CS244405B2 - 3-aminovinyl cephalosporines' new derivatives production method - Google Patents
3-aminovinyl cephalosporines' new derivatives production method Download PDFInfo
- Publication number
- CS244405B2 CS244405B2 CS803543A CS354380A CS244405B2 CS 244405 B2 CS244405 B2 CS 244405B2 CS 803543 A CS803543 A CS 803543A CS 354380 A CS354380 A CS 354380A CS 244405 B2 CS244405 B2 CS 244405B2
- Authority
- CS
- Czechoslovakia
- Prior art keywords
- formula
- mixture
- radical
- group
- solution
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- C07D501/14—Compounds having a nitrogen atom directly attached in position 7
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/02—Nutrients, e.g. vitamins, minerals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Life Sciences & Earth Sciences (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Diabetes (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Obesity (AREA)
- Hematology (AREA)
- Nutrition Science (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Cephalosporin Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR7913096A FR2457296A1 (fr) | 1979-05-23 | 1979-05-23 | Nouveaux derives de vinyl-3 cephalosporines et leur preparation |
Publications (2)
Publication Number | Publication Date |
---|---|
CS354380A2 CS354380A2 (bg) | 1985-09-17 |
CS244405B2 true CS244405B2 (en) | 1986-07-17 |
Family
ID=9225762
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CS803543A CS244405B2 (en) | 1979-05-23 | 1980-05-21 | 3-aminovinyl cephalosporines' new derivatives production method |
Country Status (31)
Country | Link |
---|---|
US (1) | US4307233A (bg) |
JP (1) | JPS55154981A (bg) |
AT (1) | AT369375B (bg) |
AU (1) | AU534806B2 (bg) |
BE (1) | BE883416A (bg) |
CA (1) | CA1144919A (bg) |
CH (1) | CH645379A5 (bg) |
CS (1) | CS244405B2 (bg) |
DD (1) | DD150899A5 (bg) |
DE (1) | DE3019462A1 (bg) |
DK (1) | DK222080A (bg) |
ES (1) | ES8102136A1 (bg) |
FI (1) | FI801641A (bg) |
FR (1) | FR2457296A1 (bg) |
GB (1) | GB2051062B (bg) |
GR (1) | GR68426B (bg) |
HU (1) | HU185890B (bg) |
IE (1) | IE49814B1 (bg) |
IL (1) | IL60139A (bg) |
IT (1) | IT1140974B (bg) |
LU (1) | LU82477A1 (bg) |
NL (1) | NL8003023A (bg) |
NO (1) | NO801502L (bg) |
NZ (1) | NZ193799A (bg) |
PH (1) | PH15946A (bg) |
PL (1) | PL126481B1 (bg) |
PT (1) | PT71276A (bg) |
SE (1) | SE451072B (bg) |
SU (1) | SU1031409A3 (bg) |
YU (1) | YU136880A (bg) |
ZA (1) | ZA803038B (bg) |
Families Citing this family (14)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DK480679A (da) * | 1978-11-15 | 1980-05-16 | Glaxo Group Ltd | Fremgangsmaade til fremstilling af cephalosporinforbindelser |
FR2494275A2 (fr) * | 1980-11-20 | 1982-05-21 | Rhone Poulenc Ind | Nouveaux derives de vinyl-3 cephalosporines et leur preparation |
FR2494280A1 (fr) * | 1980-11-20 | 1982-05-21 | Rhone Poulenc Ind | Nouveaux derives de la cephalosporine et leur preparation |
FR2494279A1 (fr) * | 1980-11-20 | 1982-05-21 | Rhone Poulenc Ind | Nouvelles oxacephalosporines, leur preparation et les medicaments qui les contiennent |
FR2505334A1 (fr) * | 1981-05-11 | 1982-11-12 | Rhone Poulenc Sante | Nouvelles oxacephalosporines et leur preparation |
FR2511372A1 (fr) * | 1981-08-17 | 1983-02-18 | Rhone Poulenc Sante | Nouveaux derives de la cephalosporine et leur preparation |
US4486586A (en) * | 1983-02-10 | 1984-12-04 | Bristol-Myers Company | Cephalosporin derivatives |
US4560749A (en) * | 1983-11-18 | 1985-12-24 | Eli Lilly And Company | Cephem-3-imidates and 3-amidines |
US4874856A (en) * | 1985-06-24 | 1989-10-17 | Bristol-Myers Company | 3-(substituted)propenyl-7-(aminothiazolylacetamido) ceph-3-em-4-carboxylic acids and esters thereof |
US4708955A (en) * | 1985-06-24 | 1987-11-24 | Bristol-Myers Company | 3-(substituted)propenyl-7-aminothiazol-ylcephalosporanic acids and esters thereof |
EP0346465B1 (en) * | 1986-04-14 | 1993-08-11 | Banyu Pharmaceutical Co., Ltd. | 1-carboxy-1-vyniloxyiminoaminothiazole cephalosporing derivatives and process for their preparation |
EP0841339B1 (en) | 1996-11-06 | 2007-02-21 | Basilea Pharmaceutica AG | Vinylpyrrolidinon cephalosporin derivatives |
EP2209474A4 (en) | 2007-10-09 | 2013-07-24 | Sopharmia Inc | BROAD SPECTRUM BETA-LACTAMASE INHIBITORS |
EP3441071A1 (en) | 2013-03-12 | 2019-02-13 | Gladius Pharmaceuticals Corporation | Derivatized cephalosporins |
Family Cites Families (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4065620A (en) * | 1971-06-14 | 1977-12-27 | Eli Lilly And Company | 3-(Substituted) vinyl cephalosporins |
GB1463077A (en) * | 1973-04-19 | 1977-02-02 | Glaxo Lab Ltd | 7-substituted-ethyl-cephalosporin derivatives |
IL46302A (en) * | 1973-12-21 | 1978-09-29 | Glaxo Lab Ltd | 7 -( -(etherified oxyimino)-acylamido)cephalosporanic acid derivatives |
US4144393A (en) * | 1973-12-21 | 1979-03-13 | Glaxo Laboratories Limited | 3-Acetoxymethyl cephalosporins having at position-7 a carboxy substituted α-etherified hydroxyiminoarylacetamido group |
JPS5129492A (en) * | 1974-09-04 | 1976-03-12 | Sankyo Co | Sefuarosuhorinjudotai no seiho |
DK154939C (da) * | 1974-12-19 | 1989-06-12 | Takeda Chemical Industries Ltd | Analogifremgangsmaade til fremstilling af thiazolylacetamido-cephemforbindelser eller farmaceutisk acceptable salte eller estere deraf |
JPS5253890A (en) * | 1975-10-14 | 1977-04-30 | Syntex Inc | Production of cephalosporin type compound |
PT71654B (en) * | 1979-08-15 | 1982-01-22 | Merck & Co Inc | Process for preparing allylsulfoxide enzyme inhibitor |
-
1979
- 1979-05-23 FR FR7913096A patent/FR2457296A1/fr active Granted
-
1980
- 1980-05-21 SE SE8003821A patent/SE451072B/sv not_active IP Right Cessation
- 1980-05-21 FI FI801641A patent/FI801641A/fi not_active Application Discontinuation
- 1980-05-21 GR GR62015A patent/GR68426B/el unknown
- 1980-05-21 PT PT71276A patent/PT71276A/pt unknown
- 1980-05-21 SU SU802926697A patent/SU1031409A3/ru active
- 1980-05-21 BE BE0/200707A patent/BE883416A/fr not_active IP Right Cessation
- 1980-05-21 GB GB8016727A patent/GB2051062B/en not_active Expired
- 1980-05-21 DE DE19803019462 patent/DE3019462A1/de not_active Ceased
- 1980-05-21 HU HU801278A patent/HU185890B/hu unknown
- 1980-05-21 NZ NZ193799A patent/NZ193799A/xx unknown
- 1980-05-21 IT IT22243/80A patent/IT1140974B/it active
- 1980-05-21 AU AU58595/80A patent/AU534806B2/en not_active Ceased
- 1980-05-21 CA CA000352324A patent/CA1144919A/fr not_active Expired
- 1980-05-21 YU YU01368/80A patent/YU136880A/xx unknown
- 1980-05-21 IE IE1062/80A patent/IE49814B1/en unknown
- 1980-05-21 LU LU82477A patent/LU82477A1/fr unknown
- 1980-05-21 PL PL1980224391A patent/PL126481B1/pl unknown
- 1980-05-21 AT AT0270980A patent/AT369375B/de active
- 1980-05-21 ZA ZA00803038A patent/ZA803038B/xx unknown
- 1980-05-21 DD DD80221272A patent/DD150899A5/de unknown
- 1980-05-21 DK DK222080A patent/DK222080A/da not_active Application Discontinuation
- 1980-05-21 NO NO801502A patent/NO801502L/no unknown
- 1980-05-21 CH CH398980A patent/CH645379A5/fr not_active IP Right Cessation
- 1980-05-21 CS CS803543A patent/CS244405B2/cs unknown
- 1980-05-21 ES ES491687A patent/ES8102136A1/es not_active Expired
- 1980-05-21 US US06/152,085 patent/US4307233A/en not_active Expired - Lifetime
- 1980-05-22 IL IL60139A patent/IL60139A/xx unknown
- 1980-05-22 PH PH24056A patent/PH15946A/en unknown
- 1980-05-23 JP JP6800980A patent/JPS55154981A/ja active Granted
- 1980-05-23 NL NL8003023A patent/NL8003023A/nl not_active Application Discontinuation
Also Published As
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