CN116585316A - 包含pde9抑制剂的药物组合物 - Google Patents
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| PCT/JP2018/020643 WO2018221546A1 (en) | 2017-06-01 | 2018-05-30 | Pharmaceutical composition comprising pde9 inhibitor |
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| CN119302958A (zh) * | 2023-12-01 | 2025-01-14 | 郑州大学第一附属医院 | 含有bay 73-6691或其衍生物的药物制剂在制备治疗脑损伤疾病药物中的应用 |
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| RU2019135834A (ru) | 2017-06-01 | 2021-07-13 | Эйсай Ар Энд Ди Менеджмент Ко., Лтд. | Терапевтическое средство для лечения деменции, представляющее собой комбинацию производного пиразолохинолина и донепезила |
| BR112019023552A2 (pt) | 2017-06-01 | 2020-06-02 | Eisai R&D Management Co., Ltd. | Agente terapêutico para a demência com corpos de lewy contendo derivado de pirazoloquinolina |
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| CN120897742A (zh) * | 2022-11-15 | 2025-11-04 | 福睿德姆生物科学公司 | 通过抑制9型磷酸二酯酶增强血清素能致幻药物在治疗或预防某些神经精神障碍中的功效 |
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| DE19642591A1 (de) | 1996-10-15 | 1998-04-16 | Basf Ag | Neue Piperidin-Ketocarbonsäure-Derivate, deren Herstellung und Anwendung |
| HN2002000317A (es) | 2001-11-02 | 2003-05-21 | Pfizer | Inhibidores de pde9 para tratamiento de trastornos cardiovasculares |
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| DE102004004142A1 (de) | 2003-05-09 | 2004-11-25 | Bayer Healthcare Ag | 6-Cyclylmethyl- und 6-Alkylmethyl-substituierte Pyrazolopyrimidine |
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| WO2013051639A1 (ja) | 2011-10-07 | 2013-04-11 | エーザイ・アール・アンド・ディー・マネジメント株式会社 | ピラゾロキノリン誘導体 |
| CN107847499A (zh) | 2015-05-07 | 2018-03-27 | 阿速万科学有限责任公司 | 治疗神经退行性疾病的方法 |
| BR112019023552A2 (pt) | 2017-06-01 | 2020-06-02 | Eisai R&D Management Co., Ltd. | Agente terapêutico para a demência com corpos de lewy contendo derivado de pirazoloquinolina |
| RU2019135834A (ru) | 2017-06-01 | 2021-07-13 | Эйсай Ар Энд Ди Менеджмент Ко., Лтд. | Терапевтическое средство для лечения деменции, представляющее собой комбинацию производного пиразолохинолина и донепезила |
| WO2018221550A1 (ja) | 2017-06-01 | 2018-12-06 | エーザイ・アール・アンド・ディー・マネジメント株式会社 | ピラゾロキノリン誘導体とメマンチンの併用による認知症治療剤 |
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2018
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- 2018-05-30 CN CN202310559688.6A patent/CN116585316A/zh active Pending
- 2018-05-30 US US16/609,514 patent/US11484502B2/en active Active
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- 2018-05-30 JP JP2019559117A patent/JP7293129B2/ja active Active
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- 2018-05-30 MX MX2019013198A patent/MX2019013198A/es unknown
- 2018-05-30 AU AU2018276566A patent/AU2018276566A1/en not_active Abandoned
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2022
- 2022-06-03 US US17/831,863 patent/US20220378706A1/en not_active Abandoned
Patent Citations (1)
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|---|---|---|---|---|
| US20160046623A1 (en) * | 2013-04-05 | 2016-02-18 | Eisai R&D Management Co., Ltd. | Salt of pyrazoloquinoline derivative, and crystal thereof |
Cited By (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN119302958A (zh) * | 2023-12-01 | 2025-01-14 | 郑州大学第一附属医院 | 含有bay 73-6691或其衍生物的药物制剂在制备治疗脑损伤疾病药物中的应用 |
| CN119302958B (zh) * | 2023-12-01 | 2025-10-21 | 郑州大学第一附属医院 | 含有bay 73-6691或其衍生物的药物制剂在制备治疗脑损伤疾病药物中的应用 |
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| WO2018221546A1 (en) | 2018-12-06 |
| SG11201909359YA (en) | 2019-11-28 |
| KR20200010211A (ko) | 2020-01-30 |
| RU2019135261A (ru) | 2021-07-09 |
| CA3059539A1 (en) | 2018-12-06 |
| JP7293129B2 (ja) | 2023-06-19 |
| EP3630113A4 (en) | 2021-02-24 |
| JP2020521726A (ja) | 2020-07-27 |
| RU2019135261A3 (https=) | 2021-09-08 |
| CN110545812A (zh) | 2019-12-06 |
| US11484502B2 (en) | 2022-11-01 |
| AU2018276566A1 (en) | 2019-11-07 |
| BR112019023557A2 (pt) | 2020-06-02 |
| US20220378706A1 (en) | 2022-12-01 |
| MX2019013198A (es) | 2020-01-20 |
| US20200078306A1 (en) | 2020-03-12 |
| EP3630113A1 (en) | 2020-04-08 |
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