme medicament
US9422235B2 (en) 2006-12-19 2016-08-23 Pharmos Corporation Sulfonamide derivatives with therapeutic indications
TW200841879A (en) 2007-04-27 2008-11-01 Eisai R&D Man Co Ltd Pyridine derivatives substituted by heterocyclic ring and phosphonoamino group, and anti-fungal agent containing same
CA2685194A1 (en) 2007-04-27 2008-11-13 Eisai R&D Management Co., Ltd. Heterocycle-substituted pyridine derivatives salt or crystal thereof
JP5300225B2 (ja) 2007-08-03 2013-09-25 バイエル・クロップサイエンス・アーゲー 除草剤トリアゾリルピリジンケトン類
EP2217565B1 (de) 2007-11-07 2013-05-22 Boehringer Ingelheim International GmbH Cb2 rezeptor-modulierende verbindungen
US8513287B2 (en) 2007-12-27 2013-08-20 Eisai R&D Management Co., Ltd. Heterocyclic ring and phosphonoxymethyl group substituted pyridine derivatives and antifungal agent containing same
JP2011520972A (ja) * 2008-05-19 2011-07-21 ユニヴァーシティ オブ テネシー リサーチ ファウンデーション，ザ ピリジンの古典的カンナビノイド化合物及び関連する使用方法
US8349876B2 (en) 2008-05-19 2013-01-08 The University Of Tennesee Research Foundation Pyridine non-classical cannabinoid compounds and related methods of use
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US20070129367A1 (en) 2007-06-07
ATE345329T1 (de) 2006-12-15
DE60309739T2 (de) 2007-10-31
EP1562907A1 (de) 2005-08-17
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ES2277149T3 (es) 2007-07-01
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