CO4650030A1 - Derivados de n-(benzotiazol-2-il) piperidina-1-etanamina, proceso para su preparacion y producto farmaceutico que los contiene - Google Patents

Derivados de n-(benzotiazol-2-il) piperidina-1-etanamina, proceso para su preparacion y producto farmaceutico que los contiene

Info

Publication number
CO4650030A1
CO4650030A1 CO97056315A CO97056315A CO4650030A1 CO 4650030 A1 CO4650030 A1 CO 4650030A1 CO 97056315 A CO97056315 A CO 97056315A CO 97056315 A CO97056315 A CO 97056315A CO 4650030 A1 CO4650030 A1 CO 4650030A1
Authority
CO
Colombia
Prior art keywords
benzotiazol
ethanamine
piperidine
derivatives
preparation
Prior art date
Application number
CO97056315A
Other languages
English (en)
Spanish (es)
Inventor
Dargazanli Gihad
George Pascal
Patrick Lardenois
Jonathan Frost
Schoemaker Jahannes
Maria Carmen Renones
Magat Pascale
Original Assignee
Sanofi Synthelabo
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi Synthelabo filed Critical Sanofi Synthelabo
Publication of CO4650030A1 publication Critical patent/CO4650030A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425Thiazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Neurosurgery (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
CO97056315A 1996-10-01 1997-09-26 Derivados de n-(benzotiazol-2-il) piperidina-1-etanamina, proceso para su preparacion y producto farmaceutico que los contiene CO4650030A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR9611925A FR2753970B1 (fr) 1996-10-01 1996-10-01 Derives de n-(benzothiazol-2-yl) piperidine-1-ethanamine, leur preparation et leur application en therapeutique

Publications (1)

Publication Number Publication Date
CO4650030A1 true CO4650030A1 (es) 1998-09-03

Family

ID=9496217

Family Applications (1)

Application Number Title Priority Date Filing Date
CO97056315A CO4650030A1 (es) 1996-10-01 1997-09-26 Derivados de n-(benzotiazol-2-il) piperidina-1-etanamina, proceso para su preparacion y producto farmaceutico que los contiene

Country Status (23)

Country Link
EP (1) EP0929550A1 (cs)
JP (1) JP2001501217A (cs)
KR (1) KR20000048767A (cs)
CN (1) CN1230959A (cs)
AR (1) AR009105A1 (cs)
AU (1) AU722147B2 (cs)
BG (1) BG103271A (cs)
BR (1) BR9711842A (cs)
CA (1) CA2266510A1 (cs)
CO (1) CO4650030A1 (cs)
CZ (1) CZ112699A3 (cs)
EE (1) EE9900135A (cs)
FR (1) FR2753970B1 (cs)
HU (1) HUP9904091A3 (cs)
IL (1) IL128902A (cs)
NO (1) NO991581L (cs)
NZ (1) NZ334553A (cs)
PL (1) PL332648A1 (cs)
SK (1) SK42299A3 (cs)
TR (1) TR199900634T2 (cs)
TW (1) TW438800B (cs)
WO (1) WO1998014444A1 (cs)
ZA (1) ZA978772B (cs)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9725541D0 (en) * 1997-12-02 1998-02-04 Pharmacia & Upjohn Spa Amino-benzothiazole derivatives
US6107313A (en) * 1998-10-02 2000-08-22 Combichem, Inc. Dopamine receptor antagonists
HRP20020962A2 (en) 2000-06-21 2005-02-28 F. Hoffmann - La Roche Ag Benzothiazole derivatives
US7087761B2 (en) 2003-01-07 2006-08-08 Hoffmann-La Roche Inc. Cyclization process for substituted benzothiazole derivatives
MXPA06004304A (es) * 2003-10-24 2006-06-05 Hoffmann La Roche Antagonistas del receptor ccr-3.
SI1753760T1 (sl) 2004-05-24 2008-04-30 Hoffmann La Roche (4-metoksi-7-morfolin-4-il-benzotiazol-2-il)-amid4- hidroksi-4-metil-piperidin-1-karboksilne kisline
ES2309814T3 (es) 2004-11-05 2008-12-16 F. Hoffmann-La Roche Ag Proceso para la obtencion de derivados del acido isonicotinico.
BRPI0609719B8 (pt) 2005-03-23 2021-05-25 Hoffmann La Roche derivados de acetilenil-pirazol-pirimidina como antagonistas de mgbur2
WO2007039439A1 (en) 2005-09-27 2007-04-12 F.Hoffmann-La Roche Ag Oxadiazolyl pyrazolo-pyrimidines as mglur2 antagonists

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA1260474A (en) * 1984-12-03 1989-09-26 Raymond A. Stokbroekx Benzoxazol- and benzothiazolamine derivatives
KR930005004B1 (ko) * 1985-04-15 1993-06-11 쟈안센 파아마슈우티카 엔. 부이. 치환된 n-[(4-피페리디닐)알킬]이환 축합 옥사졸아민 및 티아졸아민의 제조방법

Also Published As

Publication number Publication date
EP0929550A1 (fr) 1999-07-21
HUP9904091A2 (hu) 2000-05-28
KR20000048767A (ko) 2000-07-25
AU722147B2 (en) 2000-07-20
SK42299A3 (en) 1999-12-10
FR2753970A1 (fr) 1998-04-03
CN1230959A (zh) 1999-10-06
NO991581L (no) 1999-06-01
HUP9904091A3 (en) 2000-07-28
NO991581D0 (no) 1999-03-30
WO1998014444A1 (fr) 1998-04-09
TW438800B (en) 2001-06-07
JP2001501217A (ja) 2001-01-30
FR2753970B1 (fr) 1998-10-30
NZ334553A (en) 2000-11-24
CZ112699A3 (cs) 1999-06-16
AR009105A1 (es) 2000-03-08
IL128902A (en) 2001-07-24
TR199900634T2 (xx) 1999-06-21
PL332648A1 (en) 1999-09-27
EE9900135A (et) 1999-12-15
AU4463897A (en) 1998-04-24
BG103271A (en) 2000-05-31
BR9711842A (pt) 1999-08-24
ZA978772B (en) 1998-03-27
IL128902A0 (en) 2000-02-17
CA2266510A1 (en) 1998-04-09

Similar Documents

Publication Publication Date Title
ES2071510T3 (es) Derivados de pirrolidina y de tiazolidina, su preparacion y los medicamentos que les contienen.
ES2072627T3 (es) Derivados de piridina y n-oxido de piridina de diarilmetilpiperidinas o piperazinas, composiciones y uso de las mismas.
UY24555A1 (es) Nuevos compuestos
ES2160640T3 (es) Nuevos (r)-5-carbamoil-8-fluoro-3-amino disustituido en n,n-3,4-dihidro-2h-1-benzopiranos.
MX9203677A (es) Derivados ciclicos, medicamentos que contienen estos compuestos y procedimiento para su preparacion.
ES2075202T3 (es) Nuevas arilpiridazinas, su preparacion, su utilizacion, y medicamentos que las contienen.
UY25242A1 (es) Inhibidores de benzotiazol de la proteína tirosina cinasa
ES8604548A1 (es) Procedimiento para preparar nuevos derivados de acidos feni-laceticos
ES2179823T3 (es) Inmunosupresor macrolido.
MX9206847A (es) Derivados de indolpirrolcarbazol, proceso para su preparacion y medicamento que los contiene
DK0639179T3 (da) 23-oxaderivater i D-vitaminserien, fremgangsmåde til fremstilling heraf, farmaceutiske præparater indeholdende disse derivater samt deres anvendelse som lægemidler
ES2035824T3 (es) Procedimiento para preparar compuestos profarmacos y preparaciones que los contienen.
AR006360A1 (es) Derivados de 1,2,3,4-tetrahidronaftaleno substituidos, uso de los mismos para la preparacion de medicamentos y procedimiento para su preparacion.
MX9205155A (es) Derivados heterociclicos n-substituidos, procedimiento para su preparacion y composicion farmaceutica que los contiene.
CO4650030A1 (es) Derivados de n-(benzotiazol-2-il) piperidina-1-etanamina, proceso para su preparacion y producto farmaceutico que los contiene
ES2091310T3 (es) Nuevos derivados de la n-benzoil-prolina, su procedimiento de preparacion y composiciones farmaceuticas que los contienen.
MX9303123A (es) Ciclopentano-y-penteno-beta-aminoacidos, procedimiento para su preparacion y medicamentos que los contienen.
MX9204342A (es) Indoles.
ES2135722T3 (es) 1,5-benzodiacepinas 5-heterociclicas moduladoras de la cck o de la gastrina.
ES2153019T3 (es) Derivados de benzo-dioxano, su procedimiento de preparacion y las composiciones farmaceuticas que los contienen.
ES2077998T3 (es) Derivados de 2-aminopirimidina-4-carboxamida, su preparacion y su aplicacion terapeutica.
SE9003973L (sv) Glycerol, ett framstaellningsfoerfarande foer desamma samt terapeutiska kompositioner innehaallande dem
ES2043943T3 (es) Procedimiento para la preparacion de compuestos con actividad analgesica central.
NO884005D0 (no) Fluorerte derivater av aminosyrer saerlig for bruk som oveflateaktive midler.
DE69710909D1 (de) Substituierte tetrahydropyridinderivate, verfahren zu ihrer herstellung und diese enthaltende arzneimittel