DD213927A5 - Verfahren zur herstellung von (3-benzothienyl)-glycylamidocephalosporin-derivaten - Google Patents
Verfahren zur herstellung von (3-benzothienyl)-glycylamidocephalosporin-derivaten Download PDFInfo
- Publication number
- DD213927A5 DD213927A5 DD84261874A DD26187484A DD213927A5 DD 213927 A5 DD213927 A5 DD 213927A5 DD 84261874 A DD84261874 A DD 84261874A DD 26187484 A DD26187484 A DD 26187484A DD 213927 A5 DD213927 A5 DD 213927A5
- Authority
- DD
- German Democratic Republic
- Prior art keywords
- formula
- hydrogen
- benzothienyl
- compound
- methyl
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- C07D501/14—Compounds having a nitrogen atom directly attached in position 7
- C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
- C07D501/59—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3 with hetero atoms directly attached in position 3
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
- C07D333/52—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
- C07D333/54—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
- C07D333/56—Radicals substituted by oxygen atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
- C07D333/52—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
- C07D333/54—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
- C07D333/60—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Cephalosporin Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US06/484,129 US4492693A (en) | 1983-04-12 | 1983-04-12 | Benzothienylglycyl cephalosporin derivatives |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DD213927A5 true DD213927A5 (de) | 1984-09-26 |
Family
ID=23922870
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DD84261874A DD213927A5 (de) | 1983-04-12 | 1984-04-11 | Verfahren zur herstellung von (3-benzothienyl)-glycylamidocephalosporin-derivaten |
Country Status (23)
| Country | Link |
|---|---|
| US (1) | US4492693A (xx) |
| EP (1) | EP0122154A3 (xx) |
| JP (1) | JPS59199692A (xx) |
| KR (1) | KR840008654A (xx) |
| AU (1) | AU2673684A (xx) |
| CA (1) | CA1212938A (xx) |
| CS (1) | CS243485B2 (xx) |
| DD (1) | DD213927A5 (xx) |
| DK (1) | DK187384A (xx) |
| ES (1) | ES531531A0 (xx) |
| FI (1) | FI841437A (xx) |
| GB (1) | GB2137995A (xx) |
| GR (1) | GR79908B (xx) |
| GT (1) | GT198400056A (xx) |
| IL (1) | IL71497A0 (xx) |
| MA (1) | MA20093A1 (xx) |
| NO (1) | NO841441L (xx) |
| OA (1) | OA07701A (xx) |
| PL (1) | PL247170A1 (xx) |
| PT (1) | PT78403A (xx) |
| RO (1) | RO88220B (xx) |
| ZA (1) | ZA842694B (xx) |
| ZW (1) | ZW4384A1 (xx) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4581352A (en) * | 1984-12-03 | 1986-04-08 | Eli Lilly And Company | Thienothienylglycyl cephalosporin derivatives |
| US4692587A (en) * | 1986-02-19 | 1987-09-08 | Spirk Jr John W | Hand tool and support |
| EP1451147A4 (en) * | 2001-07-24 | 2007-06-06 | Pharmacore Inc | AMINO ACID DERIVATIVES |
| CN103588790A (zh) * | 2013-11-29 | 2014-02-19 | 中国科学院长春应用化学研究所 | 7-氨基-3-氯-3-头孢-4-羧酸-对硝基苄基酯的制备方法 |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE1445685A1 (de) * | 1961-09-11 | 1968-12-05 | Lilly Co Eli | Antibiotisch wirksame Cephalospransaeurederivate und Verfahren zu ihrer Herstellung |
| US3560489A (en) * | 1966-08-12 | 1971-02-02 | Lilly Co Eli | 7-alpha-aminoacyl cephalosporins |
| US3575969A (en) * | 1968-03-04 | 1971-04-20 | Lilly Co Eli | Desacetoxycephalosporin antibiotics |
| US4024133A (en) * | 1971-05-14 | 1977-05-17 | Glaxo Laboratories Limited | 7β-[2-Etherified oximino-2-(thienyl-,furyl- or pyridylacetamido)]cephalosporins |
| GB1445979A (en) * | 1972-10-25 | 1976-08-11 | Glaxo Lab Ltd | Cephalosporin derivatives |
| GB1399086A (en) * | 1971-05-14 | 1975-06-25 | Glaxo Lab Ltd | Cephalosporin compounds |
-
1983
- 1983-04-12 US US06/484,129 patent/US4492693A/en not_active Expired - Lifetime
-
1984
- 1984-03-12 ZW ZW43/84A patent/ZW4384A1/xx unknown
- 1984-04-10 IL IL71497A patent/IL71497A0/xx unknown
- 1984-04-10 RO RO114217A patent/RO88220B/ro unknown
- 1984-04-11 FI FI841437A patent/FI841437A/fi not_active Application Discontinuation
- 1984-04-11 MA MA20314A patent/MA20093A1/fr unknown
- 1984-04-11 CA CA000451712A patent/CA1212938A/en not_active Expired
- 1984-04-11 OA OA58274A patent/OA07701A/xx unknown
- 1984-04-11 PT PT78403A patent/PT78403A/pt unknown
- 1984-04-11 GB GB08409381A patent/GB2137995A/en not_active Withdrawn
- 1984-04-11 DD DD84261874A patent/DD213927A5/de unknown
- 1984-04-11 EP EP84302456A patent/EP0122154A3/en not_active Ceased
- 1984-04-11 KR KR1019840001916A patent/KR840008654A/ko not_active Application Discontinuation
- 1984-04-11 JP JP59074847A patent/JPS59199692A/ja active Pending
- 1984-04-11 ES ES531531A patent/ES531531A0/es active Granted
- 1984-04-11 GR GR74378A patent/GR79908B/el unknown
- 1984-04-11 AU AU26736/84A patent/AU2673684A/en not_active Abandoned
- 1984-04-11 NO NO841441A patent/NO841441L/no unknown
- 1984-04-11 DK DK187384A patent/DK187384A/da not_active Application Discontinuation
- 1984-04-11 PL PL24717084A patent/PL247170A1/xx unknown
- 1984-04-11 ZA ZA842694A patent/ZA842694B/xx unknown
- 1984-04-11 GT GT198400056A patent/GT198400056A/es unknown
- 1984-04-12 CS CS842795A patent/CS243485B2/cs unknown
Also Published As
| Publication number | Publication date |
|---|---|
| AU2673684A (en) | 1984-10-18 |
| IL71497A0 (en) | 1984-07-31 |
| PL247170A1 (en) | 1985-08-13 |
| NO841441L (no) | 1984-10-15 |
| GR79908B (xx) | 1984-10-31 |
| GT198400056A (es) | 1985-10-03 |
| FI841437A0 (fi) | 1984-04-11 |
| ES8600308A1 (es) | 1985-10-01 |
| CS279584A2 (en) | 1985-08-15 |
| KR840008654A (ko) | 1984-12-17 |
| EP0122154A3 (en) | 1985-10-23 |
| PT78403A (en) | 1984-05-01 |
| DK187384A (da) | 1984-10-13 |
| DK187384D0 (da) | 1984-04-11 |
| JPS59199692A (ja) | 1984-11-12 |
| RO88220B (ro) | 1985-12-31 |
| ES531531A0 (es) | 1985-10-01 |
| MA20093A1 (fr) | 1984-12-31 |
| CS243485B2 (en) | 1986-06-12 |
| EP0122154A2 (en) | 1984-10-17 |
| GB2137995A (en) | 1984-10-17 |
| FI841437A (fi) | 1984-10-13 |
| OA07701A (fr) | 1985-08-30 |
| US4492693A (en) | 1985-01-08 |
| CA1212938A (en) | 1986-10-21 |
| ZA842694B (en) | 1985-11-27 |
| ZW4384A1 (en) | 1984-10-03 |
| RO88220A (ro) | 1985-12-30 |
| GB8409381D0 (en) | 1984-05-23 |
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