CY1119402T1 - Παραγωγα κινολινης ως αντιβακτηριακοι παραγοντες - Google Patents

Παραγωγα κινολινης ως αντιβακτηριακοι παραγοντες

Info

Publication number
CY1119402T1
CY1119402T1 CY20171100071T CY171100071T CY1119402T1 CY 1119402 T1 CY1119402 T1 CY 1119402T1 CY 20171100071 T CY20171100071 T CY 20171100071T CY 171100071 T CY171100071 T CY 171100071T CY 1119402 T1 CY1119402 T1 CY 1119402T1
Authority
CY
Cyprus
Prior art keywords
antibacterial agents
kinolin
products
compound
bacterial infection
Prior art date
Application number
CY20171100071T
Other languages
Greek (el)
English (en)
Inventor
Anil Koul
Koenraad Jozef Lodewijk Andries
Jérome Emile Georges Guillemont
Magali Madeleine Simone Motte
David Francis Alain LANÇOIS
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=35447198&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CY1119402(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Publication of CY1119402T1 publication Critical patent/CY1119402T1/el

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D215/00Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/20Oxygen atoms
    • C07D215/22Oxygen atoms attached in position 2 or 4
    • C07D215/227Oxygen atoms attached in position 2 or 4 only one oxygen atom which is attached in position 2
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D215/00Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/36Sulfur atoms
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02ATECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Quinoline Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
CY20171100071T 2005-06-28 2017-01-18 Παραγωγα κινολινης ως αντιβακτηριακοι παραγοντες CY1119402T1 (el)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP05105755 2005-06-28

Publications (1)

Publication Number Publication Date
CY1119402T1 true CY1119402T1 (el) 2018-03-07

Family

ID=35447198

Family Applications (1)

Application Number Title Priority Date Filing Date
CY20171100071T CY1119402T1 (el) 2005-06-28 2017-01-18 Παραγωγα κινολινης ως αντιβακτηριακοι παραγοντες

Country Status (31)

Country Link
US (1) US20130030016A1 (https=)
EP (1) EP1898909B1 (https=)
JP (1) JP5193857B2 (https=)
KR (1) KR101329587B1 (https=)
CN (1) CN101252927B (https=)
AP (1) AP2547A (https=)
AR (1) AR054804A1 (https=)
AU (1) AU2006263882B2 (https=)
BR (1) BRPI0613999B8 (https=)
CA (1) CA2612614C (https=)
CY (1) CY1119402T1 (https=)
DK (1) DK1898909T3 (https=)
EA (1) EA014431B1 (https=)
ES (1) ES2610472T3 (https=)
HR (1) HRP20170044T1 (https=)
HU (1) HUE030264T2 (https=)
IL (1) IL188395A (https=)
JO (1) JO3322B1 (https=)
LT (1) LT1898909T (https=)
MX (1) MX2008000079A (https=)
MY (1) MY173664A (https=)
NO (1) NO341285B1 (https=)
NZ (1) NZ564340A (https=)
PL (1) PL1898909T3 (https=)
PT (1) PT1898909T (https=)
RS (1) RS55601B1 (https=)
SG (1) SG166798A1 (https=)
TW (1) TWI413520B (https=)
UA (1) UA88701C2 (https=)
WO (1) WO2007000434A1 (https=)
ZA (1) ZA200711148B (https=)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JO2752B1 (en) 2005-06-28 2014-03-15 شركة جانسين فارماسوتيكا ان. في Quinoline derivatives acting as antibacterial agents
JO2683B1 (en) * 2006-12-06 2013-03-03 جانسين فارماسوتيكا ان. في Quinoline antibacterial derivatives
JO2970B1 (en) 2006-12-06 2016-03-15 جانسين فارماسوتيكا ان. في Quinoline antibacterial derivatives
JP5397881B2 (ja) * 2008-09-04 2014-01-22 昇一 城武 グラム陽性細菌用抗菌剤及び抗菌活性増強剤
CN104254527B (zh) 2012-04-27 2017-05-31 詹森药业有限公司 抗菌的喹啉衍生物
ES2607879T3 (es) 2012-04-27 2017-04-04 Janssen Pharmaceutica N.V. Derivados de quinolina antibacterianos
JP7514763B2 (ja) * 2017-10-13 2024-07-11 ザ ユニバーシティー オブ クイーンズランド 亜鉛イオノフォアおよびその使用
CN110606825A (zh) * 2019-10-30 2019-12-24 成都海杰亚医药科技有限公司 一种制备吡啶-2-硫醇的方法

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6103905A (en) * 1997-06-19 2000-08-15 Sepracor, Inc. Quinoline-indole antimicrobial agents, uses and compositions related thereto
ATE463482T1 (de) * 2002-07-25 2010-04-15 Janssen Pharmaceutica Nv Chinolinderivate und deren verwendung als mycobakterielle inhibitoren
PL1753427T3 (pl) * 2004-05-28 2008-09-30 Janssen Pharmaceutica Nv Zastosowanie podstawionych pochodnych chinoliny do leczenia chorób wywoływanych przez prątki lekooporne
EE05394B1 (et) * 2004-12-24 2011-04-15 Janssen Pharmaceutica N.V. Kinoliinihendid kasutamiseks latentse tuberkuloosi ravis
CA2528849C (en) * 2005-06-08 2014-01-14 Janssen Pharmaceutica N.V. Quinoline derivatives as antibacterial agents

Also Published As

Publication number Publication date
CA2612614C (en) 2017-07-25
BRPI0613999B1 (pt) 2020-04-22
CN101252927B (zh) 2014-01-01
EP1898909B1 (en) 2016-10-19
RS55601B1 (sr) 2017-06-30
EA014431B1 (ru) 2010-12-30
TWI413520B (zh) 2013-11-01
PT1898909T (pt) 2016-12-07
EA200800151A1 (ru) 2008-06-30
BRPI0613999A2 (pt) 2011-03-01
KR101329587B1 (ko) 2013-11-15
JP5193857B2 (ja) 2013-05-08
AU2006263882B2 (en) 2012-12-13
CN101252927A (zh) 2008-08-27
BRPI0613999B8 (pt) 2021-05-25
LT1898909T (lt) 2017-02-10
KR20080028459A (ko) 2008-03-31
MX2008000079A (es) 2008-03-19
DK1898909T3 (en) 2017-02-06
NO20080499L (no) 2008-02-29
TW200800183A (en) 2008-01-01
AP2547A (en) 2012-12-26
UA88701C2 (ru) 2009-11-10
US20130030016A1 (en) 2013-01-31
IL188395A (en) 2012-05-31
HK1120732A1 (en) 2009-04-09
ES2610472T3 (es) 2017-04-27
EP1898909A1 (en) 2008-03-19
AR054804A1 (es) 2007-07-18
IL188395A0 (en) 2008-08-07
JO3322B1 (ar) 2019-03-13
NO341285B1 (no) 2017-10-02
PL1898909T3 (pl) 2017-03-31
SG166798A1 (en) 2010-12-29
MY173664A (en) 2020-02-14
HRP20170044T1 (hr) 2017-03-10
HUE030264T2 (en) 2017-04-28
JP2008546824A (ja) 2008-12-25
WO2007000434A1 (en) 2007-01-04
ZA200711148B (en) 2013-03-27
CA2612614A1 (en) 2007-01-04
AU2006263882A1 (en) 2007-01-04
NZ564340A (en) 2011-02-25

Similar Documents

Publication Publication Date Title
CY1119402T1 (el) Παραγωγα κινολινης ως αντιβακτηριακοι παραγοντες
CY1121885T1 (el) Αντι-ογκικες ενωσεις
CY1121433T1 (el) Παραγωγα δικυκλικων ετεροκυκλυλιων ως αναστολεις irak4
CY1123705T1 (el) Αλατα και πολυμορφα μιας ενωσης τετρακυκλινης
GEAP202215535A (en) Compounds
CR20220251A (es) Nuevos derivados de metilquinazolinona
CY1124086T1 (el) Παραγωγα 3-τετραζολυλ-βενζεν-1,2-δισουλφοναμιδιου ως αναστολεις μεταλλο-βητα-λακταμασης
CY1125047T1 (el) Διεργασιες για την παρασκευη ενωσεων τυπου οξαθειαζινης
CY1106801T1 (el) Νεες ετεροκυκλικες ενωσεις, η παρασκευη τους και η χρηση τους ως φαρμακα, ιδιαιτερα ως αντιβακτηριακα
CY1109644T1 (el) 2,4-διαμινο-πυριμιδινες ως αναστολεις audora
CY1113924T1 (el) Ενωσεις καρβαζολης και θεραπευτικες χρησεις των ενωσεων
CY1110127T1 (el) Υποκατεστημενες 1-προπιολυλο-πιπεραζινες με χημικη συγγενεια για τον υποδοχεα mglur5 για τη θεραπεια καταστασεων πονου
CY1114318T1 (el) Παραγωγα κινολινης ως αντιβακτηριακοι παραγοντες
CR9113A (es) Compuestos acetamida como fungicidas
CY1115227T1 (el) Νεοι καταστολεις φωσφοδιεστερασης (phosphodiesterase)
CY1118515T1 (el) Παραγωγα κινολινης ως αντιβακτηριακοι παραγοντες
CY1111830T1 (el) Παραγωγα πυριδινης ως ρυθμιστες υποδοχεων s1p1/edg1
CY1111188T1 (el) Αντιβακτηριακα παραγωγα κινολινης
CY1117461T1 (el) Παραγωγα κιναζολινοδιονης, παρασκευη αυτων και οι θεραπευτικες εφαρμογες τους
CY1112614T1 (el) Αγωγη με κλαδριβινη για τη θεραπεια πολλαπλης σκληρυνσης
CY1124577T1 (el) Καινοτομες ενωσεις τετραζολιου και η χρηση τους στη θεραπεια της φυματιωσης
MX2019009354A (es) Piridinas sustituidas con heterociclilsulfonilo y su uso en el tratamiento del cancer.
CY1115729T1 (el) Τρικυκλικη ενωση και φαρμακευτικη χρηση αυτης
CY1113733T1 (el) Παραγωγα κινολινονης και οι φαρμακευτικες συνθεσεις αυτων
MX2019009351A (es) Piridinas sustituidas con heteroarilsulfonilo y su uso en el tratamiento del cancer.