CZ239392A3 - 6-oxo-azepinindole compounds, processes and intermediates for their preparation and medicaments in which said compounds are comprised - Google Patents
6-oxo-azepinindole compounds, processes and intermediates for their preparation and medicaments in which said compounds are comprised Download PDFInfo
- Publication number
- CZ239392A3 CZ239392A3 CS922393A CS239392A CZ239392A3 CZ 239392 A3 CZ239392 A3 CZ 239392A3 CS 922393 A CS922393 A CS 922393A CS 239392 A CS239392 A CS 239392A CZ 239392 A3 CZ239392 A3 CZ 239392A3
- Authority
- CZ
- Czechia
- Prior art keywords
- formula
- compounds
- lower alkyl
- hydrogen
- group
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/06—Peri-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/14—Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/06—Antimigraine agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Engineering & Computer Science (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pain & Pain Management (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Nutrition Science (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Plural Heterocyclic Compounds (AREA)
- Indole Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE4125292A DE4125292A1 (de) | 1991-07-31 | 1991-07-31 | 6-oxo-azepinoindol-verbindungen sowie verfahren und zwischenprodukte zu ihrer herstellung und diese verbindungen enthaltende arzneimittel |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CZ239392A3 true CZ239392A3 (en) | 1993-04-14 |
Family
ID=6437366
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CS922393A CZ239392A3 (en) | 1991-07-31 | 1992-07-31 | 6-oxo-azepinindole compounds, processes and intermediates for their preparation and medicaments in which said compounds are comprised |
Country Status (21)
| Country | Link |
|---|---|
| US (1) | US5272143A (enExample) |
| EP (1) | EP0525584B1 (enExample) |
| JP (1) | JP3174158B2 (enExample) |
| KR (1) | KR930002353A (enExample) |
| CN (2) | CN1069733A (enExample) |
| AT (1) | ATE161012T1 (enExample) |
| AU (1) | AU649153B2 (enExample) |
| CA (1) | CA2075102A1 (enExample) |
| CZ (1) | CZ239392A3 (enExample) |
| DE (2) | DE4125292A1 (enExample) |
| ES (1) | ES2110454T3 (enExample) |
| FI (1) | FI923440A7 (enExample) |
| HU (2) | HU211105B (enExample) |
| IE (1) | IE922310A1 (enExample) |
| IL (1) | IL102503A (enExample) |
| MX (1) | MX9204457A (enExample) |
| NO (1) | NO300375B1 (enExample) |
| NZ (1) | NZ243715A (enExample) |
| RU (1) | RU2078765C1 (enExample) |
| TW (1) | TW207541B (enExample) |
| ZA (1) | ZA925093B (enExample) |
Families Citing this family (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5414130A (en) * | 1993-12-23 | 1995-05-09 | The Dow Chemical Company | Process for the preparation of diaminoresorcinol |
| PL210415B1 (pl) | 1999-01-11 | 2012-01-31 | Agouron Pharma | Pochodne indolu, środek farmaceutyczny i zastosowanie pochodnych indolu |
| ECSP003637A (es) | 1999-08-31 | 2002-03-25 | Agouron Pharma | Inhibidores triciclicos de poli (adp-ribosa) polimerasas |
| BRPI0515567A (pt) * | 2004-09-22 | 2008-07-29 | Pfizer | combinações terapêuticas compreendendo inibidor de poli (adp-ribose) polimerase |
| PT1794163E (pt) * | 2004-09-22 | 2010-03-01 | Pfizer | Método para a preparação de inibidores de poli(adpribose)- polimerases |
| AU2009260469B2 (en) | 2008-05-29 | 2014-02-13 | Albany Molecular Research, Inc. | 5-HT3 receptor modulators, methods of making, and use thereof |
| DK3150610T3 (da) * | 2010-02-12 | 2019-11-04 | Pfizer | Salte og polymorfer af 8-fluor-2-{4-[(methylamino}methyl]phenyl}-1,3,4,5-tetrahydro-6h-azepino[5,4,3-cd]indol-6-on |
| US10513515B2 (en) | 2017-08-25 | 2019-12-24 | Biotheryx, Inc. | Ether compounds and uses thereof |
| US11236103B2 (en) | 2018-07-27 | 2022-02-01 | Biotheryx, Inc. | Bifunctional compounds |
| EP4143329A4 (en) | 2020-04-28 | 2024-10-16 | Anwita Biosciences, Inc. | Interleukin-2 polypeptides and fusion proteins thereof, and their pharmaceutical compositions and therapeutic applications |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4910193A (en) * | 1985-12-16 | 1990-03-20 | Sandoz Ltd. | Treatment of gastrointestinal disorders |
-
1991
- 1991-07-31 DE DE4125292A patent/DE4125292A1/de not_active Withdrawn
-
1992
- 1992-07-08 ZA ZA925093A patent/ZA925093B/xx unknown
- 1992-07-15 IE IE231092A patent/IE922310A1/en not_active Application Discontinuation
- 1992-07-15 IL IL10250392A patent/IL102503A/en not_active IP Right Cessation
- 1992-07-21 DE DE59209055T patent/DE59209055D1/de not_active Expired - Fee Related
- 1992-07-21 ES ES92112431T patent/ES2110454T3/es not_active Expired - Lifetime
- 1992-07-21 EP EP92112431A patent/EP0525584B1/de not_active Expired - Lifetime
- 1992-07-21 AT AT92112431T patent/ATE161012T1/de not_active IP Right Cessation
- 1992-07-24 HU HU9202430A patent/HU211105B/hu not_active IP Right Cessation
- 1992-07-24 NZ NZ243715A patent/NZ243715A/en unknown
- 1992-07-30 MX MX9204457A patent/MX9204457A/es not_active IP Right Cessation
- 1992-07-30 CN CN92108977A patent/CN1069733A/zh active Pending
- 1992-07-30 KR KR1019920013719A patent/KR930002353A/ko not_active Withdrawn
- 1992-07-30 RU SU925052604A patent/RU2078765C1/ru active
- 1992-07-30 NO NO923004A patent/NO300375B1/no unknown
- 1992-07-30 JP JP20377092A patent/JP3174158B2/ja not_active Expired - Fee Related
- 1992-07-30 FI FI923440A patent/FI923440A7/fi not_active Application Discontinuation
- 1992-07-30 AU AU20677/92A patent/AU649153B2/en not_active Ceased
- 1992-07-31 CZ CS922393A patent/CZ239392A3/cs unknown
- 1992-07-31 CA CA002075102A patent/CA2075102A1/en not_active Abandoned
- 1992-07-31 US US07/922,527 patent/US5272143A/en not_active Expired - Lifetime
- 1992-09-10 TW TW081107187A patent/TW207541B/zh active
-
1994
- 1994-09-30 HU HU94P/P00032P patent/HU210217A9/hu unknown
-
1996
- 1996-01-19 CN CN96100699A patent/CN1141773A/zh active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| NO923004L (no) | 1993-02-01 |
| DE4125292A1 (de) | 1993-02-04 |
| JP3174158B2 (ja) | 2001-06-11 |
| EP0525584A1 (de) | 1993-02-03 |
| AU649153B2 (en) | 1994-05-12 |
| CA2075102A1 (en) | 1993-02-01 |
| KR930002353A (ko) | 1993-02-23 |
| CN1141773A (zh) | 1997-02-05 |
| ATE161012T1 (de) | 1997-12-15 |
| EP0525584B1 (de) | 1997-12-10 |
| NZ243715A (en) | 1995-03-28 |
| IL102503A0 (en) | 1993-01-14 |
| MX9204457A (es) | 1993-05-01 |
| HUT65453A (en) | 1994-06-28 |
| RU2078765C1 (ru) | 1997-05-10 |
| US5272143A (en) | 1993-12-21 |
| FI923440A7 (fi) | 1993-02-01 |
| JPH05202052A (ja) | 1993-08-10 |
| HU211105B (en) | 1995-10-30 |
| IL102503A (en) | 1995-12-31 |
| FI923440A0 (fi) | 1992-07-30 |
| NO300375B1 (no) | 1997-05-20 |
| IE922310A1 (en) | 1993-02-10 |
| CN1069733A (zh) | 1993-03-10 |
| NO923004D0 (no) | 1992-07-30 |
| ES2110454T3 (es) | 1998-02-16 |
| DE59209055D1 (de) | 1998-01-22 |
| TW207541B (enExample) | 1993-06-11 |
| ZA925093B (en) | 1993-04-28 |
| HU9202430D0 (en) | 1992-10-28 |
| AU2067792A (en) | 1993-02-04 |
| HU210217A9 (en) | 1995-02-28 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| PD00 | Pending as of 2000-06-30 in czech republic |