CS205010B2 - Method of producing 7-hydroxy estradiols - Google Patents

Method of producing 7-hydroxy estradiols Download PDF

Info

Publication number
CS205010B2
CS205010B2 CS756759A CS752576A CS205010B2 CS 205010 B2 CS205010 B2 CS 205010B2 CS 756759 A CS756759 A CS 756759A CS 752576 A CS752576 A CS 752576A CS 205010 B2 CS205010 B2 CS 205010B2
Authority
CS
Czechoslovakia
Prior art keywords
acid
group
formula
ethynyl
hydroxy
Prior art date
Application number
CS756759A
Other languages
Czech (cs)
English (en)
Inventor
Karl Petzoldt
Hans-Joerg Vidic
Klaus Prezewowsky
Yukishige Nishino
Rudolf Wiechert
Original Assignee
Laurent Henry
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from DE2449327A external-priority patent/DE2449327C2/de
Priority claimed from DE19752535997 external-priority patent/DE2535997A1/de
Application filed by Laurent Henry filed Critical Laurent Henry
Publication of CS205010B2 publication Critical patent/CS205010B2/cs

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J31/00—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring
    • C07J31/006—Normal steroids containing one or more sulfur atoms not belonging to a hetero ring not covered by C07J31/003
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C07J1/0051—Estrane derivatives
    • C07J1/0059—Estrane derivatives substituted in position 17 by a keto group
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C07J1/0051—Estrane derivatives
    • C07J1/0081—Substituted in position 17 alfa and 17 beta
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C07J1/0051—Estrane derivatives
    • C07J1/0081—Substituted in position 17 alfa and 17 beta
    • C07J1/0088—Substituted in position 17 alfa and 17 beta the substituent in position 17 alfa being an unsaturated hydrocarbon group
    • C07J1/0096—Alkynyl derivatives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J17/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, having an oxygen-containing hetero ring not condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10—TECHNICAL SUBJECTS COVERED BY FORMER USPC
    • Y10S—TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10S435/00—Chemistry: molecular biology and microbiology
    • Y10S435/8215—Microorganisms
    • Y10S435/911—Microorganisms using fungi
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10—TECHNICAL SUBJECTS COVERED BY FORMER USPC
    • Y10S—TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10S435/00—Chemistry: molecular biology and microbiology
    • Y10S435/8215—Microorganisms
    • Y10S435/911—Microorganisms using fungi
    • Y10S435/912—Absidia
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10—TECHNICAL SUBJECTS COVERED BY FORMER USPC
    • Y10S—TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10S435/00—Chemistry: molecular biology and microbiology
    • Y10S435/8215—Microorganisms
    • Y10S435/911—Microorganisms using fungi
    • Y10S435/913—Aspergillus
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10—TECHNICAL SUBJECTS COVERED BY FORMER USPC
    • Y10S—TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10S435/00—Chemistry: molecular biology and microbiology
    • Y10S435/8215—Microorganisms
    • Y10S435/911—Microorganisms using fungi
    • Y10S435/939—Rhizopus

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Steroid Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
CS756759A 1974-10-14 1975-10-06 Method of producing 7-hydroxy estradiols CS205010B2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE2449327A DE2449327C2 (de) 1974-10-14 1974-10-14 7 α-Hydroxy-östradiole, Verfahren zu deren Herstellung und diese enthaltende Arzneimittel
DE19752535997 DE2535997A1 (de) 1975-08-08 1975-08-08 7-hydroxy-oestradiole

Publications (1)

Publication Number Publication Date
CS205010B2 true CS205010B2 (en) 1981-04-30

Family

ID=25767825

Family Applications (2)

Application Number Title Priority Date Filing Date
CS756759A CS205009B2 (en) 1974-10-14 1975-10-06 Process for preparing 7-hydroxyestradioles
CS756759A CS205010B2 (en) 1974-10-14 1975-10-06 Method of producing 7-hydroxy estradiols

Family Applications Before (1)

Application Number Title Priority Date Filing Date
CS756759A CS205009B2 (en) 1974-10-14 1975-10-06 Process for preparing 7-hydroxyestradioles

Country Status (23)

Country Link
US (1) US4011314A (de)
JP (1) JPS5165747A (de)
AT (1) AT348695B (de)
CA (1) CA1054143A (de)
CH (2) CH619240A5 (de)
CS (2) CS205009B2 (de)
DD (1) DD125588A5 (de)
DK (1) DK135378C (de)
ES (1) ES441784A1 (de)
FI (1) FI54603C (de)
FR (1) FR2287908A1 (de)
GB (1) GB1528796A (de)
HU (1) HU176715B (de)
IE (1) IE42167B1 (de)
IL (1) IL48276A (de)
NL (1) NL7512041A (de)
NO (1) NO140824C (de)
NZ (1) NZ178886A (de)
PH (1) PH13802A (de)
PL (2) PL103989B1 (de)
SE (1) SE405254B (de)
SU (2) SU676170A3 (de)
YU (2) YU243975A (de)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8327256D0 (en) * 1983-10-12 1983-11-16 Ici Plc Steroid derivatives
DE3741800A1 (de) * 1987-12-07 1989-06-15 Schering Ag 17-halogenmethylen-estratriene
US5861431A (en) * 1995-06-07 1999-01-19 Iotek, Inc. Incontinence treatment
JP2000511404A (ja) 1996-04-09 2000-09-05 ビー・テイー・ジー・インターナシヨナル・リミテツド 神経精神、免疫又は内分泌障害を治療するための７α置換ステロイドの使用
EP2322182A1 (de) 1999-09-30 2011-05-18 Harbor BioSciences, Inc. Androstenolderivate als Androgenrezeptormodulator
GB0003524D0 (en) * 2000-02-15 2000-04-05 Btg Int Ltd Cytoprotective steroids (II)
GB2363983A (en) * 2000-06-29 2002-01-16 Hunter Fleming Ltd Protection against neuronal damage using 7-hydroxyepiandrosterone
DK1624878T3 (da) * 2003-05-22 2007-01-08 Pantarhei Bioscience Bv Anvendelse af præparater som omfatter en östrogen komponent til behandling og forebyggelse af muskel-skelet-smerte
GB0403889D0 (en) * 2004-02-21 2004-03-24 Univ Edinburgh Uses of er-beta modulators
US7910755B2 (en) 2004-09-29 2011-03-22 Harbor Biosciences, Inc. Stem cell expansion and uses

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3115444A (en) * 1962-01-22 1963-12-24 Olin Mathieson Process for microbial hydroxylation of steroids containing aromatic alpha-rings

Also Published As

Publication number Publication date
DK135378C (da) 1977-10-03
IE42167B1 (en) 1980-06-18
PL103989B1 (pl) 1979-07-31
NL7512041A (nl) 1976-04-20
DK439975A (da) 1976-04-15
HU176715B (en) 1981-04-28
GB1528796A (en) 1978-10-18
YU243975A (en) 1982-06-30
IE42167L (en) 1976-04-14
US4011314A (en) 1977-03-08
CS205009B2 (en) 1981-04-30
NZ178886A (en) 1978-04-28
PH13802A (en) 1980-10-01
IL48276A (en) 1979-03-12
IL48276A0 (en) 1975-12-31
NO140824B (no) 1979-08-13
FR2287908B1 (de) 1980-04-30
JPS5165747A (en) 1976-06-07
ES441784A1 (es) 1977-04-01
ATA775475A (de) 1978-07-15
NO140824C (no) 1979-11-21
DD125588A5 (de) 1977-05-04
NO753455L (de) 1976-04-20
DK135378B (da) 1977-04-18
SE7511438L (sv) 1976-04-15
SE405254B (sv) 1978-11-27
FR2287908A1 (fr) 1976-05-14
CA1054143A (en) 1979-05-08
PL101461B1 (pl) 1978-12-30
CH619240A5 (de) 1980-09-15
YU294281A (en) 1982-06-30
AU8571075A (en) 1977-04-21
SU677666A1 (ru) 1981-11-30
AT348695B (de) 1979-02-26
FI752836A (de) 1976-04-15
FI54603B (fi) 1978-09-29
SU676170A3 (ru) 1979-07-25
SU677666A3 (en) 1981-11-30
FI54603C (fi) 1979-01-10
CH619268A5 (de) 1980-09-15

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