DE602005009318D1 - Kondensierte heteroyralderivate zur verwendung als p38-kinase-inhibitoren - Google Patents

Kondensierte heteroyralderivate zur verwendung als p38-kinase-inhibitoren

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Publication number
DE602005009318D1
DE602005009318D1 DE602005009318T DE602005009318T DE602005009318D1 DE 602005009318 D1 DE602005009318 D1 DE 602005009318D1 DE 602005009318 T DE602005009318 T DE 602005009318T DE 602005009318 T DE602005009318 T DE 602005009318T DE 602005009318 D1 DE602005009318 D1 DE 602005009318D1
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Germany
Prior art keywords
heteroyral
condensed
derivatives
kinase inhibitors
kinase
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Active
Application number
DE602005009318T
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English (en)
Inventor
Paul Bamborough
Sebastien Andre Campos
Vipulkumar Kantibhai Patel
Stephen Swanson
Ann Louise Walker
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
SmithKline Beecham Corp
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SmithKline Beecham Corp
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Application filed by SmithKline Beecham Corp filed Critical SmithKline Beecham Corp
Publication of DE602005009318D1 publication Critical patent/DE602005009318D1/de
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    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
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    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D413/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

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  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
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  • Engineering & Computer Science (AREA)
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  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Pain & Pain Management (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Pulmonology (AREA)
  • Rheumatology (AREA)
  • Diabetes (AREA)
  • Cardiology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Dermatology (AREA)
  • Hospice & Palliative Care (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Urology & Nephrology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Hematology (AREA)
  • Transplantation (AREA)
  • Psychiatry (AREA)
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  • Vascular Medicine (AREA)
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DE602005009318T 2004-01-30 2005-01-27 Kondensierte heteroyralderivate zur verwendung als p38-kinase-inhibitoren Active DE602005009318D1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB0402143.2A GB0402143D0 (en) 2004-01-30 2004-01-30 Novel compounds
PCT/GB2005/000265 WO2005073189A1 (en) 2004-01-30 2005-01-27 Fused heteroyral derivatives for use as p38 kinase inhibitors

Publications (1)

Publication Number Publication Date
DE602005009318D1 true DE602005009318D1 (de) 2008-10-09

Family

ID=31971803

Family Applications (1)

Application Number Title Priority Date Filing Date
DE602005009318T Active DE602005009318D1 (de) 2004-01-30 2005-01-27 Kondensierte heteroyralderivate zur verwendung als p38-kinase-inhibitoren

Country Status (8)

Country Link
US (1) US20090023725A1 (de)
EP (1) EP1708996B1 (de)
JP (1) JP2007519692A (de)
AT (1) ATE406351T1 (de)
DE (1) DE602005009318D1 (de)
ES (1) ES2313283T3 (de)
GB (1) GB0402143D0 (de)
WO (1) WO2005073189A1 (de)

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GB0402138D0 (en) 2004-01-30 2004-03-03 Smithkline Beecham Corp Novel compounds
US20090192164A1 (en) * 2006-06-28 2009-07-30 Aska Pharmaceutical Co., Ltd. Treating agent of inflammatory bowel disease
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GB0402143D0 (en) 2004-03-03
US20090023725A1 (en) 2009-01-22
WO2005073189A1 (en) 2005-08-11
EP1708996B1 (de) 2008-08-27
ES2313283T3 (es) 2009-03-01
JP2007519692A (ja) 2007-07-19
EP1708996A1 (de) 2006-10-11

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