CS196333B2 - Method of producing/alpha-aminoacetyl/benzene derivatives - Google Patents

Method of producing/alpha-aminoacetyl/benzene derivatives Download PDF

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Publication number
CS196333B2
CS196333B2 CS767604A CS760476A CS196333B2 CS 196333 B2 CS196333 B2 CS 196333B2 CS 767604 A CS767604 A CS 767604A CS 760476 A CS760476 A CS 760476A CS 196333 B2 CS196333 B2 CS 196333B2
Authority
CS
Czechoslovakia
Prior art keywords
formula
pharmaceutically acceptable
acid
methyl
compound
Prior art date
Application number
CS767604A
Other languages
Czech (cs)
English (en)
Inventor
Clifford R Hughes
Stephen J Jackson
John Preston
Peter L Walton
Original Assignee
Ici Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ici Ltd filed Critical Ici Ltd
Priority to CS776119A priority Critical patent/CS196334B2/cs
Publication of CS196333B2 publication Critical patent/CS196333B2/cs

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
    • C07D263/30—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D263/34—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C323/00—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C59/00—Compounds having carboxyl groups bound to acyclic carbon atoms and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups
    • C07C59/40—Unsaturated compounds
    • C07C59/76—Unsaturated compounds containing keto groups
    • C07C59/88—Unsaturated compounds containing keto groups containing halogen
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
    • C07D295/18—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carboxylic acids, or sulfur or nitrogen analogues thereof
    • C07D295/182—Radicals derived from carboxylic acids
    • C07D295/185—Radicals derived from carboxylic acids from aliphatic carboxylic acids

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Diabetes (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Hematology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
CS767604A 1975-11-25 1976-11-24 Method of producing/alpha-aminoacetyl/benzene derivatives CS196333B2 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
CS776119A CS196334B2 (cs) 1975-11-25 1977-09-21 Způsob výroby derivátů («-aminoacntylj benzenu

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB48402/75A GB1559977A (en) 1975-11-25 1975-11-25 Amines

Publications (1)

Publication Number Publication Date
CS196333B2 true CS196333B2 (en) 1980-03-31

Family

ID=10448487

Family Applications (1)

Application Number Title Priority Date Filing Date
CS767604A CS196333B2 (en) 1975-11-25 1976-11-24 Method of producing/alpha-aminoacetyl/benzene derivatives

Country Status (28)

Country Link
US (1) US4105790A (da)
JP (2) JPS5265240A (da)
AR (1) AR215871A1 (da)
AT (1) AT348993B (da)
AU (1) AU503657B2 (da)
BE (1) BE848707A (da)
CA (1) CA1068695A (da)
CH (1) CH624383A5 (da)
CS (1) CS196333B2 (da)
DD (1) DD127474A5 (da)
DE (1) DE2653635C2 (da)
DK (1) DK531276A (da)
ES (2) ES453632A1 (da)
FI (1) FI763399A (da)
FR (1) FR2332747A1 (da)
GB (1) GB1559977A (da)
IE (1) IE44030B1 (da)
IL (1) IL50904A (da)
IN (1) IN145003B (da)
LU (1) LU76251A1 (da)
NL (1) NL7613081A (da)
NO (1) NO764012L (da)
NZ (1) NZ182581A (da)
PL (2) PL105491B1 (da)
PT (1) PT65892B (da)
SE (1) SE7613079L (da)
SU (1) SU722481A3 (da)
ZA (1) ZA766696B (da)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH02130656U (da) * 1989-03-31 1990-10-29
JPH028457U (da) * 1988-07-01 1990-01-19
US5348969A (en) * 1992-04-03 1994-09-20 Bristol-Myers Squibb Company Diphenyloxazolyl-oxazoles as platelet aggregation inhibitors
ATE230395T1 (de) 1993-06-25 2003-01-15 Merrell Pharma Inc Neue zwischenprodukte für die herstellung von antihistaminschen 4- diphenylmethyl/diphenylmethoxypiperidin-derivat n
US6147216A (en) * 1993-06-25 2000-11-14 Merrell Pharmaceuticals Inc. Intermediates useful for the preparation of antihistaminic piperidine derivatives
US6683094B2 (en) 1998-07-02 2004-01-27 Aventis Pharmaceuticals Inc. Antihistaminic piperidine derivatives and intermediates for the preparation thereof
US6689898B2 (en) 1998-07-02 2004-02-10 Aventis Pharmaceuticals Inc. Antihistaminic piperidine derivatives and intermediates for the preparation thereof
FR2880887B1 (fr) * 2005-01-14 2009-01-30 Merck Sante Soc Par Actions Si Derives d'hydroxyphenols, procedes pour leur preparation, compositions pharmaceutiques les contenant et applications en therapeutique
TW200740779A (en) 2005-07-22 2007-11-01 Mitsubishi Pharma Corp Intermediate compound for synthesizing pharmaceutical agent and production method thereof
CN106661139A (zh) * 2014-07-16 2017-05-10 株式会社艾迪科 感光性组合物

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH543472A (fr) * 1969-01-31 1973-10-31 Orchimed Sa Procédé pour la préparation d'acides phénoxyalcoyl-carboxyliques

Also Published As

Publication number Publication date
CH624383A5 (da) 1981-07-31
JPS61158922A (ja) 1986-07-18
CA1068695A (en) 1979-12-25
AU1962576A (en) 1978-05-25
SE7613079L (sv) 1977-05-26
FR2332747A1 (fr) 1977-06-24
LU76251A1 (da) 1977-12-13
IL50904A (en) 1980-02-29
SU722481A3 (ru) 1980-03-15
ZA766696B (en) 1977-10-26
US4105790A (en) 1978-08-08
JPS5265240A (en) 1977-05-30
DE2653635C2 (de) 1986-10-02
NZ182581A (en) 1978-09-20
PL193861A1 (pl) 1978-03-28
NO764012L (da) 1977-05-26
FI763399A (da) 1977-05-26
IE44030L (en) 1977-05-25
NL7613081A (nl) 1977-05-27
BE848707A (fr) 1977-05-24
PL105799B1 (pl) 1979-10-31
PT65892A (en) 1976-12-01
AT348993B (de) 1979-03-12
JPS6360004B2 (da) 1988-11-22
IE44030B1 (en) 1981-07-29
IN145003B (da) 1978-08-12
AU503657B2 (en) 1979-09-13
PL105491B1 (pl) 1979-10-31
FR2332747B1 (da) 1980-03-14
PT65892B (en) 1978-05-18
GB1559977A (en) 1980-01-30
DD127474A5 (da) 1977-09-28
JPS6120538B2 (da) 1986-05-22
DE2653635A1 (de) 1977-06-02
AR215871A1 (es) 1979-11-15
ES453632A1 (es) 1978-03-16
DK531276A (da) 1977-05-26
ES465152A1 (es) 1978-10-01
ATA870976A (de) 1978-08-15

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