CS251790B2 - Method of pyrrole's new condensed derivatives production - Google Patents
Method of pyrrole's new condensed derivatives production Download PDFInfo
- Publication number
- CS251790B2 CS251790B2 CS855248A CS524885A CS251790B2 CS 251790 B2 CS251790 B2 CS 251790B2 CS 855248 A CS855248 A CS 855248A CS 524885 A CS524885 A CS 524885A CS 251790 B2 CS251790 B2 CS 251790B2
- Authority
- CS
- Czechoslovakia
- Prior art keywords
- het
- pyrrolo
- integer
- dihydro
- pyrrole
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Life Sciences & Earth Sciences (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Pharmacology & Pharmacy (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR8320474A FR2557111B1 (fr) | 1983-12-21 | 1983-12-21 | Nouveaux derives ortho-condenses du pyrrole, leur preparation et les medicaments qui les contiennent |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| CS524885A2 CS524885A2 (en) | 1986-12-18 |
| CS251790B2 true CS251790B2 (en) | 1987-08-13 |
Family
ID=9295399
Family Applications (3)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CS855248A CS251790B2 (en) | 1983-12-21 | 1984-12-21 | Method of pyrrole's new condensed derivatives production |
| CS855249A CS251791B2 (en) | 1983-12-21 | 1984-12-21 | Method of pyrrole's new condensed derivatives production |
| CS8410201A CS251782B2 (en) | 1983-12-21 | 1984-12-21 | Method of pyrrole's new condensed derivatives productio( |
Family Applications After (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CS855249A CS251791B2 (en) | 1983-12-21 | 1984-12-21 | Method of pyrrole's new condensed derivatives production |
| CS8410201A CS251782B2 (en) | 1983-12-21 | 1984-12-21 | Method of pyrrole's new condensed derivatives productio( |
Country Status (15)
| Country | Link |
|---|---|
| US (1) | US4684658A (fi) |
| EP (1) | EP0147317A3 (fi) |
| JP (1) | JPS60172977A (fi) |
| KR (1) | KR850004768A (fi) |
| AU (1) | AU573666B2 (fi) |
| CA (1) | CA1250286A (fi) |
| CS (3) | CS251790B2 (fi) |
| DK (1) | DK616584A (fi) |
| FI (1) | FI76809C (fi) |
| FR (1) | FR2557111B1 (fi) |
| HU (2) | HU194238B (fi) |
| IL (1) | IL73888A (fi) |
| NZ (1) | NZ210671A (fi) |
| SU (2) | SU1436883A3 (fi) |
| ZA (1) | ZA849958B (fi) |
Families Citing this family (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5260451A (en) * | 1989-05-11 | 1993-11-09 | Merckle Gmbh | Substituted pyrrole compounds and use thereof in pharmaceutical compositions |
| DE3915450A1 (de) * | 1989-05-11 | 1990-11-15 | Gerd Prof Dr Dannhardt | Substituierte pyrrolverbindungen und deren anwendung in der pharmazie |
| AU5938390A (en) * | 1989-06-26 | 1991-01-17 | Research Foundation Of The State University Of New York, The | Bis-acyloxymethyl derivatives |
| US5395846A (en) * | 1993-06-25 | 1995-03-07 | Rhone-Poulenc Rorer Pharmaceuticals Inc. | Amino Bi- and tri-carbocyclic aklane bis-aryl squalene synthase inhibitors |
| DE4419246A1 (de) * | 1994-06-01 | 1995-12-07 | Merckle Gmbh | Heteroarylsubstituierte Pyrrolizinverbindungen und deren Anwendung in der Pharmazie |
| DE4419247A1 (de) * | 1994-06-01 | 1995-12-07 | Merckle Gmbh | Sulfonylierte Pyrrolizincarbonsäureamide und deren Anwendung in der Pharmazie |
| DE4419315A1 (de) * | 1994-06-01 | 1995-12-07 | Merckle Gmbh | Heteropyrrolizinverbindungen und deren Anwendung in der Pharmazie |
| FR2735476B1 (fr) * | 1995-06-14 | 1997-07-18 | Rhone Poulenc Rorer Sa | Nouvelle application de derives du pyrrole |
| FR2757166B1 (fr) * | 1996-12-12 | 1999-01-29 | Rhone Poulenc Rorer Sa | Derives du pyrrole, leur preparation et les compositions pharmaceutiques qui les contiennent |
| FR2757059B1 (fr) * | 1996-12-12 | 1999-01-29 | Rhone Poulenc Rorer Sa | Nouvelle application therapeutique des derives du pyrrole |
| US6191925B1 (en) | 1999-06-18 | 2001-02-20 | Storage Technology Corporation | Dual element read with shaped elements |
| HK1047095B (zh) | 1999-11-23 | 2004-10-15 | Merckle Gmbh | 抗發炎的吡咯裏嗪氧化衍生物和氫氧衍生物安定它們的藥物作用 |
| DE10004157A1 (de) | 2000-02-01 | 2001-08-02 | Merckle Gmbh Chem Pharm Fabrik | 4-Pyridyl-und 2,4-Pyrimidinyl-substituierte Pyrrolderivate und ihre Anwendung in der Pharmazie |
| JP5442949B2 (ja) * | 2004-03-08 | 2014-03-19 | ベーリンガー インゲルハイム ファーマシューティカルズ インコーポレイテッド | インドールのクロスカップリング方法 |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3429885A (en) * | 1965-10-22 | 1969-02-25 | American Home Prod | Pyridylethyl and piperidylethyl pyrroles |
| GB1174124A (en) * | 1967-06-30 | 1969-12-10 | Beecham Group Ltd | Pharmacologically Active Indolizine Compounds |
| FR2539417A1 (fr) * | 1983-01-13 | 1984-07-20 | Rhone Poulenc Sante | Nouveaux pyrrolo-1, 2 heterocycles, leur preparation et les medicaments qui les contiennent |
| DD216021A5 (de) * | 1983-01-13 | 1984-11-28 | Rhone Poulenc Sante | Verfahren zur herstellung eines neuen pyrrolderivates |
| FR2541280B1 (fr) * | 1983-01-13 | 1985-06-21 | Rhone Poulenc Sante | Nouveaux derives du 1h, 3h-pyrrolo (1,2c) thiazolecarboxamide-7, leur preparation et les medicaments qui les contiennent |
-
1983
- 1983-12-21 FR FR8320474A patent/FR2557111B1/fr not_active Expired
-
1984
- 1984-12-20 US US06/684,061 patent/US4684658A/en not_active Expired - Fee Related
- 1984-12-20 AU AU36960/84A patent/AU573666B2/en not_active Ceased
- 1984-12-20 HU HU844758A patent/HU194238B/hu not_active IP Right Cessation
- 1984-12-20 SU SU843826152A patent/SU1436883A3/ru active
- 1984-12-20 KR KR1019840008153A patent/KR850004768A/ko not_active Withdrawn
- 1984-12-20 NZ NZ210671A patent/NZ210671A/xx unknown
- 1984-12-20 EP EP84402675A patent/EP0147317A3/fr not_active Withdrawn
- 1984-12-20 CA CA000470656A patent/CA1250286A/fr not_active Expired
- 1984-12-20 DK DK616584A patent/DK616584A/da not_active Application Discontinuation
- 1984-12-20 FI FI845064A patent/FI76809C/fi not_active IP Right Cessation
- 1984-12-20 JP JP59267581A patent/JPS60172977A/ja active Pending
- 1984-12-20 IL IL73888A patent/IL73888A/xx unknown
- 1984-12-20 HU HU844960A patent/HU196801B/hu not_active IP Right Cessation
- 1984-12-20 ZA ZA849958A patent/ZA849958B/xx unknown
- 1984-12-21 CS CS855248A patent/CS251790B2/cs unknown
- 1984-12-21 CS CS855249A patent/CS251791B2/cs unknown
- 1984-12-21 CS CS8410201A patent/CS251782B2/cs unknown
-
1985
- 1985-09-23 SU SU853954499A patent/SU1440349A3/ru active
Also Published As
| Publication number | Publication date |
|---|---|
| US4684658A (en) | 1987-08-04 |
| SU1436883A3 (ru) | 1988-11-07 |
| FI845064L (fi) | 1985-06-22 |
| HU194238B (en) | 1988-01-28 |
| NZ210671A (en) | 1989-08-29 |
| EP0147317A3 (fr) | 1986-06-25 |
| SU1440349A3 (ru) | 1988-11-23 |
| FR2557111A1 (fr) | 1985-06-28 |
| FI76809B (fi) | 1988-08-31 |
| FI76809C (fi) | 1988-12-12 |
| AU3696084A (en) | 1985-07-04 |
| HUT40435A (en) | 1986-12-28 |
| CS524885A2 (en) | 1986-12-18 |
| KR850004768A (ko) | 1985-07-27 |
| FI845064A0 (fi) | 1984-12-20 |
| CS524985A2 (en) | 1986-12-18 |
| IL73888A0 (en) | 1985-03-31 |
| JPS60172977A (ja) | 1985-09-06 |
| CS251791B2 (en) | 1987-08-13 |
| EP0147317A2 (fr) | 1985-07-03 |
| DK616584D0 (da) | 1984-12-20 |
| CA1250286A (fr) | 1989-02-21 |
| HU196801B (en) | 1989-01-30 |
| ZA849958B (en) | 1985-08-28 |
| DK616584A (da) | 1985-06-22 |
| AU573666B2 (en) | 1988-06-16 |
| IL73888A (en) | 1987-11-30 |
| FR2557111B1 (fr) | 1986-04-11 |
| CS251782B2 (en) | 1987-08-13 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| CS231957B2 (en) | Manufacturing process of heterocyclic compounds | |
| Julino et al. | Antitumour polycyclic acridines. Part 5. 1 Synthesis of 7 H-pyrido [4, 3, 2-kl] acridines with exploitable functionality in the pyridine ring | |
| SU1630612A3 (ru) | Способ получени производных пиррола | |
| EP0095289B1 (en) | Imidazo(1,2-c)pyrazolo(3,4-e)pyrimidines and their production | |
| Wamhoff et al. | On the synthesis of zwitterionic heteropolycyclic pyrazoles by a three-component reaction. Some mechanistic considerations | |
| FI76809B (fi) | Foerfarande foer framstaellning av terapeutiskt anvaendbara nya 5-(3-pyridyl)pyrrolo/1,2-c/tiazol-7- karboxamid-derivat. | |
| Avan et al. | Synthesis and antimicrobial investigation of some 5H-pyridazino [4, 5-b] indoles | |
| SE410857B (sv) | Forfarande for framstellning av nya derivat av naftyridin | |
| US4705793A (en) | Pyrazolo[3,4-b]pyrrolo[3,4-e]pyridine-5(1H)-one and 1-H-pyrazolo[3,4-b][1,6]naphthyridine-5(6H)-one derivations, useful as anti-anxiety agents | |
| Kharaneko | New approach to the synthesis of pyrrolo [3, 4-c] pyridines | |
| Hajinasiri | Acetylenic esters in organic synthesis | |
| Niopas et al. | Reactions of 2H, 5H-imidazo [1, 5-b] isoquinoline-1, 3-diones with bromine | |
| Rakib et al. | Synthesis of new pyrazolo [3, 4-b] pyridin-3-ones and pyrazolo [1, 5-a] pyrimidin-2 (1H)-one and study of the pyrazolic nitrogen reactivity | |
| PT86154B (pt) | Processo para a preparacao de novos pirrolobenzimidazoles e de composicoes farmaceuticas que os contem | |
| US3553207A (en) | Phenylpyrazolodiazepinone compounds | |
| EP1572696B1 (en) | Process for the direct preparation of 5-alkoxy and 5-acyloxy analogues of campthothecins or mappicene ketones | |
| PL100184B1 (pl) | Sposob wytwarzania nowych pochodnych naftyrydynylo-piroliny | |
| Abass | Chemistry of substituted quinolinones. Part 8. Synthesis and cyclization reactions of ethyl 5-amino-1-(1-methyl-2-oxoquinolin-4-YL)-3-methylsulfanylpyrazole-4-carboxylate | |
| KINOSHITA et al. | Synthesis and Reactions of 2, 3-Dihydrothiazolo [3, 2-a] pyrimidine Derivatives | |
| US6872829B2 (en) | Process for the direct preparation of 5-alkoxy and 5-acyloxy analogues of camptothecins or mappicene ketones | |
| Merslavič et al. | 1, 3‐dipolar cycloaddition of diazomethane to azolopyridazines. The synthesis of 8‐methyl‐8H‐and 9‐methyl‐9H‐pyrazolo [3, 4‐d]‐s‐triazolo [4, 3‐b] pyridazine and 1‐methyl‐1H‐and 2‐methyl‐2H‐imidazo [1, 2‐b] pyrazolo [3, 4‐b] pyridazine derivatives | |
| Zubkov et al. | Short approach to pyrrolopyrazino-, pyrrolodiazepino-isoindoles and their benzo analogues via the IMDAF reaction | |
| Meng et al. | A general synthesis of furo [3, 2-c][1, 2, 4] triazolo [1, 5-a] azepine and furo [2, 3-f][1, 2, 4] triazolo [1, 5-a] azepine derivatives | |
| Krbavcic et al. | The synthesis of furo/2, 3-c/pyridazine, a novel heterocyclic system | |
| FI79324C (fi) | Foerfarande foer framstaellning av terapeutiskt anvaendbara pyrrolo/1,2-c/tiazol-7-karboxamid- eller -7-acetamidderivat. |