CR9864A - Formas de presentacion farmaceutica solidas de administracion oral con liberacion rapida de principio activo - Google Patents

Formas de presentacion farmaceutica solidas de administracion oral con liberacion rapida de principio activo

Info

Publication number
CR9864A
CR9864A CR9864A CR9864A CR9864A CR 9864 A CR9864 A CR 9864A CR 9864 A CR9864 A CR 9864A CR 9864 A CR9864 A CR 9864A CR 9864 A CR9864 A CR 9864A
Authority
CR
Costa Rica
Prior art keywords
oral administration
solid pharmaceutical
quick release
active principle
prophylaxis
Prior art date
Application number
CR9864A
Other languages
English (en)
Inventor
Klaus Benke
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=37852804&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CR9864(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed filed Critical
Publication of CR9864A publication Critical patent/CR9864A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2072Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2077Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/53751,4-Oxazines, e.g. morpholine
    • A61K31/53771,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1682Processes
    • A61K9/1694Processes resulting in granules or microspheres of the matrix type containing more than 5% of excipient
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Abstract

La invencion se refiere a formas de dosificacion farmaceutica solidas de administracion oral con liberacion del principio activo rapida, 5-cloro-N-({5S)-2-oxo-3-[4-(3-oxo-4-morfolinil)fenil]-1,3-oxazolidin-5-il}metil)-2- tiofenocarboxamida, que estan en forma amorfa y/o contienen una modificacion cristalina termodinamicamente metaestable con liberacion rapida de principio activo, asi como a procedimientos para su preparacion, su uso como medicamento, su uso para profilaxis, profilaxis secundaria y/o tratamiento de enfermedades, asi como su uso para la preparacion de un medicamento para la profilaxis, profilaxis secundaria y/o tratamiento de enfermedades.
CR9864A 2005-10-04 2008-04-03 Formas de presentacion farmaceutica solidas de administracion oral con liberacion rapida de principio activo CR9864A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE102005047561A DE102005047561A1 (de) 2005-10-04 2005-10-04 Feste, oral applizierbare pharmazeutische Darreichungsformen mit schneller Wirkstofffreisetzung

Publications (1)

Publication Number Publication Date
CR9864A true CR9864A (es) 2008-10-31

Family

ID=37852804

Family Applications (1)

Application Number Title Priority Date Filing Date
CR9864A CR9864A (es) 2005-10-04 2008-04-03 Formas de presentacion farmaceutica solidas de administracion oral con liberacion rapida de principio activo

Country Status (27)

Country Link
US (1) US8586082B2 (es)
EP (1) EP1957048A2 (es)
JP (1) JP5147703B2 (es)
KR (1) KR101445398B1 (es)
CN (1) CN101321517B (es)
AR (1) AR056564A1 (es)
AU (1) AU2006299192B2 (es)
BR (1) BRPI0616874A2 (es)
CA (1) CA2624306C (es)
CR (1) CR9864A (es)
CU (1) CU23808B7 (es)
DE (1) DE102005047561A1 (es)
DO (1) DOP2006000209A (es)
EC (1) ECSP088339A (es)
GT (1) GT200600445A (es)
HK (1) HK1127284A1 (es)
IL (1) IL190618A0 (es)
MY (1) MY143351A (es)
NZ (1) NZ567094A (es)
PE (1) PE20070588A1 (es)
RU (1) RU2440119C2 (es)
SV (1) SV2009002857A (es)
TW (1) TWI389691B (es)
UA (1) UA90545C2 (es)
UY (1) UY29835A1 (es)
WO (1) WO2007039122A2 (es)
ZA (1) ZA200802873B (es)

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KR102333463B1 (ko) * 2014-07-02 2021-12-03 한미약품 주식회사 리바록사반을 포함하는 경구 투여용 약학 조성물 및 이의 제조방법
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WO2007039122A3 (de) 2007-10-11
NZ567094A (en) 2011-05-27
DE102005047561A1 (de) 2007-04-05
DOP2006000209A (es) 2007-04-30
CU23808B7 (es) 2012-04-15
AR056564A1 (es) 2007-10-10
EP1957048A2 (de) 2008-08-20
CU20080052A7 (es) 2011-04-26
PE20070588A1 (es) 2007-08-17
CN101321517B (zh) 2012-11-28
US20100151011A1 (en) 2010-06-17
CN101321517A (zh) 2008-12-10
UA90545C2 (ru) 2010-05-11
RU2008116831A (ru) 2009-11-10
TW200803866A (en) 2008-01-16
RU2440119C2 (ru) 2012-01-20
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ECSP088339A (es) 2008-06-30
CA2624306C (en) 2014-12-09
TWI389691B (zh) 2013-03-21
SV2009002857A (es) 2009-01-14
UY29835A1 (es) 2007-05-31
WO2007039122A2 (de) 2007-04-12
MY143351A (en) 2011-04-29
JP2009510138A (ja) 2009-03-12
AU2006299192A1 (en) 2007-04-12
AU2006299192B2 (en) 2012-04-19
CA2624306A1 (en) 2007-04-12
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US8586082B2 (en) 2013-11-19
JP5147703B2 (ja) 2013-02-20
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