CS251790B2 - Method of pyrrole's new condensed derivatives production - Google Patents

Method of pyrrole's new condensed derivatives production Download PDF

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Publication number
CS251790B2
CS251790B2 CS855248A CS524885A CS251790B2 CS 251790 B2 CS251790 B2 CS 251790B2 CS 855248 A CS855248 A CS 855248A CS 524885 A CS524885 A CS 524885A CS 251790 B2 CS251790 B2 CS 251790B2
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CS
Czechoslovakia
Prior art keywords
het
pyrrolo
integer
dihydro
pyrrole
Prior art date
Application number
CS855248A
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Czech (cs)
English (en)
Other versions
CS524885A2 (en
Inventor
Jaen-Louis Fabre
Daniel Farge
Claude James
Daniel Lave
Original Assignee
Rhone Poulenc Sante
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Rhone Poulenc Sante filed Critical Rhone Poulenc Sante
Publication of CS524885A2 publication Critical patent/CS524885A2/cs
Publication of CS251790B2 publication Critical patent/CS251790B2/cs

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/06Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D513/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04Ortho-condensed systems

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Hematology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
CS855248A 1983-12-21 1984-12-21 Method of pyrrole's new condensed derivatives production CS251790B2 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR8320474A FR2557111B1 (fr) 1983-12-21 1983-12-21 Nouveaux derives ortho-condenses du pyrrole, leur preparation et les medicaments qui les contiennent

Publications (2)

Publication Number Publication Date
CS524885A2 CS524885A2 (en) 1986-12-18
CS251790B2 true CS251790B2 (en) 1987-08-13

Family

ID=9295399

Family Applications (3)

Application Number Title Priority Date Filing Date
CS855248A CS251790B2 (en) 1983-12-21 1984-12-21 Method of pyrrole's new condensed derivatives production
CS8410201A CS251782B2 (en) 1983-12-21 1984-12-21 Method of pyrrole's new condensed derivatives productio(
CS855249A CS251791B2 (en) 1983-12-21 1984-12-21 Method of pyrrole's new condensed derivatives production

Family Applications After (2)

Application Number Title Priority Date Filing Date
CS8410201A CS251782B2 (en) 1983-12-21 1984-12-21 Method of pyrrole's new condensed derivatives productio(
CS855249A CS251791B2 (en) 1983-12-21 1984-12-21 Method of pyrrole's new condensed derivatives production

Country Status (15)

Country Link
US (1) US4684658A (fi)
EP (1) EP0147317A3 (fi)
JP (1) JPS60172977A (fi)
KR (1) KR850004768A (fi)
AU (1) AU573666B2 (fi)
CA (1) CA1250286A (fi)
CS (3) CS251790B2 (fi)
DK (1) DK616584A (fi)
FI (1) FI76809C (fi)
FR (1) FR2557111B1 (fi)
HU (2) HU194238B (fi)
IL (1) IL73888A (fi)
NZ (1) NZ210671A (fi)
SU (2) SU1436883A3 (fi)
ZA (1) ZA849958B (fi)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5260451A (en) * 1989-05-11 1993-11-09 Merckle Gmbh Substituted pyrrole compounds and use thereof in pharmaceutical compositions
DE3915450A1 (de) * 1989-05-11 1990-11-15 Gerd Prof Dr Dannhardt Substituierte pyrrolverbindungen und deren anwendung in der pharmazie
AU5938390A (en) * 1989-06-26 1991-01-17 Research Foundation Of The State University Of New York, The Bis-acyloxymethyl derivatives
US5395846A (en) * 1993-06-25 1995-03-07 Rhone-Poulenc Rorer Pharmaceuticals Inc. Amino Bi- and tri-carbocyclic aklane bis-aryl squalene synthase inhibitors
DE4419246A1 (de) * 1994-06-01 1995-12-07 Merckle Gmbh Heteroarylsubstituierte Pyrrolizinverbindungen und deren Anwendung in der Pharmazie
DE4419315A1 (de) * 1994-06-01 1995-12-07 Merckle Gmbh Heteropyrrolizinverbindungen und deren Anwendung in der Pharmazie
DE4419247A1 (de) * 1994-06-01 1995-12-07 Merckle Gmbh Sulfonylierte Pyrrolizincarbonsäureamide und deren Anwendung in der Pharmazie
FR2735476B1 (fr) * 1995-06-14 1997-07-18 Rhone Poulenc Rorer Sa Nouvelle application de derives du pyrrole
FR2757059B1 (fr) * 1996-12-12 1999-01-29 Rhone Poulenc Rorer Sa Nouvelle application therapeutique des derives du pyrrole
FR2757166B1 (fr) * 1996-12-12 1999-01-29 Rhone Poulenc Rorer Sa Derives du pyrrole, leur preparation et les compositions pharmaceutiques qui les contiennent
US6191925B1 (en) 1999-06-18 2001-02-20 Storage Technology Corporation Dual element read with shaped elements
CA2391871C (en) 1999-11-23 2009-01-27 Merckle Gmbh Anti-inflammatory oxo derivatives and hydroxy derivatives of pyrrolizines, and their pharmaceutical use
DE10004157A1 (de) 2000-02-01 2001-08-02 Merckle Gmbh Chem Pharm Fabrik 4-Pyridyl-und 2,4-Pyrimidinyl-substituierte Pyrrolderivate und ihre Anwendung in der Pharmazie
KR20060128045A (ko) * 2004-03-08 2006-12-13 베링거 인겔하임 파마슈티칼즈, 인코포레이티드 교차 커플링 인돌의 제조방법

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3429885A (en) * 1965-10-22 1969-02-25 American Home Prod Pyridylethyl and piperidylethyl pyrroles
GB1174124A (en) * 1967-06-30 1969-12-10 Beecham Group Ltd Pharmacologically Active Indolizine Compounds
FR2541280B1 (fr) * 1983-01-13 1985-06-21 Rhone Poulenc Sante Nouveaux derives du 1h, 3h-pyrrolo (1,2c) thiazolecarboxamide-7, leur preparation et les medicaments qui les contiennent
AU562833B2 (en) * 1983-01-13 1987-06-18 Rhone-Poulenc Sante Ortho-fused pyrrole derivatives
FR2539417A1 (fr) * 1983-01-13 1984-07-20 Rhone Poulenc Sante Nouveaux pyrrolo-1, 2 heterocycles, leur preparation et les medicaments qui les contiennent

Also Published As

Publication number Publication date
FR2557111B1 (fr) 1986-04-11
DK616584A (da) 1985-06-22
IL73888A0 (en) 1985-03-31
ZA849958B (en) 1985-08-28
CS524885A2 (en) 1986-12-18
SU1440349A3 (ru) 1988-11-23
CS251791B2 (en) 1987-08-13
HUT40435A (en) 1986-12-28
FI845064A0 (fi) 1984-12-20
FI76809C (fi) 1988-12-12
CS251782B2 (en) 1987-08-13
DK616584D0 (da) 1984-12-20
HU196801B (en) 1989-01-30
CA1250286A (fr) 1989-02-21
FR2557111A1 (fr) 1985-06-28
CS524985A2 (en) 1986-12-18
NZ210671A (en) 1989-08-29
FI76809B (fi) 1988-08-31
FI845064L (fi) 1985-06-22
IL73888A (en) 1987-11-30
AU573666B2 (en) 1988-06-16
EP0147317A3 (fr) 1986-06-25
EP0147317A2 (fr) 1985-07-03
US4684658A (en) 1987-08-04
KR850004768A (ko) 1985-07-27
AU3696084A (en) 1985-07-04
JPS60172977A (ja) 1985-09-06
HU194238B (en) 1988-01-28
SU1436883A3 (ru) 1988-11-07

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