CO6950480A2 - Tableta que contiene 7-[4-(4-benzo[b]tiofen-4-il-piperazin-1-il)butoxi]-1h-quinolin-2-ona o una de sus sales - Google Patents

Tableta que contiene 7-[4-(4-benzo[b]tiofen-4-il-piperazin-1-il)butoxi]-1h-quinolin-2-ona o una de sus sales

Info

Publication number
CO6950480A2
CO6950480A2 CO14098041A CO14098041A CO6950480A2 CO 6950480 A2 CO6950480 A2 CO 6950480A2 CO 14098041 A CO14098041 A CO 14098041A CO 14098041 A CO14098041 A CO 14098041A CO 6950480 A2 CO6950480 A2 CO 6950480A2
Authority
CO
Colombia
Prior art keywords
quinolin
thiophen
piperazin
benzo
butoxy
Prior art date
Application number
CO14098041A
Other languages
English (en)
Inventor
Yoshiharu Inoue
Original Assignee
Otsuka Pharma Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=48081918&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CO6950480(A2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Otsuka Pharma Co Ltd filed Critical Otsuka Pharma Co Ltd
Publication of CO6950480A2 publication Critical patent/CO6950480A2/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0053Mouth and digestive tract, i.e. intraoral and peroral administration
    • A61K9/0056Mouth soluble or dispersible forms; Suckable, eatable, chewable coherent forms; Forms rapidly disintegrating in the mouth; Lozenges; Lollipops; Bite capsules; Baked products; Baits or other oral forms for animals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/496Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2013Organic compounds, e.g. phospholipids, fats
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2013Organic compounds, e.g. phospholipids, fats
    • A61K9/2018Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2059Starch, including chemically or physically modified derivatives; Amylose; Amylopectin; Dextrin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806Coating materials
    • A61K9/2813Inorganic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806Coating materials
    • A61K9/2833Organic macromolecular compounds
    • A61K9/286Polysaccharides, e.g. gums; Cyclodextrin
    • A61K9/2866Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Physiology (AREA)
  • Zoology (AREA)
  • Inorganic Chemistry (AREA)
  • Nutrition Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Psychiatry (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
CO14098041A 2011-10-14 2014-05-07 Tableta que contiene 7-[4-(4-benzo[b]tiofen-4-il-piperazin-1-il)butoxi]-1h-quinolin-2-ona o una de sus sales CO6950480A2 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP2011227057 2011-10-14

Publications (1)

Publication Number Publication Date
CO6950480A2 true CO6950480A2 (es) 2014-05-20

Family

ID=48081918

Family Applications (1)

Application Number Title Priority Date Filing Date
CO14098041A CO6950480A2 (es) 2011-10-14 2014-05-07 Tableta que contiene 7-[4-(4-benzo[b]tiofen-4-il-piperazin-1-il)butoxi]-1h-quinolin-2-ona o una de sus sales

Country Status (32)

Country Link
US (7) US20140234417A1 (es)
EP (1) EP2767285B1 (es)
JP (2) JP6084161B2 (es)
KR (1) KR102072371B1 (es)
CN (2) CN107397730A (es)
AP (1) AP2014007564A0 (es)
AR (1) AR088319A1 (es)
AU (1) AU2012321723C1 (es)
BR (1) BR112014008603A2 (es)
CA (1) CA2851588C (es)
CL (1) CL2014000909A1 (es)
CO (1) CO6950480A2 (es)
CY (1) CY1122460T1 (es)
DK (1) DK2767285T3 (es)
EA (1) EA032930B1 (es)
ES (1) ES2762479T3 (es)
HR (1) HRP20200037T1 (es)
HU (1) HUE047493T2 (es)
IL (1) IL231513B (es)
IN (1) IN2014DN02055A (es)
JO (1) JO3753B1 (es)
LT (1) LT2767285T (es)
MX (1) MX2014004135A (es)
MY (1) MY173370A (es)
PL (1) PL2767285T3 (es)
PT (1) PT2767285T (es)
SG (2) SG2014013783A (es)
SI (1) SI2767285T1 (es)
TW (1) TWI634908B (es)
UA (1) UA114411C2 (es)
WO (1) WO2013054872A1 (es)
ZA (1) ZA201402333B (es)

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TWI320783B (en) 2005-04-14 2010-02-21 Otsuka Pharma Co Ltd Heterocyclic compound
JO3753B1 (ar) * 2011-10-14 2021-01-31 Otsuka Pharma Co Ltd قرص يتألف من 7-[4-(4-بينزو[بي]ثيوفين-4-ايل-ببرازين-1-1ايل)بوتكسيل]-1اتش-كوينولين-2-وان أو ملح منه
JOP20200109A1 (ar) 2012-04-23 2017-06-16 Otsuka Pharma Co Ltd مستحضر قابل للحقن
JP5936732B1 (ja) * 2015-03-05 2016-06-22 日本カラコン合同会社 フィルムコーティング組成物
CN105106142B (zh) * 2015-09-22 2018-05-22 成都欣捷高新技术开发有限公司 一种含有依匹哌唑的冻干口服制剂及其制备方法
CN106994119A (zh) * 2016-01-22 2017-08-01 浙江华海药业股份有限公司 含有依匹哌唑或其盐的口腔崩解片及其制备方法
CA3014090A1 (en) * 2016-02-19 2017-08-24 Jiangsu Hengrui Medicine Co., Ltd. Pharmaceutical composition containing jak kinase inhibitor or pharmaceutically acceptable salt thereof
JP7020688B2 (ja) * 2016-06-28 2022-02-16 株式会社日本抗菌総合研究所 賦形剤及び錠剤
JP7060878B2 (ja) * 2016-07-27 2022-04-27 日本臓器製薬株式会社 メトトレキサート含有フィルムコーティング錠
WO2018033481A1 (en) 2016-08-16 2018-02-22 H E X A L Aktiengesellschaft Immediate release tablet of a benzothiophene compound
WO2018033483A1 (en) 2016-08-16 2018-02-22 H E X A L Aktiengesellschaft Pharmaceutical compositions of a benzothiophene compound
CN106496206A (zh) * 2016-08-31 2017-03-15 安徽省润生医药股份有限公司 一种依匹哌唑新的制备方法
US10919898B2 (en) * 2017-02-23 2021-02-16 Boehringer Ingelheim International Gmbh Medical use of compound III
JP7166754B2 (ja) 2017-11-22 2022-11-08 沢井製薬株式会社 ダサチニブ無水物含有製剤
EP3501506B1 (en) 2017-12-19 2019-10-09 Alfred E. Tiefenbacher (GmbH & Co. KG) Pharmaceutical tablet composition comprising brexpiprazole
EP3545950A1 (en) 2018-03-26 2019-10-02 Adamed sp. z o.o. Pharmaceutical composition comprising brexpiprazole
JPWO2021029020A1 (es) * 2019-08-13 2021-02-18
CN112168794A (zh) * 2020-10-27 2021-01-05 浙江诺得药业有限公司 一种布瑞哌唑片的制备方法
CN115192549A (zh) * 2021-04-13 2022-10-18 上海博志研新药物技术有限公司 一种布瑞哌唑物口腔薄膜剂、其制备方法及应用

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US6562375B1 (en) * 1999-08-04 2003-05-13 Yamanouchi Pharmaceuticals, Co., Ltd. Stable pharmaceutical composition for oral use
AU2002353659A1 (en) * 2001-12-18 2003-07-15 Synthon B.V. Simvastatin dosage forms
AU2003223093B2 (en) * 2002-05-03 2010-02-04 Israel Institute For Biological Research Methods and compositions for treatment of central and peripheral nervous system disorders and novel compounds useful therefor
WO2004096810A1 (en) 2003-04-29 2004-11-11 Pfizer Limited 5,7-diaminopyrazolo`4,3-d!pyrimidines useful in the treatment of hypertension
CA2531694A1 (en) * 2003-06-09 2004-12-09 Dow Global Technologies Inc. Stabilized organoborane polymerization initiators and polymerizable compositions
JP2006061067A (ja) * 2004-08-26 2006-03-09 Asahi Kasei Life & Living Corp 酸素インジケーター
GB0504203D0 (en) * 2005-03-01 2005-04-06 Novartis Ag Organic compounds
ES2526415T3 (es) 2005-03-17 2015-01-12 Synthon B.V. Comprimidos farmacéuticos de aripiprazol cristalino de tipo II
TWI320783B (en) * 2005-04-14 2010-02-21 Otsuka Pharma Co Ltd Heterocyclic compound
JP4315393B2 (ja) * 2005-04-14 2009-08-19 大塚製薬株式会社 複素環化合物
ES2318693T5 (es) 2006-01-05 2018-10-04 Teva Pharmaceutical Industries Ltd Procedimiento de granulación en húmedo para la preparación de composiciones farmacéuticas de aripiprazol
JP4806595B2 (ja) * 2006-07-05 2011-11-02 富士フイルム株式会社 固体撮像素子駆動装置及びデジタルカメラ
JP4540700B2 (ja) * 2006-10-13 2010-09-08 大塚製薬株式会社 医薬
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US7994183B2 (en) * 2007-03-13 2011-08-09 Takeda Pharmaceutical Company Limited Solid preparation comprising 2-[[6-[(3R)-3-amino-1-piperidinyl]-3,4-dihydro-3-methyl-2,4-dioxo-1(2H)-pyrimidinyl]methyl]-4-fluorobenzonitrile
JP2008308489A (ja) * 2007-05-11 2008-12-25 Santen Pharmaceut Co Ltd ロピニロール又はその塩を有効成分として含有する後眼部疾患の予防又は治療剤
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AR085840A1 (es) * 2011-04-05 2013-10-30 Otsuka Pharma Co Ltd Medicamento que contiene un compuesto que es 7-[4-(4-benzo[b]tiofen-4-il-piperazin-1-il)butoxi]-1h-quinolin-2-ona
EP3173096A1 (en) 2011-04-06 2017-05-31 Biovaxim Limited Pharmaceutical compositions for preventing and/or treating an hiv disease in humans
JO3753B1 (ar) * 2011-10-14 2021-01-31 Otsuka Pharma Co Ltd قرص يتألف من 7-[4-(4-بينزو[بي]ثيوفين-4-ايل-ببرازين-1-1ايل)بوتكسيل]-1اتش-كوينولين-2-وان أو ملح منه

Also Published As

Publication number Publication date
US20170165258A1 (en) 2017-06-15
ZA201402333B (en) 2015-07-29
US20180008600A1 (en) 2018-01-11
CA2851588C (en) 2019-07-02
AR088319A1 (es) 2014-05-28
JPWO2013054872A1 (ja) 2015-03-30
IL231513B (en) 2020-01-30
US20220331311A1 (en) 2022-10-20
CA2851588A1 (en) 2013-04-18
PL2767285T3 (pl) 2020-04-30
MX2014004135A (es) 2014-07-24
NZ622639A (en) 2015-11-27
CN103889425B (zh) 2018-08-03
US20210023078A1 (en) 2021-01-28
CY1122460T1 (el) 2021-01-27
JO3753B1 (ar) 2021-01-31
AP2014007564A0 (en) 2014-04-30
US20160158227A1 (en) 2016-06-09
EP2767285B1 (en) 2019-11-27
KR102072371B1 (ko) 2020-02-03
AU2012321723A1 (en) 2014-05-15
WO2013054872A1 (ja) 2013-04-18
SG2014013783A (en) 2014-06-27
EP2767285A1 (en) 2014-08-20
SI2767285T1 (sl) 2020-03-31
LT2767285T (lt) 2020-02-10
PT2767285T (pt) 2020-01-21
JP6084161B2 (ja) 2017-02-22
US10307419B2 (en) 2019-06-04
TWI634908B (zh) 2018-09-11
CN107397730A (zh) 2017-11-28
EA032930B1 (ru) 2019-08-30
SG10201608412SA (en) 2016-12-29
EA201490783A1 (ru) 2014-07-30
TW201318651A (zh) 2013-05-16
IN2014DN02055A (es) 2015-05-15
HUE047493T2 (hu) 2020-04-28
KR20140075754A (ko) 2014-06-19
US20140234417A1 (en) 2014-08-21
JP2017088610A (ja) 2017-05-25
UA114411C2 (uk) 2017-06-12
DK2767285T3 (da) 2020-01-27
CN103889425A (zh) 2014-06-25
HRP20200037T1 (hr) 2020-03-20
MY173370A (en) 2020-01-21
AU2012321723C1 (en) 2017-11-02
CL2014000909A1 (es) 2014-11-21
ES2762479T3 (es) 2020-05-25
BR112014008603A2 (pt) 2017-04-18
US20190240215A1 (en) 2019-08-08
IL231513A0 (en) 2014-04-30
EP2767285A4 (en) 2015-03-11
AU2012321723B2 (en) 2017-07-20

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