DD91496B3 - Verfahren zur herstellung neuer penicilline - Google Patents

Verfahren zur herstellung neuer penicilline Download PDF

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Publication number
DD91496B3
DD91496B3 DD71155308A DD15530871A DD91496B3 DD 91496 B3 DD91496 B3 DD 91496B3 DD 71155308 A DD71155308 A DD 71155308A DD 15530871 A DD15530871 A DD 15530871A DD 91496 B3 DD91496 B3 DD 91496B3
Authority
DD
German Democratic Republic
Prior art keywords
parts
acid
weight
methyl
benzylpenicillin
Prior art date
Application number
DD71155308A
Other languages
German (de)
English (en)
Other versions
DD91496A5 (de
Inventor
Hans B Koenig
Wilfried Schroeck
Hans Disselnkoetter
Karl G Metzger
Original Assignee
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Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from DE2025415A external-priority patent/DE2025415C3/de
Priority claimed from DE19712104579 external-priority patent/DE2104579C3/de
Application filed by �������@������������@��k�� filed Critical �������@������������@��k��
Publication of DD91496A5 publication Critical patent/DD91496A5/xx
Publication of DD91496B3 publication Critical patent/DD91496B3/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D261/00Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
    • C07D261/02Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings
    • C07D261/06Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members
    • C07D261/10Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D261/18Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C275/00Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups
    • C07C275/46Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups containing any of the groups, X being a hetero atom, Y being any atom, e.g. acylureas
    • C07C275/58Y being a hetero atom
    • C07C275/60Y being an oxygen atom, e.g. allophanic acids
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/04Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D233/28Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D233/30Oxygen or sulfur atoms
    • C07D233/32One oxygen atom
    • C07D233/38One oxygen atom with acyl radicals or hetero atoms directly attached to ring nitrogen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D333/00Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/06Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring carbon atoms
    • C07D333/24Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D333/00Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/26Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D333/38Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F7/00Compounds containing elements of Groups 4 or 14 of the Periodic Table
    • C07F7/02Silicon compounds
    • C07F7/08Compounds having one or more C—Si linkages
    • C07F7/10Compounds having one or more C—Si linkages containing nitrogen having a Si-N linkage

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Cephalosporin Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
DD71155308A 1970-05-25 1971-05-24 Verfahren zur herstellung neuer penicilline DD91496B3 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE2025415A DE2025415C3 (de) 1970-05-25 1970-05-25 Verfahren zur Herstellung von cyclischen Acylureido-Penicillinen
DE19712104579 DE2104579C3 (de) 1971-02-01 1971-02-01 Cyclische Acylureidopenicilline und sie enthaltende Arzneimittel

Publications (2)

Publication Number Publication Date
DD91496A5 DD91496A5 (de) 1972-07-20
DD91496B3 true DD91496B3 (de) 1988-01-27

Family

ID=25759180

Family Applications (1)

Application Number Title Priority Date Filing Date
DD71155308A DD91496B3 (de) 1970-05-25 1971-05-24 Verfahren zur herstellung neuer penicilline

Country Status (26)

Country Link
JP (1) JPS55390B1 (cs)
AT (1) AT306924B (cs)
BE (1) BE767648A (cs)
BG (1) BG23753A3 (cs)
CA (1) CA932722A (cs)
CH (1) CH571524A5 (cs)
CS (1) CS185564B2 (cs)
CY (1) CY830A (cs)
DD (1) DD91496B3 (cs)
DK (1) DK134438C (cs)
EG (1) EG10490A (cs)
ES (4) ES391533A1 (cs)
FI (1) FI54485C (cs)
FR (1) FR2100682B1 (cs)
GB (1) GB1301962A (cs)
IE (1) IE35404B1 (cs)
IL (1) IL36904A (cs)
KE (1) KE2591A (cs)
LU (1) LU63204A1 (cs)
NL (1) NL172659C (cs)
NO (1) NO141759C (cs)
PH (1) PH12110A (cs)
RO (1) RO59290A (cs)
SE (1) SE395895B (cs)
SU (1) SU420181A3 (cs)
YU (1) YU35889B (cs)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2260118C2 (de) * 1972-12-08 1982-06-03 Bayer Ag, 5090 Leverkusen Penicilline sowie ihre Verwendung als Arzneimittel
US4039673A (en) 1973-10-30 1977-08-02 Bayer Aktiengesellschaft Penicillins and cephalosporins and their production
DE2354219A1 (de) * 1973-10-30 1975-05-07 Bayer Ag Beta-lactam-antibiotica, ein verfahren zu ihrer herstellung sowie ihre verwendung als arzneimittel
GB1486349A (en) * 1974-11-28 1977-09-21 Bayer Ag Beta-lactam antibiotics process for their preparation and their use as medicaments
GB1584400A (en) * 1976-12-24 1981-02-11 Bayer Ag (2-oxo-imidazoliden-1-yl(carbonylamino)-acetamido-cephalosporins and penicillins
KR860000300B1 (ko) * 1983-12-19 1986-03-31 보령제약 주식회사 아실우레이도 페니실린 유도체의 제조방법

Also Published As

Publication number Publication date
IE35404L (en) 1971-11-25
CY830A (en) 1976-03-19
ES411675A1 (es) 1976-01-01
GB1301962A (cs) 1973-01-04
IL36904A (en) 1975-11-25
FR2100682B1 (cs) 1975-01-17
CS185564B2 (en) 1978-10-31
EG10490A (en) 1976-08-31
NL7107176A (cs) 1971-11-29
CA932722A (en) 1973-08-28
DK134438C (da) 1977-05-31
ES411674A1 (es) 1976-01-01
CH571524A5 (cs) 1976-01-15
NL172659C (nl) 1983-10-03
ES391533A1 (es) 1974-08-01
IE35404B1 (en) 1976-02-04
LU63204A1 (cs) 1971-09-01
JPS55390B1 (cs) 1980-01-08
BG23753A3 (en) 1977-10-12
NO141759B (no) 1980-01-28
NL172659B (nl) 1983-05-02
FI54485B (fi) 1978-08-31
YU35889B (en) 1981-08-31
YU129671A (en) 1981-02-28
BE767648A (fr) 1971-11-25
PH12110A (en) 1978-11-02
RO59290A (cs) 1976-03-15
FI54485C (fi) 1978-12-11
ES411676A1 (es) 1976-01-01
DD91496A5 (de) 1972-07-20
FR2100682A1 (cs) 1972-03-24
DK134438B (da) 1976-11-08
SE395895B (sv) 1977-08-29
IL36904A0 (en) 1971-07-28
KE2591A (en) 1976-01-09
AT306924B (de) 1973-04-25
NO141759C (no) 1980-05-07
SU420181A3 (ru) 1974-03-15

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