CN1157392C - 在尼古丁ach受体上作为胆碱能配体的8-氮杂双环(3,2,1)辛-2-烯以及辛烷衍生物 - Google Patents

在尼古丁ach受体上作为胆碱能配体的8-氮杂双环(3,2,1)辛-2-烯以及辛烷衍生物 Download PDF

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CN1157392C
CN1157392C CNB988054132A CN98805413A CN1157392C CN 1157392 C CN1157392 C CN 1157392C CN B988054132 A CNB988054132 A CN B988054132A CN 98805413 A CN98805413 A CN 98805413A CN 1157392 C CN1157392 C CN 1157392C
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azabicyclo
oct
ene
methyl
thienyl
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CN1257499A (zh
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D
D·彼得斯
�¶�ɭ
G·M·奥尔森
�������ɭ
S·F·尼尔森
E·O·尼尔森
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NTG Nordic Transport Group AS
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Neurosearch AS
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D451/00—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
    • C07D451/02—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
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    • A61P1/12—Antidiarrhoeals
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    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
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  • Chemical Kinetics & Catalysis (AREA)
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  • General Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Animal Behavior & Ethology (AREA)
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  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
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  • Addiction (AREA)
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  • Endocrinology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Psychology (AREA)
  • Pulmonology (AREA)
  • Diabetes (AREA)
  • Child & Adolescent Psychology (AREA)
  • Obesity (AREA)
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  • Hospice & Palliative Care (AREA)
  • Anesthesiology (AREA)
  • Vascular Medicine (AREA)
  • Hematology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Urology & Nephrology (AREA)
  • Nutrition Science (AREA)
  • Cardiology (AREA)
  • Dermatology (AREA)
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CNB988054132A 1997-05-30 1998-05-29 在尼古丁ach受体上作为胆碱能配体的8-氮杂双环(3,2,1)辛-2-烯以及辛烷衍生物 Expired - Fee Related CN1157392C (zh)

Applications Claiming Priority (8)

Application Number Priority Date Filing Date Title
DK62797 1997-05-30
DK0627/1997 1997-05-30
DK1502/1997 1997-12-19
DK150297 1997-12-19
DK0408/1998 1998-03-24
DK40898 1998-03-24
DK0534/1998 1998-04-16
DK53498 1998-04-16

Publications (2)

Publication Number Publication Date
CN1257499A CN1257499A (zh) 2000-06-21
CN1157392C true CN1157392C (zh) 2004-07-14

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CNB988054132A Expired - Fee Related CN1157392C (zh) 1997-05-30 1998-05-29 在尼古丁ach受体上作为胆碱能配体的8-氮杂双环(3,2,1)辛-2-烯以及辛烷衍生物

Country Status (22)

Country Link
US (2) US6645977B1 (https=)
EP (1) EP0984965B1 (https=)
JP (1) JP4447663B2 (https=)
KR (1) KR100589872B1 (https=)
CN (1) CN1157392C (https=)
AT (1) ATE267199T1 (https=)
AU (1) AU745964B2 (https=)
BR (1) BR9809697A (https=)
CA (1) CA2289574C (https=)
CZ (1) CZ298824B6 (https=)
DE (1) DE69823994T2 (https=)
DK (1) DK0984965T3 (https=)
EE (1) EE04057B1 (https=)
HU (1) HUP0002713A3 (https=)
IL (2) IL132437A0 (https=)
IS (1) IS2092B (https=)
NO (1) NO325513B1 (https=)
NZ (1) NZ500642A (https=)
RU (1) RU2186780C2 (https=)
SK (1) SK284994B6 (https=)
TR (1) TR199902942T2 (https=)
WO (1) WO1998054181A1 (https=)

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US20040019207A1 (en) 2004-01-29
CA2289574A1 (en) 1998-12-03
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