CR11601A - Pirimidil ciclopentanos hidroxilados en forma de inhibidores de akt proteina quinasa - Google Patents
Pirimidil ciclopentanos hidroxilados en forma de inhibidores de akt proteina quinasaInfo
- Publication number
- CR11601A CR11601A CR11601A CR11601A CR11601A CR 11601 A CR11601 A CR 11601A CR 11601 A CR11601 A CR 11601A CR 11601 A CR11601 A CR 11601A CR 11601 A CR11601 A CR 11601A
- Authority
- CR
- Costa Rica
- Prior art keywords
- pyrimidil
- quinasa
- cyclopentanes
- proteina
- akt
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Pain & Pain Management (AREA)
- Hospice & Palliative Care (AREA)
- Cardiology (AREA)
- Psychiatry (AREA)
- Heart & Thoracic Surgery (AREA)
- Rheumatology (AREA)
- Dermatology (AREA)
- Endocrinology (AREA)
- Reproductive Health (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Preparation Of Compounds By Using Micro-Organisms (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Abstract
La presente invencion provee compuestos, que incluyen sales aceptables para uso farmaceutico, que comprenden la formula I.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US2009208P | 2008-01-09 | 2008-01-09 |
Publications (1)
Publication Number | Publication Date |
---|---|
CR11601A true CR11601A (es) | 2010-08-19 |
Family
ID=40552865
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CR11601A CR11601A (es) | 2008-01-09 | 2010-07-27 | Pirimidil ciclopentanos hidroxilados en forma de inhibidores de akt proteina quinasa |
Country Status (18)
Country | Link |
---|---|
US (1) | US8835434B2 (es) |
EP (1) | EP2247578B1 (es) |
JP (1) | JP5346345B2 (es) |
KR (1) | KR101624753B1 (es) |
CN (1) | CN101932564B (es) |
AU (1) | AU2009204025B2 (es) |
BR (1) | BRPI0906798A2 (es) |
CA (1) | CA2711699A1 (es) |
CR (1) | CR11601A (es) |
EC (1) | ECSP10010389A (es) |
ES (1) | ES2422733T3 (es) |
IL (1) | IL206575A0 (es) |
MA (1) | MA32183B1 (es) |
NZ (1) | NZ586346A (es) |
RU (1) | RU2504542C2 (es) |
UA (1) | UA100545C2 (es) |
WO (1) | WO2009089459A1 (es) |
ZA (1) | ZA201004769B (es) |
Families Citing this family (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN103396409B (zh) * | 2007-07-05 | 2015-03-11 | 阵列生物制药公司 | 作为akt蛋白激酶抑制剂的嘧啶基环戊烷 |
US9409886B2 (en) | 2007-07-05 | 2016-08-09 | Array Biopharma Inc. | Pyrimidyl cyclopentanes as AKT protein kinase inhibitors |
US8846683B2 (en) | 2007-07-05 | 2014-09-30 | Array Biopharma, Inc. | Pyrimidyl cyclopentanes as Akt protein kinase inhibitors |
JP5608097B2 (ja) | 2008-01-08 | 2014-10-15 | アレイ バイオファーマ、インコーポレイテッド | キナーゼ阻害薬としてのピロロピリジン |
US8329709B2 (en) | 2008-01-09 | 2012-12-11 | Genentech, Inc. | 5H-cyclopenta[D]pyrimidines as AKT protein kinase inhibitors |
JP5608098B2 (ja) | 2008-01-09 | 2014-10-15 | アレイ バイオファーマ、インコーポレイテッド | キナーゼ阻害薬としてのピラゾロピリジン |
NZ702513A (en) * | 2012-05-17 | 2016-09-30 | Genentech Inc | Amorphous form of an akt inhibiting pyrimidinyl - cyclopentane compound, compositions and methods thereof |
WO2013173736A1 (en) * | 2012-05-17 | 2013-11-21 | Array Biopharma Inc. | Process for making hydroxylated cyclopentylpyrimidine compounds |
EP4282973A3 (en) | 2013-11-15 | 2024-03-27 | F. Hoffmann-La Roche AG | Processes for the preparation of pyrimidinylcyclopentane compounds |
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US4060615A (en) | 1976-02-18 | 1977-11-29 | Mead Johnson & Company | 2-Piperazinyl-6,7-dimethoxyquinazolines |
JPS562968A (en) | 1979-06-21 | 1981-01-13 | Mitsubishi Yuka Yakuhin Kk | Novel pyrimidine derivative |
JPS6270A (ja) | 1985-03-07 | 1987-01-06 | Sankyo Co Ltd | シクロペンタ〔d〕ピリミジン誘導体 |
WO1990007926A1 (en) | 1989-01-20 | 1990-07-26 | Pfizer Inc. | 3-(1,2,5,6-tetrahydropyridyl)-pyrrolopyridines |
CA2146333A1 (en) | 1992-10-05 | 1994-04-14 | Tomio Kimura | Pyrimidine compound |
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GB9416189D0 (en) | 1994-08-10 | 1994-09-28 | Merck Sharp & Dohme | Therapeutic agents |
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US5525625A (en) | 1995-01-24 | 1996-06-11 | Warner-Lambert Company | 2-(2-Amino-3-methoxyphenyl)-4-oxo-4H-[1]benzopyran for treating proliferative disorders |
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ZA979961B (en) | 1996-11-15 | 1999-05-05 | Lilly Co Eli | 5-HT1F agonists |
UA73073C2 (uk) | 1997-04-03 | 2005-06-15 | Уайт Холдінгз Корпорейшн | Заміщені 3-ціанохіноліни, спосіб їх одержання та фармацевтична композиція |
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ES2274572T3 (es) | 1997-07-01 | 2007-05-16 | Warner-Lambert Company Llc | Derivados de acido 2-(4-bromo- o 4-yodo-fenilamino) benzoico y su uso como inhibidor de mek. |
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DE69943144D1 (de) | 1998-03-31 | 2011-03-03 | Kyowa Hakko Kirin Co Ltd | Stickstoffenthaltende heterocyclische verbindungen |
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CA2358438A1 (en) | 1999-01-07 | 2000-07-13 | David Thomas Dudley | Antiviral method using mek inhibitors |
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ATE250932T1 (de) | 1999-07-16 | 2003-10-15 | Warner Lambert Co | Verfahren zur behandlung von chronischem schmerz durch verabreichung von einem mek hemmer |
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NO320062B1 (no) * | 2003-11-19 | 2005-10-17 | New Interaction Devices And Te | Anordning til a detektere naerhet mellom et forste objekt (malobjekt) og et annet objekt (referanseobjekt), samt tegne-, skrive- og/eller pekeredskap for datapresentasjon etc. |
KR101223914B1 (ko) * | 2003-11-21 | 2013-01-18 | 어레이 바이오파마 인크. | Akt 단백질 키나제 억제제 |
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EA200800664A1 (ru) | 2005-10-13 | 2009-02-27 | Глаксо Груп Лимитед | Производные пирролопиримидина в качестве ингибиторов syk |
US20090253687A1 (en) | 2005-12-28 | 2009-10-08 | Shoji Fukumoto | Fused Heterocyclic Compounds and Their Use as Mineralocorticoid Receptor Ligands |
US20090124610A1 (en) | 2006-04-25 | 2009-05-14 | Gordon Saxty | Pharmaceutical compounds |
RU2008152171A (ru) | 2006-07-05 | 2010-08-10 | Интермьюн, Инк. (Us) | Новые ингибиторы вирусной репликации гепатита с |
US7910747B2 (en) | 2006-07-06 | 2011-03-22 | Bristol-Myers Squibb Company | Phosphonate and phosphinate pyrazolylamide glucokinase activators |
TW200808325A (en) | 2006-07-06 | 2008-02-16 | Astrazeneca Ab | Novel compounds |
US8063050B2 (en) | 2006-07-06 | 2011-11-22 | Array Biopharma Inc. | Hydroxylated and methoxylated pyrimidyl cyclopentanes as AKT protein kinase inhibitors |
EP2049478B1 (en) | 2006-07-06 | 2012-05-30 | Glaxo Group Limited | Substituted n-phenylmethyl -5-oxo-proline-2-amides as p2x7-receptor antagonists and their methods of use |
GB0613518D0 (en) | 2006-07-06 | 2006-08-16 | Phytopharm Plc | Chemical compounds |
MY147628A (en) | 2006-07-06 | 2012-12-31 | Array Biopharma Inc | Cyclopenta [d] pyrimidines as akt protein kinase inhibitors |
UA95641C2 (en) * | 2006-07-06 | 2011-08-25 | Эррей Биофарма Инк. | Hydroxylated cyclopenta [d] pyrimidines as akt protein kinase inhibitors |
JP4960450B2 (ja) | 2006-07-14 | 2012-06-27 | ノバルティス アーゲー | Alk−5阻害剤としてのピリミジン誘導体 |
WO2008012635A2 (en) | 2006-07-26 | 2008-01-31 | Pfizer Products Inc. | Amine derivatives useful as anticancer agents |
CN103396409B (zh) | 2007-07-05 | 2015-03-11 | 阵列生物制药公司 | 作为akt蛋白激酶抑制剂的嘧啶基环戊烷 |
-
2009
- 2009-01-09 CA CA2711699A patent/CA2711699A1/en not_active Withdrawn
- 2009-01-09 ES ES09700422T patent/ES2422733T3/es active Active
- 2009-01-09 NZ NZ586346A patent/NZ586346A/en not_active IP Right Cessation
- 2009-01-09 WO PCT/US2009/030610 patent/WO2009089459A1/en active Application Filing
- 2009-01-09 KR KR1020107017605A patent/KR101624753B1/ko active IP Right Grant
- 2009-01-09 BR BRPI0906798-1A patent/BRPI0906798A2/pt not_active Application Discontinuation
- 2009-01-09 CN CN2009801019017A patent/CN101932564B/zh active Active
- 2009-01-09 AU AU2009204025A patent/AU2009204025B2/en not_active Ceased
- 2009-01-09 EP EP09700422.0A patent/EP2247578B1/en active Active
- 2009-01-09 RU RU2010132911/04A patent/RU2504542C2/ru active
- 2009-01-09 JP JP2010542376A patent/JP5346345B2/ja active Active
- 2009-01-09 US US12/811,957 patent/US8835434B2/en active Active
- 2009-09-01 UA UAA201009871A patent/UA100545C2/ru unknown
-
2010
- 2010-06-23 IL IL206575A patent/IL206575A0/en unknown
- 2010-07-06 ZA ZA2010/04769A patent/ZA201004769B/en unknown
- 2010-07-23 MA MA33047A patent/MA32183B1/fr unknown
- 2010-07-27 CR CR11601A patent/CR11601A/es not_active Application Discontinuation
- 2010-08-06 EC EC2010010389A patent/ECSP10010389A/es unknown
Also Published As
Publication number | Publication date |
---|---|
ZA201004769B (en) | 2011-12-28 |
US8835434B2 (en) | 2014-09-16 |
EP2247578A1 (en) | 2010-11-10 |
RU2010132911A (ru) | 2012-02-20 |
AU2009204025A1 (en) | 2009-07-16 |
RU2504542C2 (ru) | 2014-01-20 |
KR20100118110A (ko) | 2010-11-04 |
JP5346345B2 (ja) | 2013-11-20 |
JP2011509308A (ja) | 2011-03-24 |
AU2009204025B2 (en) | 2014-02-20 |
CA2711699A1 (en) | 2009-07-16 |
BRPI0906798A2 (pt) | 2015-07-14 |
UA100545C2 (ru) | 2013-01-10 |
ES2422733T3 (es) | 2013-09-13 |
ECSP10010389A (es) | 2010-11-30 |
CN101932564A (zh) | 2010-12-29 |
US20110065716A1 (en) | 2011-03-17 |
WO2009089459A1 (en) | 2009-07-16 |
EP2247578B1 (en) | 2013-05-22 |
NZ586346A (en) | 2012-02-24 |
IL206575A0 (en) | 2010-12-30 |
KR101624753B1 (ko) | 2016-05-26 |
CN101932564B (zh) | 2012-12-26 |
MA32183B1 (fr) | 2011-04-01 |
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