CN109096119A - 一种制备盐酸西那卡塞的方法 - Google Patents
一种制备盐酸西那卡塞的方法 Download PDFInfo
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- CN109096119A CN109096119A CN201811265663.0A CN201811265663A CN109096119A CN 109096119 A CN109096119 A CN 109096119A CN 201811265663 A CN201811265663 A CN 201811265663A CN 109096119 A CN109096119 A CN 109096119A
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C209/00—Preparation of compounds containing amino groups bound to a carbon skeleton
- C07C209/04—Preparation of compounds containing amino groups bound to a carbon skeleton by substitution of functional groups by amino groups
- C07C209/14—Preparation of compounds containing amino groups bound to a carbon skeleton by substitution of functional groups by amino groups by substitution of hydroxy groups or of etherified or esterified hydroxy groups
- C07C209/16—Preparation of compounds containing amino groups bound to a carbon skeleton by substitution of functional groups by amino groups by substitution of hydroxy groups or of etherified or esterified hydroxy groups with formation of amino groups bound to acyclic carbon atoms or to carbon atoms of rings other than six-membered aromatic rings
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C209/00—Preparation of compounds containing amino groups bound to a carbon skeleton
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C303/00—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides
- C07C303/26—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides of esters of sulfonic acids
- C07C303/28—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides of esters of sulfonic acids by reaction of hydroxy compounds with sulfonic acids or derivatives thereof
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- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
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Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
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CN201811265663.0A CN109096119B (zh) | 2018-10-29 | 2018-10-29 | 一种制备盐酸西那卡塞的方法 |
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CN201811265663.0A CN109096119B (zh) | 2018-10-29 | 2018-10-29 | 一种制备盐酸西那卡塞的方法 |
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CN109096119A true CN109096119A (zh) | 2018-12-28 |
CN109096119B CN109096119B (zh) | 2019-10-25 |
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CN201811265663.0A Active CN109096119B (zh) | 2018-10-29 | 2018-10-29 | 一种制备盐酸西那卡塞的方法 |
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Cited By (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN110903212A (zh) * | 2019-12-25 | 2020-03-24 | 江苏正大清江制药有限公司 | 一种合成西那卡塞中间体的方法 |
CN113620855A (zh) * | 2021-08-27 | 2021-11-09 | 山东威高药业股份有限公司 | 一种伊万卡塞中间体ii及其合成方法 |
Citations (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2006127932A2 (en) * | 2005-05-23 | 2006-11-30 | Teva Pharmaceutical Industries Ltd. | Purification of cinacalcet |
CN104774134A (zh) * | 2014-01-09 | 2015-07-15 | 成都自豪药业有限公司 | 盐酸西那卡塞及其中间体化合物的合成方法 |
CN107473993A (zh) * | 2017-08-30 | 2017-12-15 | 山东新华制药股份有限公司 | 高纯度间三氟甲基苯丙醇甲磺酸酯的制备方法 |
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2018
- 2018-10-29 CN CN201811265663.0A patent/CN109096119B/zh active Active
Patent Citations (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2006127932A2 (en) * | 2005-05-23 | 2006-11-30 | Teva Pharmaceutical Industries Ltd. | Purification of cinacalcet |
CN104774134A (zh) * | 2014-01-09 | 2015-07-15 | 成都自豪药业有限公司 | 盐酸西那卡塞及其中间体化合物的合成方法 |
CN107473993A (zh) * | 2017-08-30 | 2017-12-15 | 山东新华制药股份有限公司 | 高纯度间三氟甲基苯丙醇甲磺酸酯的制备方法 |
Cited By (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN110903212A (zh) * | 2019-12-25 | 2020-03-24 | 江苏正大清江制药有限公司 | 一种合成西那卡塞中间体的方法 |
CN113620855A (zh) * | 2021-08-27 | 2021-11-09 | 山东威高药业股份有限公司 | 一种伊万卡塞中间体ii及其合成方法 |
CN113620855B (zh) * | 2021-08-27 | 2023-12-01 | 山东威高药业股份有限公司 | 一种伊万卡塞中间体ii及其合成方法 |
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Publication number | Publication date |
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CN109096119B (zh) | 2019-10-25 |
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Inventor after: Luo Huan Inventor after: Kang Yanlong Inventor after: Li Qian Inventor after: Qiu Chunfang Inventor after: Liu Kelei Inventor after: Wang Shuaiwei Inventor before: Luo Huan Inventor before: Kang Yanlong Inventor before: Li Qian Inventor before: Qiu Chunfang Inventor before: Liu Kelei Inventor before: Wang Shuaiwei |
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