CN1898255B - 制备吡啶衍生物的方法 - Google Patents

制备吡啶衍生物的方法 Download PDF

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Publication number
CN1898255B
CN1898255B CN2004800388844A CN200480038884A CN1898255B CN 1898255 B CN1898255 B CN 1898255B CN 2004800388844 A CN2004800388844 A CN 2004800388844A CN 200480038884 A CN200480038884 A CN 200480038884A CN 1898255 B CN1898255 B CN 1898255B
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CN
China
Prior art keywords
reaction
mixture
pyridine
general formula
trifluoromethyl
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Expired - Lifetime
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CN2004800388844A
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English (en)
Chinese (zh)
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CN1898255A (zh
Inventor
J·格巴尔
N·格茨
H·耶迪克
G·马耶尔
M·拉克
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Kedihua Agricultural Technology Co ltd
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Dow AgroSciences LLC
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C323/00—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
    • C07C323/50—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton
    • C07C323/51—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton
    • C07C323/60—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton with the carbon atom of at least one of the carboxyl groups bound to nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/62—Oxygen or sulfur atoms
    • C07D213/63—One oxygen atom
    • C07D213/64—One oxygen atom attached in position 2 or 6
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/62—Oxygen or sulfur atoms
    • C07D213/70—Sulfur atoms
    • C07D213/71—Sulfur atoms to which a second hetero atom is attached
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/28—Phosphorus compounds with one or more P—C bonds
    • C07F9/38—Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)]
    • C07F9/40—Esters thereof
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/28—Phosphorus compounds with one or more P—C bonds
    • C07F9/38—Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)]
    • C07F9/40—Esters thereof
    • C07F9/4003—Esters thereof the acid moiety containing a substituent or a structure which is considered as characteristic
    • C07F9/4006—Esters of acyclic acids which can have further substituents on alkyl

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biochemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Molecular Biology (AREA)
  • Pyridine Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Indole Compounds (AREA)
CN2004800388844A 2003-12-23 2004-12-22 制备吡啶衍生物的方法 Expired - Lifetime CN1898255B (zh)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US53161403P 2003-12-23 2003-12-23
EP03029730 2003-12-23
US60/531,614 2003-12-23
EP03029730.3 2003-12-23
PCT/EP2004/014590 WO2005063780A1 (en) 2003-12-23 2004-12-22 Process for the preparation of pyridine derivatives

Publications (2)

Publication Number Publication Date
CN1898255A CN1898255A (zh) 2007-01-17
CN1898255B true CN1898255B (zh) 2010-06-09

Family

ID=34923925

Family Applications (1)

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CN2004800388844A Expired - Lifetime CN1898255B (zh) 2003-12-23 2004-12-22 制备吡啶衍生物的方法

Country Status (16)

Country Link
US (1) US7687632B2 (OSRAM)
EP (1) EP1723156B1 (OSRAM)
JP (3) JP5160092B2 (OSRAM)
KR (1) KR101164694B1 (OSRAM)
CN (1) CN1898255B (OSRAM)
AR (1) AR046775A1 (OSRAM)
AU (1) AU2004309054B2 (OSRAM)
BR (1) BRPI0418047B8 (OSRAM)
CA (1) CA2550693C (OSRAM)
DK (1) DK1723156T3 (OSRAM)
ES (1) ES2528716T3 (OSRAM)
IL (1) IL176472A (OSRAM)
IN (2) IN2012DN02545A (OSRAM)
PL (1) PL1723156T3 (OSRAM)
WO (1) WO2005063780A1 (OSRAM)
ZA (1) ZA200605471B (OSRAM)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2006060029A2 (en) * 2004-04-08 2006-06-08 Dow Agrosciences Llc Insecticidal n-substituted sulfoximines
WO2006012320A1 (en) * 2004-06-25 2006-02-02 Dow Agrosciences Llc Process for the preparation of 4-trifluoromethyl-2(1h)-pyridinone
TWI398433B (zh) * 2006-02-10 2013-06-11 Dow Agrosciences Llc 殺蟲性之ｎ-取代（６-鹵烷基吡啶-３-基）烷基磺醯亞胺
TWI381811B (zh) * 2006-06-23 2013-01-11 Dow Agrosciences Llc 用以防治可抵抗一般殺蟲劑之昆蟲的方法
TWI387585B (zh) * 2006-09-01 2013-03-01 Dow Agrosciences Llc 殺蟲性之ｎ-取代（雜芳基）烷基烴基硫亞胺
EP2338884A1 (en) * 2006-09-01 2011-06-29 Dow AgroSciences LLC Insecticidal N-substituted (2-substituted-1,3-thiazol) alkyl sulfoximines
TWI395736B (zh) * 2006-11-08 2013-05-11 Dow Agrosciences Llc 作為殺蟲劑之雜芳基（取代的）烷基ｎ-取代的磺醯亞胺（二）
US7709648B2 (en) * 2007-02-09 2010-05-04 Dow Agrosciences Llc Process for the preparation of 2-substituted-5-(1-alkylthio)alkylpyridines
AR066366A1 (es) * 2007-05-01 2009-08-12 Dow Agrosciences Llc Mezclas sinergicas plaguicidas
KR101512528B1 (ko) * 2007-07-20 2015-04-15 다우 아그로사이언시즈 엘엘씨 식물 생장력의 증가
CA2717069C (en) * 2008-03-03 2013-08-20 Dow Agrosciences Llc Pesticides
CN102875548A (zh) * 2011-07-14 2013-01-16 中国科学院大连化学物理研究所 一类基于肟的通过[2+2+2]环加成合成吡啶衍生物的方法
EP2607343A1 (en) 2011-12-22 2013-06-26 Solvay Sa Process for the manufacture of halogenated precursors of alkenones and of alkenones
JP7282031B2 (ja) * 2016-12-01 2023-05-26 シンジェンタ パーティシペーションズ アーゲー 硫黄含有置換基を有する殺有害生物的に活性な複素環式誘導体
EP3902785A1 (en) * 2018-12-27 2021-11-03 Corteva Agriscience LLC Preparation of sulfonamide herbicide process intermediates
EP3902786B1 (en) 2018-12-27 2022-12-14 Corteva Agriscience LLC Preparation of sulfonamide herbicide process intermediates
CN115286568B (zh) * 2022-08-24 2023-12-12 常州沃腾化工科技有限公司 一种2-羟基-4-三氟甲基吡啶的制备方法

Citations (1)

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US3993656A (en) * 1974-11-19 1976-11-23 Merck & Co., Inc. 1,8-Naphthyridine compounds

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JPS5221196A (en) * 1975-08-12 1977-02-17 Fujio Hashimoto Device for removing red tide
JPS53121764A (en) * 1977-03-31 1978-10-24 Yamanouchi Pharmaceut Co Ltd Heterocyclic compounds and process for their preparation
JPS5384990A (en) * 1976-12-29 1978-07-26 Yamanouchi Pharmaceut Co Ltd Novel nitrogen-containing heterocyclic compound and its preparation
JPS53127490A (en) * 1977-04-13 1978-11-07 Yamanouchi Pharmaceut Co Ltd Novel nitrogen-containing heterocyclic compound
JPS55104266A (en) * 1979-02-02 1980-08-09 Yamanouchi Pharmaceut Co Ltd Novel pyridone derivative
JPS6210087A (ja) * 1985-07-03 1987-01-19 Shionogi & Co Ltd ４，７−ジヒドロチエノ〔２，３−ｂ〕ピリジン誘導体，その製造法および循環器系疾患治療剤
JPS6413065A (en) * 1987-07-06 1989-01-17 Mitsubishi Chem Ind Peptide derivative of beta-chloro-l-(z)- dehydroglutamic acid
DK177191D0 (da) * 1991-10-23 1991-10-23 Novo Nordisk As Heterocyclic compounds and their preparation and use
US5391745A (en) * 1992-07-23 1995-02-21 Sloan-Kettering Institute For Cancer Research Methods of preparation of camptothecin analogs
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KR100581199B1 (ko) * 1998-06-19 2006-05-17 카이론 코포레이션 글리코겐 신타제 키나제 3의 억제제
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KNOEVENAGEL,W.CREMER.SYNTHESEN IN DER PYRIDINREIHE. UEBERDIEEINWIRKUNG VON MALONESTER UNDMALONAMIDAUF AMINOACETYLACETON.CHEM.BERICHTE.1902,2390-2396. *
REUBEN G.J. ET AL..PREPARATION AND REACTIONS OFSOMEPENTA-SUBSTITUTED PYRIDINES.JOURNAL OF THE AMERICAN CHEMICAL SOCIETY73 12.1951,73(12),5610-5614. *
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Also Published As

Publication number Publication date
CN1898255A (zh) 2007-01-17
US7687632B2 (en) 2010-03-30
US20070249837A1 (en) 2007-10-25
BRPI0418047A (pt) 2007-04-17
ZA200605471B (en) 2007-11-28
EP1723156A1 (en) 2006-11-22
CA2550693C (en) 2013-07-30
JP2013047245A (ja) 2013-03-07
CA2550693A1 (en) 2005-07-14
JP2007519625A (ja) 2007-07-19
BRPI0418047B8 (pt) 2022-06-28
ES2528716T3 (es) 2015-02-12
AU2004309054A1 (en) 2005-07-14
DK1723156T3 (en) 2015-04-27
AR046775A1 (es) 2005-12-21
JP2012214487A (ja) 2012-11-08
EP1723156B1 (en) 2015-01-21
AU2004309054B2 (en) 2010-07-08
JP5160092B2 (ja) 2013-03-13
IL176472A0 (en) 2006-10-05
KR101164694B1 (ko) 2012-07-11
BRPI0418047B1 (pt) 2013-12-31
KR20060128896A (ko) 2006-12-14
WO2005063780A1 (en) 2005-07-14
IN2012DN02545A (OSRAM) 2015-07-17
PL1723156T3 (pl) 2015-07-31
IN2012DN02546A (OSRAM) 2015-08-28
IL176472A (en) 2010-11-30

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