CS207619B2 - Method of making the new derivatives of 5,11-dihydro-6h-pyrido 2,3-b 1,4 benzodiazepin-6-on - Google Patents

Method of making the new derivatives of 5,11-dihydro-6h-pyrido 2,3-b 1,4 benzodiazepin-6-on Download PDF

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Publication number
CS207619B2
CS207619B2 CS783473A CS347378A CS207619B2 CS 207619 B2 CS207619 B2 CS 207619B2 CS 783473 A CS783473 A CS 783473A CS 347378 A CS347378 A CS 347378A CS 207619 B2 CS207619 B2 CS 207619B2
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CS
Czechoslovakia
Prior art keywords
pyrido
benzodiazepin
formula
dihydro
group
Prior art date
Application number
CS783473A
Other languages
Czech (cs)
English (en)
Inventor
Guenther Schmidt
Matyas Leitold
Original Assignee
Thomae Gmbh Dr K
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Thomae Gmbh Dr K filed Critical Thomae Gmbh Dr K
Priority to CS798394A priority Critical patent/CS207620B2/cs
Publication of CS207619B2 publication Critical patent/CS207619B2/cs

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
CS783473A 1977-05-31 1978-05-29 Method of making the new derivatives of 5,11-dihydro-6h-pyrido 2,3-b 1,4 benzodiazepin-6-on CS207619B2 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
CS798394A CS207620B2 (cs) 1977-05-31 1979-12-04 Způsob výroby nových derivátů 5,11-dihydro-BH-pyrido [ 2,3-b ] [ 1,4 ] - benzodiazepin-6-onu

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19772724501 DE2724501A1 (de) 1977-05-31 1977-05-31 Neue, in 11-stellung substituierte 5,11-dihydro-6h-pyrido eckige klammer auf 2,3-b eckige klammer zu eckige klammer auf 1,4 eckige klammer zu benzodiazepin-6- one, verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel

Publications (1)

Publication Number Publication Date
CS207619B2 true CS207619B2 (en) 1981-08-31

Family

ID=6010292

Family Applications (1)

Application Number Title Priority Date Filing Date
CS783473A CS207619B2 (en) 1977-05-31 1978-05-29 Method of making the new derivatives of 5,11-dihydro-6h-pyrido 2,3-b 1,4 benzodiazepin-6-on

Country Status (31)

Country Link
US (1) US4213985A (de)
JP (1) JPS543097A (de)
AT (1) AT361930B (de)
AU (1) AU516856B2 (de)
BE (1) BE867640A (de)
BG (2) BG28713A3 (de)
CA (1) CA1084918A (de)
CH (1) CH637653A5 (de)
CS (1) CS207619B2 (de)
DD (1) DD137105A5 (de)
DE (1) DE2724501A1 (de)
DK (1) DK239478A (de)
ES (2) ES470271A1 (de)
FI (1) FI63029C (de)
FR (1) FR2392992A1 (de)
GB (1) GB1569251A (de)
GR (1) GR64236B (de)
HK (1) HK13681A (de)
HU (1) HU180998B (de)
IE (1) IE46908B1 (de)
IL (1) IL54814A (de)
MY (1) MY8100361A (de)
NL (1) NL7805849A (de)
NO (1) NO149037C (de)
NZ (1) NZ187427A (de)
PH (1) PH14613A (de)
PL (2) PL113623B1 (de)
PT (1) PT68113A (de)
RO (1) RO79048A (de)
SE (1) SE7806289L (de)
ZA (1) ZA783085B (de)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB2053187A (en) * 1979-07-09 1981-02-04 Grissmann Chem Ltd Process for preparing pyrenzepine
IT1130973B (it) * 1980-03-17 1986-06-18 Microsules Argentina Sa De S C Processo per la preparazione di derivati di 5,11-di-idro-6h-pirido(2,3-b) (1,4)-benzodiazepin-6-one,derivati finali ed intermedi di sintesi in tal modo ottenuti
DE3113094A1 (de) * 1981-04-01 1982-10-21 Basf Ag, 6700 Ludwigshafen 5,6-dihydro-11-alkylen-morphantridin-6-one, ihre herstellung und diese enthaltende arzneimittel
DE3212794A1 (de) * 1982-04-06 1983-10-13 Basf Ag, 6700 Ludwigshafen 5,6-dihydro-11-alkylen-morphantridin-6-one, ihre herstellung und diese enthaltende arzneimittel
IT1212742B (it) * 1983-05-17 1989-11-30 Dompe Farmaceutici Spa Derivati dibenzo [1,4]diazepinonici pirido [1,4] benzodiazepinonici,pirido [1,5] benzodiazepinonici e loro attivita' farmacologica
DE3802334A1 (de) * 1988-01-27 1989-08-10 Thomae Gmbh Dr K Neue kondensierte diazepinone, verfahren zu ihrer herstellung und diese verbindungen enthaltende arzneimittel
US5298508A (en) * 1988-07-19 1994-03-29 The United States Of America As Represented By The Department Of Health And Human Services Irreversible inhibitors of adenosine receptors
US5264432A (en) * 1989-07-31 1993-11-23 Arzneimittelwerk Dresden G.M.B.H 5-(1-aminoacyl)-5,10-dihydro-11H-dibenzo[b,e](1,4)diazepin-11-ones
US5324832A (en) * 1991-07-03 1994-06-28 The United States Of America As Represented By The Department Of Health And Human Services Muscarinic antagonists
US6316423B1 (en) 1996-04-10 2001-11-13 The United States Of America As Represented By The Departmant Of Health And Human Services Method of treating ischemic, hypoxic and anoxic brain damage
GB0006337D0 (en) 2000-03-16 2000-05-03 Hopkinsons Ltd Fluid energy reduction valve
WO2010081825A2 (en) 2009-01-13 2010-07-22 Proteosys Ag Pirenzepine as an agent in cancer treatment

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1795183B1 (de) * 1968-08-20 1972-07-20 Thomae Gmbh Dr K 5,11-Dihydro-6H-pyrido[2,3-b][1,4]benzodiazepin-6-on-derivate und Arzneimittel
FI50242C (fi) * 1969-07-18 1976-01-12 Thomae Gmbh Dr K Menetelmä valmistaa farmakologisesti aktiivisia uusia diallyyliaminoal kanoyylidibenso- tai pyridobenso-diatsepiineja ja niiden happoadditios uoloja.

Also Published As

Publication number Publication date
GR64236B (en) 1980-02-19
HU180998B (en) 1983-05-30
CA1084918A (en) 1980-09-02
PL113623B1 (en) 1980-12-31
PT68113A (de) 1978-06-01
ES473464A1 (es) 1979-05-01
FR2392992A1 (fr) 1978-12-29
PL214168A1 (de) 1979-11-05
GB1569251A (en) 1980-06-11
NO149037C (no) 1984-02-01
MY8100361A (en) 1981-12-31
ATA367978A (de) 1980-09-15
PL114573B1 (en) 1981-02-28
SE7806289L (sv) 1978-12-01
RO79048A (ro) 1982-06-25
ES470271A1 (es) 1979-01-01
PL207190A1 (pl) 1979-07-16
IL54814A0 (en) 1978-07-31
US4213985A (en) 1980-07-22
IL54814A (en) 1981-09-13
IE46908B1 (en) 1983-11-02
BG28713A3 (en) 1980-06-16
DD137105A5 (de) 1979-08-15
FR2392992B1 (de) 1982-10-22
AT361930B (de) 1981-04-10
CH637653A5 (de) 1983-08-15
FI63029C (fi) 1983-04-11
BG28714A4 (en) 1980-06-16
FI781667A (fi) 1978-12-01
ZA783085B (en) 1980-02-27
DK239478A (da) 1978-12-01
BE867640A (fr) 1978-11-30
FI63029B (fi) 1982-12-31
HK13681A (en) 1981-04-16
PH14613A (en) 1981-10-02
NZ187427A (en) 1980-11-28
DE2724501A1 (de) 1978-12-21
NL7805849A (nl) 1978-12-04
JPS543097A (en) 1979-01-11
IE781072L (en) 1978-11-21
NO149037B (no) 1983-10-24
AU516856B2 (en) 1981-06-25
AU3662378A (en) 1979-12-06
NO781879L (no) 1978-12-01

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CS207620B2 (cs) Způsob výroby nových derivátů 5,11-dihydro-BH-pyrido [ 2,3-b ] [ 1,4 ] - benzodiazepin-6-onu