DE60117814D1 - Nicht-imidazol aryloxyalkylamine als h3 rezeptor liganden - Google Patents

Nicht-imidazol aryloxyalkylamine als h3 rezeptor liganden

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Publication number
DE60117814D1
DE60117814D1 DE60117814T DE60117814T DE60117814D1 DE 60117814 D1 DE60117814 D1 DE 60117814D1 DE 60117814 T DE60117814 T DE 60117814T DE 60117814 T DE60117814 T DE 60117814T DE 60117814 D1 DE60117814 D1 DE 60117814D1
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Prior art keywords
aryloxyalkylamine
liganden
imidazole
receptor
formula
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Expired - Lifetime
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DE60117814T
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English (en)
Other versions
DE60117814T2 (de
Inventor
Richard Apodaca
I Carruthers
A Dvorak
A Rudolph
R Shah
Wei Xiao
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Janssen Pharmaceuticals Inc
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Ortho McNeil Pharmaceutical Inc
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Publication of DE60117814T2 publication Critical patent/DE60117814T2/de
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    • C07D207/30—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
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    • C07C217/22—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having etherified hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated having only one etherified hydroxy group and one amino group bound to the carbon skeleton, which is not further substituted the oxygen atom of the etherified hydroxy group being further bound to a carbon atom of a six-membered aromatic ring the six-membered aromatic ring or condensed ring system containing that ring being further substituted by carbon atoms having at least two bonds to oxygen atoms
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ATE319696T1 (de) 2006-03-15
EP1313721A2 (de) 2003-05-28
US7186732B2 (en) 2007-03-06
KR100819381B1 (ko) 2008-04-04
BR0113162A (pt) 2004-04-06
AU8473301A (en) 2002-02-18
JP5279161B2 (ja) 2013-09-04
HU230055B1 (hu) 2015-06-29
US20020065278A1 (en) 2002-05-30
US20100004241A1 (en) 2010-01-07
DE60117814T2 (de) 2006-11-02
DK1313721T3 (da) 2006-06-26
HUP0302959A3 (en) 2006-04-28
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BRPI0113162B8 (pt) 2021-05-25
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PL360886A1 (en) 2004-09-20
CZ2003685A3 (cs) 2003-08-13
HUP0302959A2 (hu) 2003-12-29
US20080306085A1 (en) 2008-12-11
WO2002012214A3 (en) 2002-06-20
ES2260276T3 (es) 2006-11-01
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MXPA03001267A (es) 2004-07-30
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WO2002012214A2 (en) 2002-02-14
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