DE60100810D1 - Verfahren zur präparation von pyrimidonderivaten mit fungizidder aktivität - Google Patents

Verfahren zur präparation von pyrimidonderivaten mit fungizidder aktivität

Info

Publication number
DE60100810D1
DE60100810D1 DE60100810T DE60100810T DE60100810D1 DE 60100810 D1 DE60100810 D1 DE 60100810D1 DE 60100810 T DE60100810 T DE 60100810T DE 60100810 T DE60100810 T DE 60100810T DE 60100810 D1 DE60100810 D1 DE 60100810D1
Authority
DE
Germany
Prior art keywords
pyrimidone derivatives
fungicide activity
preparing
preparing pyrimidone
fungicide
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
DE60100810T
Other languages
English (en)
Other versions
DE60100810T2 (de
Inventor
Orpi Javier Bartroli
Lopez Manuel Anguita
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Palau Pharma SA
Original Assignee
J Uriach y Cia SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by J Uriach y Cia SA filed Critical J Uriach y Cia SA
Application granted granted Critical
Publication of DE60100810D1 publication Critical patent/DE60100810D1/de
Publication of DE60100810T2 publication Critical patent/DE60100810T2/de
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/517—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with carbocyclic ring systems, e.g. quinazoline, perimidine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
DE60100810T 2000-03-07 2001-03-05 Verfahren zur präparation von pyrimidonderivaten mit fungizidder aktivität Expired - Lifetime DE60100810T2 (de)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
ES200000625A ES2159488B1 (es) 2000-03-07 2000-03-07 Procedimiento para la preparacion de derivados de pirimidona con actividad antifungica.
ES200000625 2000-03-07
PCT/ES2001/000081 WO2001066519A2 (es) 2000-03-07 2001-03-05 Procedimiento para la preparacion de derivados de pirimidona con actividad antifungica

Publications (2)

Publication Number Publication Date
DE60100810D1 true DE60100810D1 (de) 2003-10-23
DE60100810T2 DE60100810T2 (de) 2004-07-01

Family

ID=8492714

Family Applications (1)

Application Number Title Priority Date Filing Date
DE60100810T Expired - Lifetime DE60100810T2 (de) 2000-03-07 2001-03-05 Verfahren zur präparation von pyrimidonderivaten mit fungizidder aktivität

Country Status (17)

Country Link
US (1) US6653475B2 (de)
EP (1) EP1282084B9 (de)
JP (1) JP4772248B2 (de)
KR (1) KR100735583B1 (de)
AR (1) AR027607A1 (de)
AT (1) ATE250256T1 (de)
AU (1) AU2001237447A1 (de)
BR (1) BRPI0108990B8 (de)
CA (1) CA2402390C (de)
DE (1) DE60100810T2 (de)
DK (1) DK1282084T3 (de)
ES (2) ES2159488B1 (de)
HK (1) HK1052244B (de)
MX (1) MXPA02008556A (de)
NO (1) NO323314B1 (de)
PT (1) PT1282084E (de)
WO (1) WO2001066519A2 (de)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6545004B1 (en) 1999-10-27 2003-04-08 Cytokinetics, Inc. Methods and compositions utilizing quinazolinones
WO2003064399A1 (fr) * 2002-01-28 2003-08-07 Ube Industries, Ltd. Procede de production de derive de quinazolin-4-one
US7812045B2 (en) 2005-03-30 2010-10-12 Daewoong Pharmaceutical Co., Ltd. Antifungal triazole derivatives
MX2009001208A (es) * 2006-08-07 2009-04-14 Stiefel Laboratories Compuestos cristalinos antifungicos.
EP2009009A1 (de) * 2007-06-26 2008-12-31 Palau Pharma, S.A. Antifungale Kristallverbindungen
EP1887004A1 (de) * 2006-08-07 2008-02-13 Palau Pharma, S.A. Kristalline Formen von (1R,2R)-7-Chloro-3-[2-(2,4-difluorophenyl)-2-hydroxy-1-methyl-3-(1H-1,2,4-triazol-1-yl)propyl]chinazolin-4(3H)-on
TWI395728B (zh) 2006-12-06 2013-05-11 Du Pont 製備２-胺基-５-氰基苯甲酸衍生物之方法
TWI415827B (zh) 2006-12-21 2013-11-21 Du Pont 製備２-胺基-５-氰基苯甲酸衍生物之方法
WO2009109983A1 (en) 2008-03-03 2009-09-11 National Chemical Laboratory Thieno[2,3-d]-pyrimidine-4(3h)-one compounds with antifungal properties and process thereof
SE532624C2 (sv) * 2008-06-19 2010-03-09 Andritz Technology And Asset Management Gmbh Kylning av en cellulosamassabana
WO2012123952A1 (en) * 2011-03-15 2012-09-20 Fdc Limited Enantiomers of fluconazole analogues containing thieno-[2,3-d]pyrimidin-4(3h)-one moiety as antifungal agents
CN106588889B (zh) * 2016-11-25 2019-01-22 江苏恒盛药业有限公司 一种伏立康唑的制备方法
CN111018839B (zh) * 2019-12-02 2022-12-23 中国人民解放军第二军医大学 三氮唑醇类衍生物及其制备方法和应用

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8819308D0 (en) * 1988-08-13 1988-09-14 Pfizer Ltd Triazole antifungal agents
TW218017B (de) 1992-04-28 1993-12-21 Takeda Pharm Industry Co Ltd
PT783501E (pt) * 1995-08-02 2001-04-30 Uriach & Cia Sa J Derivados de pirimidona com actividade antifungica

Also Published As

Publication number Publication date
DE60100810T2 (de) 2004-07-01
CA2402390C (en) 2009-09-15
BRPI0108990B8 (pt) 2021-05-25
ES2159488A1 (es) 2001-10-01
AU2001237447A1 (en) 2001-09-17
DK1282084T3 (da) 2004-02-02
US6653475B2 (en) 2003-11-25
NO20024256L (no) 2002-09-06
ATE250256T1 (de) 2003-10-15
ES2159488B1 (es) 2002-04-16
AR027607A1 (es) 2003-04-02
CA2402390A1 (en) 2001-09-13
EP1282084B1 (de) 2003-09-17
NO323314B1 (no) 2007-03-12
HK1052244B (zh) 2003-12-19
MXPA02008556A (es) 2003-02-24
KR100735583B1 (ko) 2007-07-04
JP4772248B2 (ja) 2011-09-14
JP2004500391A (ja) 2004-01-08
HK1052244A1 (en) 2003-09-05
BR0108990B1 (pt) 2014-03-25
EP1282084B9 (de) 2005-03-02
EP1282084A2 (de) 2003-02-05
PT1282084E (pt) 2004-02-27
WO2001066519A2 (es) 2001-09-13
KR20020075809A (ko) 2002-10-05
NO20024256D0 (no) 2002-09-06
WO2001066519A3 (es) 2002-01-31
US20030064986A1 (en) 2003-04-03
BR0108990A (pt) 2003-12-30
ES2207605T3 (es) 2004-06-01

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Legal Events

Date Code Title Description
8364 No opposition during term of opposition
8328 Change in the person/name/address of the agent

Representative=s name: PFENNING MEINIG & PARTNER GBR, 80339 MUENCHEN

8327 Change in the person/name/address of the patent owner

Owner name: PALAU PHARMA,S.A., PALAU-SOLITA I PLEGAMANS, B, ES

8328 Change in the person/name/address of the agent

Representative=s name: MAIWALD PATENTANWALTSGESELLSCHAFT MBH, 80335 MUENC