DE2258973A1 - Penicilline, verfahren zu ihrer herstellung sowie ihre verwendung als arzneimittel - Google Patents

Penicilline, verfahren zu ihrer herstellung sowie ihre verwendung als arzneimittel

Info

Publication number
DE2258973A1
DE2258973A1 DE19722258973 DE2258973A DE2258973A1 DE 2258973 A1 DE2258973 A1 DE 2258973A1 DE 19722258973 DE19722258973 DE 19722258973 DE 2258973 A DE2258973 A DE 2258973A DE 2258973 A1 DE2258973 A1 DE 2258973A1
Authority
DE
Germany
Prior art keywords
conh
carbon atoms
cooh
group
methyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
DE19722258973
Other languages
German (de)
English (en)
Inventor
Hans-Bodo Dr Koenig
Karl-Georg Dr Metzger
Wilfried Dr Schroeck
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Bayer AG
Original Assignee
Bayer AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer AG filed Critical Bayer AG
Priority to DE19722258973 priority Critical patent/DE2258973A1/de
Priority to PH15218A priority patent/PH10188A/en
Priority to AU62856/73A priority patent/AU6285673A/en
Priority to BG25084A priority patent/BG20812A3/xx
Priority to IL7343708A priority patent/IL43708A/en
Priority to RO7385228A priority patent/RO72164A/ro
Priority to RO7376805A priority patent/RO65197A/ro
Priority to BE138262A priority patent/BE807918A/xx
Priority to EG452/73A priority patent/EG11062A/xx
Priority to LU68892A priority patent/LU68892A1/xx
Priority to NL7316357A priority patent/NL7316357A/xx
Priority to JP48133147A priority patent/JPS4986519A/ja
Priority to JP13314673A priority patent/JPS576435B2/ja
Priority to CH1678673A priority patent/CH601306A5/xx
Priority to SU1972067A priority patent/SU523640A3/ru
Priority to DD174978A priority patent/DD109221A5/xx
Priority to AR251293A priority patent/AR200161A1/es
Priority to GB5566873A priority patent/GB1426199A/en
Priority to ES421006A priority patent/ES421006A1/es
Priority to FR7342743A priority patent/FR2208647B1/fr
Priority to IE2174/73A priority patent/IE38560B1/xx
Priority to ZA739121A priority patent/ZA739121B/xx
Priority to AR255998A priority patent/AR205450A1/es
Publication of DE2258973A1 publication Critical patent/DE2258973A1/de
Priority to ES444389A priority patent/ES444389A1/es
Pending legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/04—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D233/28—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D233/30—Oxygen or sulfur atoms
    • C07D233/32—One oxygen atom
    • C07D233/38—One oxygen atom with acyl radicals or hetero atoms directly attached to ring nitrogen atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Cephalosporin Compounds (AREA)
  • Fodder In General (AREA)
DE19722258973 1972-12-01 1972-12-01 Penicilline, verfahren zu ihrer herstellung sowie ihre verwendung als arzneimittel Pending DE2258973A1 (de)

Priority Applications (24)

Application Number Priority Date Filing Date Title
DE19722258973 DE2258973A1 (de) 1972-12-01 1972-12-01 Penicilline, verfahren zu ihrer herstellung sowie ihre verwendung als arzneimittel
PH15218A PH10188A (en) 1972-12-01 1973-11-12 6-(l-3-acylamidoacetamido)-penicillanic acids,their pharmaceutically acceptable salts and their medicinal uses
AU62856/73A AU6285673A (en) 1972-12-01 1973-11-23 Penicillins
BG25084A BG20812A3 (zh) 1972-12-01 1973-11-27
IL7343708A IL43708A (en) 1972-12-01 1973-11-27 Penicillins their production and pharmaceutical compositions containing them
RO7385228A RO72164A (ro) 1972-12-01 1973-11-28 Procedeu pentru prepararea unor peniciline
RO7376805A RO65197A (ro) 1972-12-01 1973-11-28 Procedeu pentru prepararea unor peniciline
BE138262A BE807918A (fr) 1972-12-01 1973-11-28 Nouvelles penicillines
JP48133147A JPS4986519A (zh) 1972-12-01 1973-11-29
LU68892A LU68892A1 (zh) 1972-12-01 1973-11-29
NL7316357A NL7316357A (zh) 1972-12-01 1973-11-29
EG452/73A EG11062A (en) 1972-12-01 1973-11-29 Process for preparing of new penicillins
JP13314673A JPS576435B2 (zh) 1972-12-01 1973-11-29
CH1678673A CH601306A5 (zh) 1972-12-01 1973-11-29
SU1972067A SU523640A3 (ru) 1972-12-01 1973-11-29 Способ получени пенициллинов или их солей,или их или изомеров,или их диастереомеров
DD174978A DD109221A5 (zh) 1972-12-01 1973-11-29
GB5566873A GB1426199A (en) 1972-12-01 1973-11-30 Penicillins their production and their medicinal use
AR251293A AR200161A1 (es) 1972-12-01 1973-11-30 Procedimiento para la produccion de nuevas penicilinas
ES421006A ES421006A1 (es) 1972-12-01 1973-11-30 Procedimiento para la produccion de hidroxi-bencil penici- linas sustituidas.
FR7342743A FR2208647B1 (zh) 1972-12-01 1973-11-30
IE2174/73A IE38560B1 (en) 1972-12-01 1973-11-30 New penicillins their production and their medicinal use
ZA739121A ZA739121B (en) 1972-12-01 1973-11-30 Penicillins,processes for their manufacture and their use as medicaments
AR255998A AR205450A1 (es) 1972-12-01 1974-01-01 Procedimiento para la produccion de nuevas penicilinas
ES444389A ES444389A1 (es) 1972-12-01 1976-01-16 Procedimiento para la produccion de hidroxi-bencil-penicili-nas sustituidas.

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19722258973 DE2258973A1 (de) 1972-12-01 1972-12-01 Penicilline, verfahren zu ihrer herstellung sowie ihre verwendung als arzneimittel

Publications (1)

Publication Number Publication Date
DE2258973A1 true DE2258973A1 (de) 1974-06-06

Family

ID=5863290

Family Applications (1)

Application Number Title Priority Date Filing Date
DE19722258973 Pending DE2258973A1 (de) 1972-12-01 1972-12-01 Penicilline, verfahren zu ihrer herstellung sowie ihre verwendung als arzneimittel

Country Status (20)

Country Link
JP (2) JPS4986519A (zh)
AR (2) AR200161A1 (zh)
AU (1) AU6285673A (zh)
BE (1) BE807918A (zh)
BG (1) BG20812A3 (zh)
CH (1) CH601306A5 (zh)
DD (1) DD109221A5 (zh)
DE (1) DE2258973A1 (zh)
EG (1) EG11062A (zh)
ES (2) ES421006A1 (zh)
FR (1) FR2208647B1 (zh)
GB (1) GB1426199A (zh)
IE (1) IE38560B1 (zh)
IL (1) IL43708A (zh)
LU (1) LU68892A1 (zh)
NL (1) NL7316357A (zh)
PH (1) PH10188A (zh)
RO (2) RO65197A (zh)
SU (1) SU523640A3 (zh)
ZA (1) ZA739121B (zh)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4235774A (en) 1978-03-08 1980-11-25 Bayer Aktiengesellschaft Penicillin derivatives

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5852996B2 (ja) * 1975-03-25 1983-11-26 バイエル・アクチエンゲゼルシヤフト β−ラクタム及び抗バクテリア剤
DE2658905A1 (de) * 1976-12-24 1978-10-19 Bayer Ag Beta-lactam-antibiotica, verfahren zu ihrer herstellung sowie ihre verwendung als arzneimittel
CA1133896A (en) * 1978-05-26 1982-10-19 Nobuhiro Oi Penicillanic acid derivative and process for preparing the same
ZA795477B (en) * 1978-10-16 1981-03-25 Bristol Myers Co Antibacterial agents
JPS5732289A (en) 1980-08-05 1982-02-20 Chugai Pharmaceut Co Ltd Alpha-substituted ureidobenzylpenicillin

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE790440A (zh) * 1971-10-23 1973-04-24 Bayer Ag

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4235774A (en) 1978-03-08 1980-11-25 Bayer Aktiengesellschaft Penicillin derivatives

Also Published As

Publication number Publication date
PH10188A (en) 1976-09-23
RO72164A (ro) 1983-08-03
JPS576435B2 (zh) 1982-02-04
ES444389A1 (es) 1977-06-01
DD109221A5 (zh) 1974-10-20
SU523640A3 (ru) 1976-07-30
RO65197A (ro) 1982-09-09
IL43708A0 (en) 1974-03-14
ES421006A1 (es) 1976-07-16
IL43708A (en) 1977-02-28
RO72164B (ro) 1983-07-30
BE807918A (fr) 1974-05-28
GB1426199A (en) 1976-02-25
AR205450A1 (es) 1976-05-07
LU68892A1 (zh) 1974-02-11
IE38560L (en) 1974-06-01
AU6285673A (en) 1975-05-29
IE38560B1 (en) 1978-04-12
ZA739121B (en) 1974-10-30
JPS49116091A (zh) 1974-11-06
CH601306A5 (zh) 1978-07-14
EG11062A (en) 1977-08-15
FR2208647B1 (zh) 1977-10-28
NL7316357A (zh) 1974-06-05
BG20812A3 (zh) 1975-12-20
FR2208647A1 (zh) 1974-06-28
JPS4986519A (zh) 1974-08-19
AR200161A1 (es) 1974-10-24

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