CS195707B2 - Method of producing novel n up 4-substituted derivatives of 1,3,4,5-tetrahydro-2h-1,4-benzodiazepine-2-one - Google Patents
Method of producing novel n up 4-substituted derivatives of 1,3,4,5-tetrahydro-2h-1,4-benzodiazepine-2-one Download PDFInfo
- Publication number
- CS195707B2 CS195707B2 CS754443A CS444375A CS195707B2 CS 195707 B2 CS195707 B2 CS 195707B2 CS 754443 A CS754443 A CS 754443A CS 444375 A CS444375 A CS 444375A CS 195707 B2 CS195707 B2 CS 195707B2
- Authority
- CS
- Czechoslovakia
- Prior art keywords
- formula
- compound
- defined above
- tetrahydro
- reaction
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D243/00—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
- C07D243/06—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
- C07D243/10—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
- C07D243/14—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
- C07D243/16—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
- C07D243/18—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals substituted in position 2 by nitrogen, oxygen or sulfur atoms
- C07D243/24—Oxygen atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P39/00—General protective or antinoxious agents
- A61P39/02—Antidotes
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D243/00—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
- C07D243/06—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
- C07D243/10—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
- C07D243/14—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
- C07D243/16—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
- C07D243/18—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals substituted in position 2 by nitrogen, oxygen or sulfur atoms
- C07D243/24—Oxygen atoms
- C07D243/26—Preparation from compounds already containing the benzodiazepine skeleton
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Anesthesiology (AREA)
- Toxicology (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| HURI540A HU170623B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | 1974-06-25 | 1974-06-25 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CS195707B2 true CS195707B2 (en) | 1980-02-29 |
Family
ID=11000952
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CS754443A CS195707B2 (en) | 1974-06-25 | 1975-06-23 | Method of producing novel n up 4-substituted derivatives of 1,3,4,5-tetrahydro-2h-1,4-benzodiazepine-2-one |
Country Status (21)
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| HU187262B (en) * | 1979-08-16 | 1985-12-28 | Richter Gedeon Vegyeszet | Process for preparing new tetrahydro-1,4-benzodiazepin-2-ones |
| CA2370141A1 (en) | 1999-05-26 | 2000-12-07 | James D. Rodgers | 1,4-benzodiazepin-2-ones useful as hiv reverse transcriptase inhibitors |
| CN105716725B (zh) * | 2016-03-10 | 2019-02-12 | 中国科学院光电技术研究所 | 一种基于叠层扫描的相位差波前探测和图像复原方法 |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3236838A (en) * | 1964-06-09 | 1966-02-22 | Hoffmann La Roche | Certain 1-substituted-benzodiazepin-2-one compounds |
-
1974
- 1974-06-25 HU HURI540A patent/HU170623B/hu not_active IP Right Cessation
-
1975
- 1975-06-17 IL IL47495A patent/IL47495A/xx unknown
- 1975-06-18 SE SE7507039A patent/SE423711B/xx not_active IP Right Cessation
- 1975-06-19 FR FR7519196A patent/FR2276054A1/fr active Granted
- 1975-06-19 AU AU82238/75A patent/AU499054B2/en not_active Expired
- 1975-06-23 DE DE19752527901 patent/DE2527901A1/de not_active Withdrawn
- 1975-06-23 CS CS754443A patent/CS195707B2/cs unknown
- 1975-06-23 US US05/589,079 patent/US4021421A/en not_active Expired - Lifetime
- 1975-06-23 CH CH811075A patent/CH632254A5/de not_active IP Right Cessation
- 1975-06-24 DK DK284675A patent/DK284675A/da not_active Application Discontinuation
- 1975-06-24 SU SU752149105A patent/SU1080744A3/ru active
- 1975-06-24 BE BE157631A patent/BE830582A/xx not_active IP Right Cessation
- 1975-06-24 JP JP7854575A patent/JPS541716B2/ja not_active Expired
- 1975-06-24 AT AT481975A patent/AT344698B/de not_active IP Right Cessation
- 1975-06-24 DD DD186853A patent/DD123887A5/xx unknown
- 1975-06-24 BG BG030386A patent/BG32569A3/xx unknown
- 1975-06-24 CA CA230,062A patent/CA1047493A/en not_active Expired
- 1975-06-24 YU YU01610/75A patent/YU161075A/xx unknown
- 1975-06-24 BG BG032384A patent/BG32570A3/xx unknown
- 1975-06-24 PL PL1975181497A patent/PL101952B1/pl unknown
- 1975-06-25 GB GB26920/75A patent/GB1509445A/en not_active Expired
- 1975-06-25 NL NL7507556A patent/NL7507556A/xx unknown
-
1977
- 1977-11-25 JP JP52140842A patent/JPS6026113B2/ja not_active Expired
-
1979
- 1979-04-11 CH CH342479A patent/CH634835A5/de not_active IP Right Cessation
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