DD266502A5 - Verwendung von beta-lactamverbindungen - Google Patents

Verwendung von beta-lactamverbindungen Download PDF

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Publication number
DD266502A5
DD266502A5 DD86311493A DD31149386A DD266502A5 DD 266502 A5 DD266502 A5 DD 266502A5 DD 86311493 A DD86311493 A DD 86311493A DD 31149386 A DD31149386 A DD 31149386A DD 266502 A5 DD266502 A5 DD 266502A5
Authority
DD
German Democratic Republic
Prior art keywords
mol
yield
optionally substituted
mmol
amino
Prior art date
Application number
DD86311493A
Other languages
German (de)
English (en)
Inventor
Gunter Schmidt
Hans-Joachim Zeitler
Karl G Metzger
Original Assignee
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Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by ������@������������k�� filed Critical ������@������������k��
Publication of DD266502A5 publication Critical patent/DD266502A5/de

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14—Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/59—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3 with hetero atoms directly attached in position 3
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • A—HUMAN NECESSITIES
    • A23—FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
    • A23K—FODDER
    • A23K20/00—Accessory food factors for animal feeding-stuffs
    • A23K20/10—Organic substances
    • A23K20/195—Antibiotics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Polymers & Plastics (AREA)
  • Health & Medical Sciences (AREA)
  • Animal Husbandry (AREA)
  • Zoology (AREA)
  • Engineering & Computer Science (AREA)
  • Food Science & Technology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Oncology (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Cephalosporin Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Hydrogenated Pyridines (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Fodder In General (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
DD86311493A 1985-03-08 1986-03-06 Verwendung von beta-lactamverbindungen DD266502A5 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19853508258 DE3508258A1 (de) 1985-03-08 1985-03-08 Ss-lactamantibiotika, verfahren zur herstellung und ihre verwendung als und in arzneimitteln

Publications (1)

Publication Number Publication Date
DD266502A5 true DD266502A5 (de) 1989-04-05

Family

ID=6264592

Family Applications (2)

Application Number Title Priority Date Filing Date
DD86311493A DD266502A5 (de) 1985-03-08 1986-03-06 Verwendung von beta-lactamverbindungen
DD86287635A DD251751A5 (de) 1985-03-08 1986-03-06 Verfahren zur herstellung von beta-lactamverbindungen

Family Applications After (1)

Application Number Title Priority Date Filing Date
DD86287635A DD251751A5 (de) 1985-03-08 1986-03-06 Verfahren zur herstellung von beta-lactamverbindungen

Country Status (20)

Country Link
US (2) US4748163A (es)
EP (1) EP0195947B1 (es)
JP (1) JPH0649708B2 (es)
KR (1) KR930007420B1 (es)
AT (1) ATE137238T1 (es)
AU (1) AU594941B2 (es)
CA (1) CA1281315C (es)
DD (2) DD266502A5 (es)
DE (2) DE3508258A1 (es)
DK (1) DK105286A (es)
ES (1) ES8800234A1 (es)
FI (1) FI85708C (es)
GR (1) GR860626B (es)
HU (1) HU200183B (es)
IE (1) IE860598L (es)
IL (1) IL78042A0 (es)
NO (1) NO165108C (es)
PH (1) PH24000A (es)
PT (1) PT82143B (es)
ZA (1) ZA861713B (es)

Families Citing this family (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3509618A1 (de) * 1985-03-16 1986-09-18 Bayer Ag, 5090 Leverkusen Ss-lactam-antibiotika, verfahren zur herstellung und ihre verwendung als arzneimittel
DE3734005A1 (de) * 1987-05-26 1988-12-15 Bayer Ag Substituierte vinylcephalosporine, verfahren zu ihrer herstellung und ihre verwendung als arzneimittel
AU637400B2 (en) * 1987-05-26 1993-05-27 Bayer Aktiengesellschaft Substituted vinylcephalosporins, processes for their preparation and their use as medicaments
DE3734004A1 (de) * 1987-05-26 1988-12-15 Bayer Ag Substituierte vinylcephalosporine, verfahren zu ihrer herstellung und ihre verwendung als arzneimittel
US5171854A (en) * 1987-05-26 1992-12-15 Bayer Aktiengesellschaft Substituted vinylcephalosporins
DE3733626A1 (de) * 1987-10-05 1989-04-13 Bayer Ag Heteroanellierte phenylglycin-(beta)-lactam-antibiotika, verfahren zu ihrer herstellung und ihre verwendung als arzneimittel
DE3803169A1 (de) 1988-02-03 1989-08-17 Bayer Ag Ss-lactam-antibiotika, verfahren zu ihrer herstellung und ihre verwendung als und in arzneimitteln
WO1994006804A1 (en) * 1992-09-18 1994-03-31 Otsuka Kagaku Kabushiki Kaisha Cephem compound, process for producing the same, and medicine containing the same
US5604222A (en) * 1993-12-27 1997-02-18 Lupin Laboratories, Ltd. Method for the preparation of 2-chloro sulfinyl azetidinones
US5578721A (en) * 1994-07-11 1996-11-26 Lupin Laboratories Limited Process for preparation of 3-exomethylene cepham sulfoxide esters
DE4443892A1 (de) * 1994-12-09 1996-06-13 Bayer Ag 4-(Chinolin-2-yl-methoxy)-phenyl-essigsäurederivate
EP1531820A1 (en) 2002-08-30 2005-05-25 Memory Pharmaceuticals Corporation Anabaseine derivatives useful in the treatment of neurodegenerative diseases
CA2653933C (en) * 2006-05-31 2013-10-08 Toyama Chemical Co., Ltd. Anti-foot-and-mouth disease virus agent for animal belonging to family suidae or sheep, and method for prevention or treatment of foot-and-mouth disease in animal belonging to family suidae or sheep
CA2895905A1 (en) 2012-12-21 2014-06-26 Zenith Epigenetics Corp. Novel heterocyclic compounds as bromodomain inhibitors
US9636328B2 (en) * 2013-06-21 2017-05-02 Zenith Epigenetics Ltd. Substituted bicyclic compounds as bromodomain inhibitors
BR112015031073B1 (pt) 2013-06-21 2022-11-29 Zenith Epigenetics Ltd Compostos inibidores bicíclicos de bromodomínio e composição farmacêutica contendo os referidos compostos
KR20160038008A (ko) 2013-07-31 2016-04-06 제니쓰 에피제네틱스 코포레이션 브로모도메인 억제제로서 신규 퀴나졸리논
US10710992B2 (en) 2014-12-01 2020-07-14 Zenith Epigenetics Ltd. Substituted pyridinones as bromodomain inhibitors
US10179125B2 (en) 2014-12-01 2019-01-15 Zenith Epigenetics Ltd. Substituted pyridines as bromodomain inhibitors
WO2016092375A1 (en) 2014-12-11 2016-06-16 Zenith Epigenetics Corp. Substituted heterocycles as bromodomain inhibitors
US10231953B2 (en) 2014-12-17 2019-03-19 Zenith Epigenetics Ltd. Inhibitors of bromodomains

Family Cites Families (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3080356A (en) * 1960-06-15 1963-03-05 Beecham Res Lab Process for the production of synthetic penicillins
SE302125B (es) * 1961-03-23 1968-07-08 Bristol Myers Co
GB1174335A (en) * 1967-03-07 1969-12-17 Lilly Co Eli 7-Alpha-Amino-3-Methyl Cephalosporin Analogues, Pharmaceutical Compositions comprising the same and processes for preparing the same
YU36970B (en) * 1973-02-23 1984-08-31 Lilly Co Eli Process for obtaining 7-(amino)-acylamido-3-halocephalosporins
IL52144A (en) * 1976-07-01 1979-10-31 Lilly Co Eli De-esterification process for -lactam antibiotic esters
DE2831568C2 (de) * 1977-07-23 1985-01-10 Toyama Chemical Co. Ltd., Tokio / Tokyo 7α-Methoxycephalosporine und Verfahren zur Herstellung derselben
US4138397A (en) * 1978-02-27 1979-02-06 Richardson-Merrell Inc. 6-(2,3-Dihydro-5-benzofuranyl)acetamido penicillin derivatives
US4229575A (en) * 1978-02-27 1980-10-21 Richardson-Merrell Inc. 7-(2,3-Dihydrobenzo-5-furanyl)-acetamido cephalosporin derivatives
US4219648A (en) * 1978-03-06 1980-08-26 Richardson-Merrell Inc. 7-[[Amino(1,3-dihydrobenzo[c]thienyl)acetyl]amino]cephalosporin derivatives
US4461767A (en) * 1978-06-16 1984-07-24 E. R. Squibb & Sons, Inc. Iminothiazolyl ureido cephalosporins
US4317775A (en) * 1980-01-07 1982-03-02 Hoffmann-La Roche Inc. Amoxicillin derivatives
FR2511375A1 (fr) * 1981-08-17 1983-02-18 Rhone Poulenc Sante Nouveaux derives de la cephalosporine, leur preparation et les medicaments qui les contiennent
US4537886A (en) * 1982-03-31 1985-08-27 Beecham Group P.L.C. β-lactam antibacterial agents and compositions containing them
US4501741A (en) * 1983-04-12 1985-02-26 Eli Lilly And Company Cephalosporin antibiotics

Also Published As

Publication number Publication date
IL78042A0 (en) 1986-07-31
NO165108C (no) 1990-12-27
CA1281315C (en) 1991-03-12
KR930007420B1 (ko) 1993-08-10
ES552683A0 (es) 1987-11-01
AU5443086A (en) 1986-09-11
DK105286D0 (da) 1986-03-07
EP0195947B1 (de) 1996-04-24
DE3508258A1 (de) 1986-09-18
ZA861713B (en) 1986-11-26
ES8800234A1 (es) 1987-11-01
USRE33948E (en) 1992-06-02
AU594941B2 (en) 1990-03-22
GR860626B (en) 1986-07-07
JPS61207388A (ja) 1986-09-13
EP0195947A2 (de) 1986-10-01
KR860007265A (ko) 1986-10-10
PT82143B (pt) 1988-07-29
DD251751A5 (de) 1987-11-25
FI85708C (fi) 1992-05-25
NO165108B (no) 1990-09-17
JPH0649708B2 (ja) 1994-06-29
US4748163A (en) 1988-05-31
FI85708B (fi) 1992-02-14
PT82143A (en) 1986-04-01
EP0195947A3 (en) 1988-05-04
FI860945A0 (fi) 1986-03-06
FI860945A (fi) 1986-09-09
PH24000A (en) 1990-02-09
DE3650518D1 (de) 1996-05-30
NO860679L (no) 1986-09-09
DK105286A (da) 1986-09-09
HUT41031A (en) 1987-03-30
ATE137238T1 (de) 1996-05-15
IE860598L (en) 1986-09-08
HU200183B (en) 1990-04-28

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ENJ Ceased due to non-payment of renewal fee