DD296923A5 - Piperidinylbenzimidazoderivate, verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneipraeperate - Google Patents

Piperidinylbenzimidazoderivate, verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneipraeperate Download PDF

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Publication number
DD296923A5
DD296923A5 DD90343200A DD34320090A DD296923A5 DD 296923 A5 DD296923 A5 DD 296923A5 DD 90343200 A DD90343200 A DD 90343200A DD 34320090 A DD34320090 A DD 34320090A DD 296923 A5 DD296923 A5 DD 296923A5
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DD
German Democratic Republic
Prior art keywords
formula
choh
compounds
reaction
meaning
Prior art date
Application number
DD90343200A
Other languages
German (de)
English (en)
Inventor
Albert A Carr
John M Kane
Francis P Miller
Original Assignee
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Publication of DD296923A5 publication Critical patent/DD296923A5/de

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

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  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
DD90343200A 1989-08-03 1990-08-02 Piperidinylbenzimidazoderivate, verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneipraeperate DD296923A5 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US38903689A 1989-08-03 1989-08-03

Publications (1)

Publication Number Publication Date
DD296923A5 true DD296923A5 (de) 1991-12-19

Family

ID=23536563

Family Applications (1)

Application Number Title Priority Date Filing Date
DD90343200A DD296923A5 (de) 1989-08-03 1990-08-02 Piperidinylbenzimidazoderivate, verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneipraeperate

Country Status (9)

Country Link
EP (1) EP0411631B1 (es)
JP (1) JP2954992B2 (es)
AT (1) ATE104294T1 (es)
AU (1) AU625238B2 (es)
CA (1) CA2022451C (es)
DD (1) DD296923A5 (es)
DE (1) DE69008069T2 (es)
DK (1) DK0411631T3 (es)
ES (1) ES2055241T3 (es)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4908372A (en) * 1988-10-13 1990-03-13 Merrell Dow Pharmaceuticals Inc. Antihistaminic piperidinyl benzimidazoles
EP0561973A1 (en) * 1990-12-14 1993-09-29 Merrell Dow Pharmaceuticals Inc. Antiallergic compounds
ATE171447T1 (de) * 1993-03-18 1998-10-15 Merck Sharp & Dohme Benzimidazole derivate
GB9305644D0 (en) * 1993-03-18 1993-05-05 Merck Sharp & Dohme Therapeutic agents
GB9306578D0 (en) * 1993-03-30 1993-05-26 Merck Sharp & Dohme Therapeutic agents
US5814644A (en) * 1993-04-15 1998-09-29 Merck Sharp & Dohme, Ltd. Indole derivatives as dopamine D4 antagonists
EP2473488A4 (en) * 2009-09-04 2013-07-17 Zalicus Pharmaceuticals Ltd SUBSTITUTED HETEROCYCLIC DERIVATIVES FOR THE TREATMENT OF PAIN AND EPILEPSY
US10208023B2 (en) 2013-03-01 2019-02-19 Mark G. DeGiacomo Heterocyclic inhibitors of the sodium channel

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PH23995A (en) * 1984-01-09 1990-02-09 Janssen Pharmaceutica Nv 4((bicycle heterocyclyl)-methyl and hetero)piperidines
US4908372A (en) * 1988-10-13 1990-03-13 Merrell Dow Pharmaceuticals Inc. Antihistaminic piperidinyl benzimidazoles

Also Published As

Publication number Publication date
ES2055241T3 (es) 1994-08-16
CA2022451C (en) 2001-01-23
JP2954992B2 (ja) 1999-09-27
DE69008069D1 (de) 1994-05-19
DK0411631T3 (da) 1994-05-16
CA2022451A1 (en) 1991-02-04
ATE104294T1 (de) 1994-04-15
EP0411631B1 (en) 1994-04-13
JPH0366683A (ja) 1991-03-22
DE69008069T2 (de) 1994-07-28
AU6012390A (en) 1991-02-07
EP0411631A1 (en) 1991-02-06
AU625238B2 (en) 1992-07-02

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Legal Events

Date Code Title Description
IF04 In force in the year 2004

Expiry date: 20100803