DE10219435A1 - Substituierte Pyrazolo-pyrimidin-4-one - Google Patents

Substituierte Pyrazolo-pyrimidin-4-one

Info

Publication number
DE10219435A1
DE10219435A1 DE10219435A DE10219435A DE10219435A1 DE 10219435 A1 DE10219435 A1 DE 10219435A1 DE 10219435 A DE10219435 A DE 10219435A DE 10219435 A DE10219435 A DE 10219435A DE 10219435 A1 DE10219435 A1 DE 10219435A1
Authority
DE
Germany
Prior art keywords
fluorine
chlorine
trifluoromethyl
methyl
cyano
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
DE10219435A
Other languages
German (de)
English (en)
Inventor
Karl-Heinz Linker
Roland Andree
Dorothee Hoischen
Hans-Georg Schwarz
Mark Wilhelm Drewes
Peter Dahmen
Dieter Feucht
Rolf Pontzen
Peter Loesel
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Bayer CropScience AG
Original Assignee
Bayer CropScience AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer CropScience AG filed Critical Bayer CropScience AG
Priority to DE10219435A priority Critical patent/DE10219435A1/de
Priority to JP2004501408A priority patent/JP2005531549A/ja
Priority to AU2003224111A priority patent/AU2003224111A1/en
Priority to BR0309873-7A priority patent/BR0309873A/pt
Priority to EP03720510A priority patent/EP1504005A2/de
Priority to CA002484997A priority patent/CA2484997A1/en
Priority to US10/512,834 priority patent/US20050209251A1/en
Priority to PCT/EP2003/004137 priority patent/WO2003093269A2/de
Priority to ARP030101462A priority patent/AR039468A1/es
Publication of DE10219435A1 publication Critical patent/DE10219435A1/de
Withdrawn legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system

Landscapes

  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Dentistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Plant Pathology (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
DE10219435A 2002-05-02 2002-05-02 Substituierte Pyrazolo-pyrimidin-4-one Withdrawn DE10219435A1 (de)

Priority Applications (9)

Application Number Priority Date Filing Date Title
DE10219435A DE10219435A1 (de) 2002-05-02 2002-05-02 Substituierte Pyrazolo-pyrimidin-4-one
JP2004501408A JP2005531549A (ja) 2002-05-02 2003-04-22 置換ピラゾロ−ピリミジン−4−オン
AU2003224111A AU2003224111A1 (en) 2002-05-02 2003-04-22 Substituted pyrazolo-pyrimidine-4-ones
BR0309873-7A BR0309873A (pt) 2002-05-02 2003-04-22 Pirazolo-pirimidin-4-onas substituìdas
EP03720510A EP1504005A2 (de) 2002-05-02 2003-04-22 Substituierte pyrazolo-pyrimidin-4-one
CA002484997A CA2484997A1 (en) 2002-05-02 2003-04-22 Substituted pyrazolo-pyrimidine-4-ones
US10/512,834 US20050209251A1 (en) 2002-05-02 2003-04-22 Substituted pyrazolo-pyrimidine-4-ones
PCT/EP2003/004137 WO2003093269A2 (de) 2002-05-02 2003-04-22 Substituierte pyrazolo-pyrimidin-4-one
ARP030101462A AR039468A1 (es) 2002-05-02 2003-04-28 Pirazolo-pirimidin-4-onas sustituidas

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE10219435A DE10219435A1 (de) 2002-05-02 2002-05-02 Substituierte Pyrazolo-pyrimidin-4-one

Publications (1)

Publication Number Publication Date
DE10219435A1 true DE10219435A1 (de) 2003-11-13

Family

ID=29224943

Family Applications (1)

Application Number Title Priority Date Filing Date
DE10219435A Withdrawn DE10219435A1 (de) 2002-05-02 2002-05-02 Substituierte Pyrazolo-pyrimidin-4-one

Country Status (9)

Country Link
US (1) US20050209251A1 (https=)
EP (1) EP1504005A2 (https=)
JP (1) JP2005531549A (https=)
AR (1) AR039468A1 (https=)
AU (1) AU2003224111A1 (https=)
BR (1) BR0309873A (https=)
CA (1) CA2484997A1 (https=)
DE (1) DE10219435A1 (https=)
WO (1) WO2003093269A2 (https=)

Families Citing this family (62)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2773482B1 (fr) 1998-01-13 2001-04-20 Oreal Composition de teinture d'oxydation des fibres keratiniques et procede de teinture mettant en oeuvre cette composition
DE10238722A1 (de) 2002-08-23 2004-03-11 Bayer Ag Selektive Phosphodiesterase 9A-Inhibitoren als Arzneimittel zur Verbesserung kognitiver Prozesse
DE10238724A1 (de) 2002-08-23 2004-03-04 Bayer Ag Alkyl-substituierte Pyrazolpyrimidine
DE10238723A1 (de) 2002-08-23 2004-03-11 Bayer Ag Phenyl-substituierte Pyrazolyprimidine
MXPA05007485A (es) 2003-01-14 2006-01-30 Arena Pharm Inc Derivados de arilo y heteroarilo 1,2,3-trisubstituidos como moduladores del metabolismo y la profilaxis y tratamiento de trastornos relacionados con ello tales como diabetes e hiperglicemia.
CA2524900C (en) * 2003-05-09 2012-03-20 Bayer Healthcare Ag 6-cyclylmethyl- and 6-alkylmethyl-substituted pyrazolopyrimidines
DE102004004142A1 (de) * 2003-05-09 2004-11-25 Bayer Healthcare Ag 6-Cyclylmethyl- und 6-Alkylmethyl-substituierte Pyrazolopyrimidine
US8044060B2 (en) 2003-05-09 2011-10-25 Boehringer Ingelheim International Gmbh 6-cyclylmethyl- and 6-alkylmethyl pyrazolo[3,4-D]pyrimidines, methods for their preparation and methods for their use to treat impairments of perception, concentration learning and/or memory
DE10320785A1 (de) 2003-05-09 2004-11-25 Bayer Healthcare Ag 6-Arylmethyl-substituierte Pyrazolopyrimidine
DE10328479A1 (de) 2003-06-25 2005-01-13 Bayer Ag 6-Arylamino-5-cyano-4-pyrimidinone
DE102004001873A1 (de) 2004-01-14 2005-09-29 Bayer Healthcare Ag Cyanopyrimidinone
DOP2006000009A (es) * 2005-01-13 2006-08-15 Arena Pharm Inc Procedimiento para preparar eteres de pirazolo [3,4-d] pirimidina
WO2006134459A1 (en) * 2005-06-15 2006-12-21 Pfizer Limited Substituted arylpyrazoles
US8097712B2 (en) 2007-11-07 2012-01-17 Beelogics Inc. Compositions for conferring tolerance to viral disease in social insects, and the use thereof
JP5498392B2 (ja) * 2007-11-30 2014-05-21 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング 1,5−ジヒドロ−ピラゾロ[3,4−d]ピリミジン−4−オン誘導体及びcns障害の治療のためのpde9aモジュレーターとしてのそれらの使用
UA105362C2 (en) * 2008-04-02 2014-05-12 Бьорингер Ингельхайм Интернациональ Гмбх 1-heterocyclyl-1, 5-dihydro-pyrazolo [3, 4-d] pyrimidin-4-one derivatives and their use as pde9a modulators
JP5453431B2 (ja) 2008-09-08 2014-03-26 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング ピラゾロピリミジン及びcns障害の治療のためのそれらの使用
PE20120505A1 (es) 2009-03-31 2012-05-09 Boehringer Ingelheim Int Derivados de 1-heterociclil-1,5-dihidro-pirazolo[3,4-d]pirimidin-4-ona como moduladores de pde9a
AR077859A1 (es) * 2009-08-12 2011-09-28 Boehringer Ingelheim Int Compuestos para el tratamiento de trastornos del snc
US8962584B2 (en) 2009-10-14 2015-02-24 Yissum Research Development Company Of The Hebrew University Of Jerusalem, Ltd. Compositions for controlling Varroa mites in bees
SG10201906876PA (en) 2010-01-27 2019-09-27 Arena Pharm Inc Processes for the preparation of (r)-2-(7-(4-cyclopentyl-3-(trifluoromethyl)benzyloxy)-1,2,3,4-tetrahydrocyclopenta[b]indol-3-yl)acetic acid and salts thereof
ES2641642T3 (es) 2010-03-08 2017-11-10 Monsanto Technology Llc Moléculas de polinucleótido para regulación génica en plantas
AP2012006631A0 (en) 2010-08-12 2012-12-31 Boehringer Ingelheim Int 6-Cycloalkyl-1, 5-dihydro-pyrazolo[3,4-D] pyrimidin-4-one derivatives and their use as PDE9A inhibitors
PH12013500547A1 (en) 2010-09-22 2013-06-10 Arena Pharm Inc Modulators of the gpr119 receptor and the treatment of disorders related thereto
US8809345B2 (en) 2011-02-15 2014-08-19 Boehringer Ingelheim International Gmbh 6-cycloalkyl-pyrazolopyrimidinones for the treatment of CNS disorders
US10760086B2 (en) 2011-09-13 2020-09-01 Monsanto Technology Llc Methods and compositions for weed control
CN103930549B (zh) 2011-09-13 2020-09-18 孟山都技术公司 用于杂草控制的方法和组合物
EP2756085B1 (en) 2011-09-13 2019-03-20 Monsanto Technology LLC Methods and compositions for weed control
US10806146B2 (en) 2011-09-13 2020-10-20 Monsanto Technology Llc Methods and compositions for weed control
MX361938B (es) 2011-09-13 2018-12-19 Monsanto Technology Llc Métodos y composiciones para el control de malezas.
EP3382027A3 (en) 2011-09-13 2018-10-31 Monsanto Technology LLC Methods and compositions for weed control
CA2848695A1 (en) 2011-09-13 2013-03-21 Monsanto Technology Llc Methods and composition for weed control comprising inhibiting ppg oxidase
WO2013040057A1 (en) 2011-09-13 2013-03-21 Monsanto Technology Llc Methods and compositions for weed control
US10829828B2 (en) 2011-09-13 2020-11-10 Monsanto Technology Llc Methods and compositions for weed control
MX348495B (es) 2011-09-13 2017-06-14 Monsanto Technology Llc Metodos y composiciones para el control de malezas.
MX360866B (es) 2012-05-24 2018-11-09 A B Seeds Ltd Composiciones y métodos para silenciar la expresión genética.
UY35252A (es) 2013-01-01 2014-07-31 Seeds Ltd Ab MÉTODOS PARA INTRODUCIR dsRNA EN SEMILLAS DE PLANTAS PARA MODULAR LA EXPRESIÓN GENÉTICA
US10683505B2 (en) 2013-01-01 2020-06-16 Monsanto Technology Llc Methods of introducing dsRNA to plant seeds for modulating gene expression
AU2014224784B2 (en) * 2013-03-07 2018-03-08 F. Hoffmann-La Roche Ag Novel pyrazol derivatives
US10612019B2 (en) 2013-03-13 2020-04-07 Monsanto Technology Llc Methods and compositions for weed control
BR112015023051A2 (pt) 2013-03-13 2017-11-14 Monsanto Technology Llc método para controle de ervas daninhas, composição herbicida, cassete de expressão microbiano e método de produção de polinucleotídeo
US10568328B2 (en) 2013-03-15 2020-02-25 Monsanto Technology Llc Methods and compositions for weed control
AU2014261585B2 (en) 2013-05-02 2018-03-08 F. Hoffmann-La Roche Ag Purine derivatives as CB2 receptor agonists
WO2014177527A1 (en) 2013-05-02 2014-11-06 F. Hoffmann-La Roche Ag Pyrrolo[2,3-d]pyrimidine derivatives as cb2 receptor agonists
US9850496B2 (en) 2013-07-19 2017-12-26 Monsanto Technology Llc Compositions and methods for controlling Leptinotarsa
EP3030663B1 (en) 2013-07-19 2019-09-04 Monsanto Technology LLC Compositions and methods for controlling leptinotarsa
AU2014341879B2 (en) 2013-11-04 2020-07-23 Greenlight Biosciences, Inc. Compositions and methods for controlling arthropod parasite and pest infestations
UA119253C2 (uk) 2013-12-10 2019-05-27 Біолоджикс, Інк. Спосіб боротьби із вірусом у кліща varroa та у бджіл
WO2015108982A2 (en) 2014-01-15 2015-07-23 Monsanto Technology Llc Methods and compositions for weed control using epsps polynucleotides
WO2015135843A1 (de) * 2014-03-10 2015-09-17 Bayer Cropscience Ag Heterocylische verbindungen als schädlingsbekämpfungsmittel
WO2015153339A2 (en) 2014-04-01 2015-10-08 Monsanto Technology Llc Compositions and methods for controlling insect pests
CN106795515B (zh) 2014-06-23 2021-06-08 孟山都技术公司 用于经由rna干扰调控基因表达的组合物和方法
US11807857B2 (en) 2014-06-25 2023-11-07 Monsanto Technology Llc Methods and compositions for delivering nucleic acids to plant cells and regulating gene expression
CN106604993A (zh) 2014-07-29 2017-04-26 孟山都技术公司 用于控制昆虫害虫的组合物和方法
MX386419B (es) 2015-01-06 2025-03-18 Arena Pharm Inc Metodos de condiciones de tratamiento relacionadas con el receptor s1p1.
CN108064288B (zh) 2015-01-22 2021-11-26 孟山都技术公司 用于控制叶甲属的组合物和方法
EP3302053B1 (en) 2015-06-02 2021-03-17 Monsanto Technology LLC Compositions and methods for delivery of a polynucleotide into a plant
WO2016196782A1 (en) 2015-06-03 2016-12-08 Monsanto Technology Llc Methods and compositions for introducing nucleic acids into plants
EP3939965A1 (en) 2015-06-22 2022-01-19 Arena Pharmaceuticals, Inc. Crystalline l-arginine salt of (r)-2-(7-(4-cyclopentyl-3-(trifluoromethyl)benzyloxy)-1,2,3,4-tetrahydrocyclo-penta[b]indol-3-yl)acetic acid for use in sipi receptor-associated disorders
MA47504A (fr) 2017-02-16 2019-12-25 Arena Pharm Inc Composés et méthodes de traitement de l'angiocholite biliaire primitive
ES2987794T3 (es) 2018-06-06 2024-11-18 Arena Pharm Inc Procedimientos de tratamiento de afecciones relacionadas con el receptor S1P1
CN110317204B (zh) * 2019-08-02 2022-02-08 安徽农业大学 吡唑并嘧啶酮类衍生物及其制备方法和应用

Family Cites Families (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2925418A (en) * 1960-02-16 Certificate of correction
GB1406412A (en) * 1974-03-04 1975-09-17 Pfizer Pyrimidinones and process for preparing them
US4496390A (en) * 1980-02-26 1985-01-29 May & Baker Limited N-Phenylpyrazole derivatives
JPS57167902A (en) * 1981-04-08 1982-10-16 Otsuka Chem Co Ltd Herbicidal composition
MA19539A1 (fr) * 1981-07-17 1983-04-01 May & Baker Ltd N Acylaminophenylpyrazoles
DE3420985A1 (de) * 1983-10-15 1985-04-25 Bayer Ag, 5090 Leverkusen Substituierte 5-acylamino-1-phenylpyrazole
DE3520331A1 (de) * 1985-06-07 1986-12-11 Bayer Ag, 5090 Leverkusen 1-aryl-5-alkoximinoalkylamino-pyrazole
DE3625686A1 (de) * 1986-07-30 1988-02-04 Bayer Ag 4-cyano(nitro)-5-oxy(thio)-pyrazol-derivate
US5167691A (en) * 1991-10-03 1992-12-01 Fmc Corporation Herbicidal 5-amino-1-phenyl pyrazole compounds
IL103678A (en) * 1991-11-13 1996-09-12 Schering Ag History of pyrazolylpyrazole, processes for their preparation and herbicidal preparations containing them
US5198014A (en) * 1991-11-20 1993-03-30 Fmc Corporation Herbicidal beta-pyrazolylacrylic acid compound
US5250504A (en) * 1991-11-20 1993-10-05 Fmc Corporation Herbicidal β-pyrazolylacrylic acids
DK0663913T3 (da) * 1992-10-12 1999-05-03 Hoechst Schering Agrevo Gmbh Nye substituerede pyrazolderivater, fremgangsmåder til deres fremstilling samt deres anvendelse som herbicider
TW370529B (en) * 1992-12-17 1999-09-21 Pfizer Pyrazolopyrimidines
DE19530606A1 (de) * 1995-08-21 1997-02-27 Basf Ag 1-(Pyridyl)-pyrazole
DE19623892A1 (de) * 1996-06-06 1997-12-11 Hoechst Schering Agrevo Gmbh Substituierte Pyrazolyl-pyrazolderivate

Also Published As

Publication number Publication date
WO2003093269A2 (de) 2003-11-13
AU2003224111A1 (en) 2003-11-17
WO2003093269A3 (de) 2004-04-08
JP2005531549A (ja) 2005-10-20
US20050209251A1 (en) 2005-09-22
CA2484997A1 (en) 2003-11-13
BR0309873A (pt) 2005-04-26
AR039468A1 (es) 2005-02-23
EP1504005A2 (de) 2005-02-09

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Legal Events

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8139 Disposal/non-payment of the annual fee