AU4463897A - N-(benzothiazol-2-yl) piperidine-1-ethanamine derivatives, their preparation and application in therapeutics - Google Patents

N-(benzothiazol-2-yl) piperidine-1-ethanamine derivatives, their preparation and application in therapeutics

Info

Publication number
AU4463897A
AU4463897A AU44638/97A AU4463897A AU4463897A AU 4463897 A AU4463897 A AU 4463897A AU 44638/97 A AU44638/97 A AU 44638/97A AU 4463897 A AU4463897 A AU 4463897A AU 4463897 A AU4463897 A AU 4463897A
Authority
AU
Australia
Prior art keywords
benzothiazol
therapeutics
piperidine
preparation
application
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
AU44638/97A
Other versions
AU722147B2 (en
Inventor
Gihad Dargazanli
Jonathan Frost
Pascal George
Patrick Lardenois
Pascale Magat
Maria-Carmen Renones
Johannes Schoemaker
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Sanofi Aventis France
Original Assignee
Synthelabo SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Synthelabo SA filed Critical Synthelabo SA
Publication of AU4463897A publication Critical patent/AU4463897A/en
Application granted granted Critical
Publication of AU722147B2 publication Critical patent/AU722147B2/en
Assigned to SANOFI-SYNTHELABO reassignment SANOFI-SYNTHELABO Amend patent request/document other than specification (104) Assignors: SYNTHELABO
Anticipated expiration legal-status Critical
Ceased legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425—Thiazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Neurosurgery (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
AU44638/97A 1996-10-01 1997-09-26 N-(benzothiazol-2-yl) piperidine-1-ethanamine derivatives, their preparation and application in therapeutics Ceased AU722147B2 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
FR9611925A FR2753970B1 (en) 1996-10-01 1996-10-01 N- (BENZOTHIAZOL-2-YL) PIPERIDINE-1-ETHANAMINE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION
FR96/11925 1996-10-01
PCT/FR1997/001692 WO1998014444A1 (en) 1996-10-01 1997-09-26 N-(benzothiazol-2-yl) piperidine-1-ethanamine derivatives, their preparation and application in therapeutics

Publications (2)

Publication Number Publication Date
AU4463897A true AU4463897A (en) 1998-04-24
AU722147B2 AU722147B2 (en) 2000-07-20

Family

ID=9496217

Family Applications (1)

Application Number Title Priority Date Filing Date
AU44638/97A Ceased AU722147B2 (en) 1996-10-01 1997-09-26 N-(benzothiazol-2-yl) piperidine-1-ethanamine derivatives, their preparation and application in therapeutics

Country Status (23)

Country Link
EP (1) EP0929550A1 (en)
JP (1) JP2001501217A (en)
KR (1) KR20000048767A (en)
CN (1) CN1230959A (en)
AR (1) AR009105A1 (en)
AU (1) AU722147B2 (en)
BG (1) BG103271A (en)
BR (1) BR9711842A (en)
CA (1) CA2266510A1 (en)
CO (1) CO4650030A1 (en)
CZ (1) CZ112699A3 (en)
EE (1) EE9900135A (en)
FR (1) FR2753970B1 (en)
HU (1) HUP9904091A3 (en)
IL (1) IL128902A (en)
NO (1) NO991581L (en)
NZ (1) NZ334553A (en)
PL (1) PL332648A1 (en)
SK (1) SK42299A3 (en)
TR (1) TR199900634T2 (en)
TW (1) TW438800B (en)
WO (1) WO1998014444A1 (en)
ZA (1) ZA978772B (en)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9725541D0 (en) * 1997-12-02 1998-02-04 Pharmacia & Upjohn Spa Amino-benzothiazole derivatives
US6107313A (en) * 1998-10-02 2000-08-22 Combichem, Inc. Dopamine receptor antagonists
KR100571161B1 (en) 2000-06-21 2006-04-17 에프. 호프만-라 로슈 아게 Benzothiazole derivatives
US7087761B2 (en) 2003-01-07 2006-08-08 Hoffmann-La Roche Inc. Cyclization process for substituted benzothiazole derivatives
KR20060061393A (en) * 2003-10-24 2006-06-07 에프. 호프만-라 로슈 아게 Ccr3 receptor antagonists
PL1753760T3 (en) 2004-05-24 2008-06-30 Hoffmann La Roche 4-hydroxy-4-methyl-piperidine-1-carboxylic acid (4-methoxy-7-morpholin-4-yl-benzothiazol-2-yl)-amide
CA2586931C (en) 2004-11-05 2013-08-06 Paul Spurr Process for preparation of isonicotinic acid derivatives
BRPI0609719B8 (en) 2005-03-23 2021-05-25 Hoffmann La Roche acetylenyl-pyrazole-pyrimidine derivatives as mgbur2 antagonists
BRPI0616571A2 (en) 2005-09-27 2011-06-21 Hoffmann La Roche oxadiazolyl pyrazol pyridimines as mglur2 antagonists, process for their preparation, pharmaceutical composition containing them and use thereof

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA1260474A (en) * 1984-12-03 1989-09-26 Raymond A. Stokbroekx Benzoxazol- and benzothiazolamine derivatives
KR930005004B1 (en) * 1985-04-15 1993-06-11 쟈안센 파아마슈우티카 엔. 부이. Process for preparing substituted n-|(4-piperidinyl) alkyl¨ bicycle condensed oxazole and thiazolamines

Also Published As

Publication number Publication date
EE9900135A (en) 1999-12-15
FR2753970A1 (en) 1998-04-03
FR2753970B1 (en) 1998-10-30
NZ334553A (en) 2000-11-24
TR199900634T2 (en) 1999-06-21
IL128902A (en) 2001-07-24
IL128902A0 (en) 2000-02-17
CN1230959A (en) 1999-10-06
HUP9904091A2 (en) 2000-05-28
CA2266510A1 (en) 1998-04-09
SK42299A3 (en) 1999-12-10
AU722147B2 (en) 2000-07-20
BG103271A (en) 2000-05-31
AR009105A1 (en) 2000-03-08
HUP9904091A3 (en) 2000-07-28
BR9711842A (en) 1999-08-24
WO1998014444A1 (en) 1998-04-09
PL332648A1 (en) 1999-09-27
KR20000048767A (en) 2000-07-25
JP2001501217A (en) 2001-01-30
CO4650030A1 (en) 1998-09-03
NO991581D0 (en) 1999-03-30
EP0929550A1 (en) 1999-07-21
ZA978772B (en) 1998-03-27
TW438800B (en) 2001-06-07
CZ112699A3 (en) 1999-06-16
NO991581L (en) 1999-06-01

Similar Documents

Publication Publication Date Title
AU3577995A (en) Urea derivatives and their use as acat-inhibitors
AU3660795A (en) Oxazolidinedione derivatives, their production and use
AU2875297A (en) N-(4-aryl-thiazol-2-yl)-sulphonamide derivatives and their use
AU7432994A (en) Imidazol-4-ylpiperidine derivatives, their preparation and their application in therapeutics
AU6124296A (en) Novel dolastatin derivatives, their preparation and use
AU1106195A (en) Heterocyclic compounds, their preparation and use
AU4777097A (en) Novel piperidineketocarboxylic acid derivatives, their preparation and use
AU9633098A (en) Benzoxazine derivatives, preparation and application in therapy
AU2636597A (en) Novel alpha-hydroxy acid derivatives, their preparation and use
CY2291B1 (en) 1H-pyridoa3,4-buindole-4-carboxamide derivatives preparation and application thereof in therapeutics
AU4800896A (en) Piperidine derivatives, process for the preparation thereof and application thereof in therapeutics
ZA978089B (en) 3,4-diaryloxazolone derivatives, their methods of preparation, and their use in therapeutics.
ZA988921B (en) 3,4-diarylthiazolin-2-one or -2-thione derivatives their methods of preparation and their uses in therapeutics
AU5652096A (en) Azacycloalcane derivatives, their preparation and their applications in therapy
AU5591296A (en) N-((1,4-diazabicyclo(2.2.2)oct-2-yl)methyl)benzamide derivatives, their preparation and their application in therapeutics
AU4463897A (en) N-(benzothiazol-2-yl) piperidine-1-ethanamine derivatives, their preparation and application in therapeutics
AU681204B2 (en) N-substituted azabicycloalkane derivatives, their preparation and use
AU4020097A (en) Benzylamine derivatives, their preparation and their application in therapeutics
AU3650695A (en) New heterocyclic substituted imidazoloquinoxalinones, their preparation and their use
AU4450789A (en) Phenyloxypropanolamine derivatives, their preparation and their application in therapeutics
AU5557698A (en) Novel calpaines, their preparation and use
AU1724697A (en) Novel aminophenol derivatives and their use
ZA9710515B (en) N-(imidazolybutyl) benezenesulphonamide derivatives, their preparation and their application in therapeutics.
AU3448097A (en) 1-oxo-1,2-dihydroisoquinoline-4-propanamide derivatives and their application in therapeutics
AU5975094A (en) 1,2,4-triazinone derivatives and their use in therapy

Legal Events

Date Code Title Description
TC Change of applicant's name (sec. 104)

Owner name: SANOFI-SYNTHELABO

Free format text: FORMER NAME: SYNTHELABO

FGA Letters patent sealed or granted (standard patent)
MK14 Patent ceased section 143(a) (annual fees not paid) or expired