TR199900634T2 - N-(Benzothiazol-2-yl) Piperidine-1-ethanamine derivatives, their preparation and application in therapy. - Google Patents
N-(Benzothiazol-2-yl) Piperidine-1-ethanamine derivatives, their preparation and application in therapy.Info
- Publication number
- TR199900634T2 TR199900634T2 TR1999/00634T TR9900634T TR199900634T2 TR 199900634 T2 TR199900634 T2 TR 199900634T2 TR 1999/00634 T TR1999/00634 T TR 1999/00634T TR 9900634 T TR9900634 T TR 9900634T TR 199900634 T2 TR199900634 T2 TR 199900634T2
- Authority
- TR
- Turkey
- Prior art keywords
- therapy
- benzothiazol
- piperidine
- preparation
- application
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Medicinal Chemistry (AREA)
- Neurosurgery (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Hydrogenated Pyridines (AREA)
Abstract
Mevcut bulus, içerisindeki n'nin 0, 1, 2 veya 3 sayisini simgeledigi, R1'in bir hidrojen veya halojen atomunu veya bir metil veya metoksi grubunu, R2'nin bir hidrojen atomu veya bir metil grubunu ve R3'ün bir hidrojen atomu veya bir veya iki halojen atomunu simgeledigi genel formül (I) ile uyumlu olan bilesikleri bildirmektedir. Mevcut bulus, terapide uygulanabilmektedir. (Formül(I)).The present invention represents a hydrogen or halogen atom or a methyl or methoxy group of R2, a hydrogen atom or a methyl group of R2, and a hydrogen atom of R3 or n, in which n represents 0, 1, 2 or 3 It reports compounds that comply with the general formula (I), in which it symbolizes one or two halogen atoms. The present invention can be applied in therapy. (Formula (I)).
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR9611925A FR2753970B1 (en) | 1996-10-01 | 1996-10-01 | N- (BENZOTHIAZOL-2-YL) PIPERIDINE-1-ETHANAMINE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| TR199900634T2 true TR199900634T2 (en) | 1999-06-21 |
Family
ID=9496217
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| TR1999/00634T TR199900634T2 (en) | 1996-10-01 | 1997-09-26 | N-(Benzothiazol-2-yl) Piperidine-1-ethanamine derivatives, their preparation and application in therapy. |
Country Status (23)
| Country | Link |
|---|---|
| EP (1) | EP0929550A1 (en) |
| JP (1) | JP2001501217A (en) |
| KR (1) | KR20000048767A (en) |
| CN (1) | CN1230959A (en) |
| AR (1) | AR009105A1 (en) |
| AU (1) | AU722147B2 (en) |
| BG (1) | BG103271A (en) |
| BR (1) | BR9711842A (en) |
| CA (1) | CA2266510A1 (en) |
| CO (1) | CO4650030A1 (en) |
| CZ (1) | CZ112699A3 (en) |
| EE (1) | EE9900135A (en) |
| FR (1) | FR2753970B1 (en) |
| HU (1) | HUP9904091A3 (en) |
| IL (1) | IL128902A (en) |
| NO (1) | NO991581L (en) |
| NZ (1) | NZ334553A (en) |
| PL (1) | PL332648A1 (en) |
| SK (1) | SK42299A3 (en) |
| TR (1) | TR199900634T2 (en) |
| TW (1) | TW438800B (en) |
| WO (1) | WO1998014444A1 (en) |
| ZA (1) | ZA978772B (en) |
Families Citing this family (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB9725541D0 (en) * | 1997-12-02 | 1998-02-04 | Pharmacia & Upjohn Spa | Amino-benzothiazole derivatives |
| US6107313A (en) * | 1998-10-02 | 2000-08-22 | Combichem, Inc. | Dopamine receptor antagonists |
| KR100571161B1 (en) | 2000-06-21 | 2006-04-17 | 에프. 호프만-라 로슈 아게 | Benzothiazole derivatives |
| US7087761B2 (en) | 2003-01-07 | 2006-08-08 | Hoffmann-La Roche Inc. | Cyclization process for substituted benzothiazole derivatives |
| KR20060061393A (en) * | 2003-10-24 | 2006-06-07 | 에프. 호프만-라 로슈 아게 | Ccr3 receptor antagonists |
| PL1753760T3 (en) | 2004-05-24 | 2008-06-30 | Hoffmann La Roche | 4-hydroxy-4-methyl-piperidine-1-carboxylic acid (4-methoxy-7-morpholin-4-yl-benzothiazol-2-yl)-amide |
| CA2586931C (en) | 2004-11-05 | 2013-08-06 | Paul Spurr | Process for preparation of isonicotinic acid derivatives |
| BRPI0609719B8 (en) | 2005-03-23 | 2021-05-25 | Hoffmann La Roche | acetylenyl-pyrazole-pyrimidine derivatives as mgbur2 antagonists |
| BRPI0616571A2 (en) | 2005-09-27 | 2011-06-21 | Hoffmann La Roche | oxadiazolyl pyrazol pyridimines as mglur2 antagonists, process for their preparation, pharmaceutical composition containing them and use thereof |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA1260474A (en) * | 1984-12-03 | 1989-09-26 | Raymond A. Stokbroekx | Benzoxazol- and benzothiazolamine derivatives |
| KR930005004B1 (en) * | 1985-04-15 | 1993-06-11 | 쟈안센 파아마슈우티카 엔. 부이. | Process for preparing substituted n-|(4-piperidinyl) alkyl¨ bicycle condensed oxazole and thiazolamines |
-
1996
- 1996-10-01 FR FR9611925A patent/FR2753970B1/en not_active Expired - Fee Related
-
1997
- 1997-09-26 KR KR1019990702753A patent/KR20000048767A/en not_active Application Discontinuation
- 1997-09-26 EE EEP199900135A patent/EE9900135A/en unknown
- 1997-09-26 TR TR1999/00634T patent/TR199900634T2/en unknown
- 1997-09-26 CA CA002266510A patent/CA2266510A1/en not_active Abandoned
- 1997-09-26 AU AU44638/97A patent/AU722147B2/en not_active Ceased
- 1997-09-26 JP JP10516272A patent/JP2001501217A/en active Pending
- 1997-09-26 HU HU9904091A patent/HUP9904091A3/en unknown
- 1997-09-26 IL IL12890297A patent/IL128902A/en not_active IP Right Cessation
- 1997-09-26 BR BR9711842A patent/BR9711842A/en not_active Application Discontinuation
- 1997-09-26 PL PL97332648A patent/PL332648A1/en unknown
- 1997-09-26 CN CN97198112A patent/CN1230959A/en active Pending
- 1997-09-26 CO CO97056315A patent/CO4650030A1/en unknown
- 1997-09-26 CZ CZ991126A patent/CZ112699A3/en unknown
- 1997-09-26 EP EP97943001A patent/EP0929550A1/en not_active Ceased
- 1997-09-26 SK SK422-99A patent/SK42299A3/en unknown
- 1997-09-26 WO PCT/FR1997/001692 patent/WO1998014444A1/en not_active Application Discontinuation
- 1997-09-26 NZ NZ334553A patent/NZ334553A/en unknown
- 1997-09-30 AR ARP970104493A patent/AR009105A1/en not_active Application Discontinuation
- 1997-09-30 TW TW086114229A patent/TW438800B/en active
- 1997-09-30 ZA ZA9708772A patent/ZA978772B/en unknown
-
1999
- 1999-03-22 BG BG103271A patent/BG103271A/en unknown
- 1999-03-30 NO NO991581A patent/NO991581L/en not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| EE9900135A (en) | 1999-12-15 |
| FR2753970A1 (en) | 1998-04-03 |
| AU4463897A (en) | 1998-04-24 |
| FR2753970B1 (en) | 1998-10-30 |
| NZ334553A (en) | 2000-11-24 |
| IL128902A (en) | 2001-07-24 |
| IL128902A0 (en) | 2000-02-17 |
| CN1230959A (en) | 1999-10-06 |
| HUP9904091A2 (en) | 2000-05-28 |
| CA2266510A1 (en) | 1998-04-09 |
| SK42299A3 (en) | 1999-12-10 |
| AU722147B2 (en) | 2000-07-20 |
| BG103271A (en) | 2000-05-31 |
| AR009105A1 (en) | 2000-03-08 |
| HUP9904091A3 (en) | 2000-07-28 |
| BR9711842A (en) | 1999-08-24 |
| WO1998014444A1 (en) | 1998-04-09 |
| PL332648A1 (en) | 1999-09-27 |
| KR20000048767A (en) | 2000-07-25 |
| JP2001501217A (en) | 2001-01-30 |
| CO4650030A1 (en) | 1998-09-03 |
| NO991581D0 (en) | 1999-03-30 |
| EP0929550A1 (en) | 1999-07-21 |
| ZA978772B (en) | 1998-03-27 |
| TW438800B (en) | 2001-06-07 |
| CZ112699A3 (en) | 1999-06-16 |
| NO991581L (en) | 1999-06-01 |
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