CN108779106B - 用于制备哒嗪酮除草剂的中间体和用于制备它们的方法 - Google Patents

用于制备哒嗪酮除草剂的中间体和用于制备它们的方法 Download PDF

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Publication number
CN108779106B
CN108779106B CN201680076619.8A CN201680076619A CN108779106B CN 108779106 B CN108779106 B CN 108779106B CN 201680076619 A CN201680076619 A CN 201680076619A CN 108779106 B CN108779106 B CN 108779106B
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China
Prior art keywords
radical
alkyl
group
cycloalkyl
haloalkyl
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Expired - Fee Related
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CN201680076619.8A
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English (en)
Chinese (zh)
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CN108779106A (zh
Inventor
T·P·塞尔比
K·M·帕特尔
T·M·史蒂文森
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FMC Corp
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FMC Corp
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/04—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/56—1,2-Diazoles; Hydrogenated 1,2-diazoles
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/58—1,2-Diazines; Hydrogenated 1,2-diazines
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/06—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom containing only hydrogen and carbon atoms in addition to the ring nitrogen atom
    • C07D213/16—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom containing only hydrogen and carbon atoms in addition to the ring nitrogen atom containing only one pyridine ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/62—Oxygen or sulfur atoms
    • C07D213/70—Sulfur atoms
    • C07D213/71—Sulfur atoms to which a second hetero atom is attached
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D237/00—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings
    • C07D237/02—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings
    • C07D237/06—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
    • C07D237/10—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D237/14—Oxygen atoms
    • C07D237/16—Two oxygen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Dentistry (AREA)
  • Wood Science & Technology (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Agronomy & Crop Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyridine Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
CN201680076619.8A 2015-10-28 2016-10-26 用于制备哒嗪酮除草剂的中间体和用于制备它们的方法 Expired - Fee Related CN108779106B (zh)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201562247438P 2015-10-28 2015-10-28
US62/247,438 2015-10-28
PCT/US2016/058755 WO2017074988A1 (en) 2015-10-28 2016-10-26 Intermediates to prepare pyridazinone herbicides, and a process to prepare them

Publications (2)

Publication Number Publication Date
CN108779106A CN108779106A (zh) 2018-11-09
CN108779106B true CN108779106B (zh) 2021-12-07

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CN201680076619.8A Expired - Fee Related CN108779106B (zh) 2015-10-28 2016-10-26 用于制备哒嗪酮除草剂的中间体和用于制备它们的方法

Country Status (17)

Country Link
US (1) US10913719B2 (cg-RX-API-DMAC10.html)
EP (1) EP3368531B1 (cg-RX-API-DMAC10.html)
JP (1) JP6782774B2 (cg-RX-API-DMAC10.html)
KR (1) KR20180075574A (cg-RX-API-DMAC10.html)
CN (1) CN108779106B (cg-RX-API-DMAC10.html)
AR (1) AR106522A1 (cg-RX-API-DMAC10.html)
AU (1) AU2016346207B2 (cg-RX-API-DMAC10.html)
BR (1) BR112018008616B1 (cg-RX-API-DMAC10.html)
CA (1) CA3003410A1 (cg-RX-API-DMAC10.html)
HU (1) HUE049157T2 (cg-RX-API-DMAC10.html)
IL (1) IL258765B (cg-RX-API-DMAC10.html)
MX (1) MX388612B (cg-RX-API-DMAC10.html)
RU (1) RU2743561C2 (cg-RX-API-DMAC10.html)
SG (1) SG11201803134VA (cg-RX-API-DMAC10.html)
TW (1) TWI739769B (cg-RX-API-DMAC10.html)
WO (1) WO2017074988A1 (cg-RX-API-DMAC10.html)
ZA (1) ZA201803362B (cg-RX-API-DMAC10.html)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PE20211761A1 (es) 2014-04-29 2021-09-07 Fmc Corp Herbicidas de piridazinona
AU2016346303B2 (en) 2015-10-28 2021-01-07 Fmc Corporation Novel pyrdazinone herbicides
EP3368531B1 (en) 2015-10-28 2020-01-15 FMC Corporation Intermediates to prepare pyridazinone herbicides, and a process to prepare them
TWI785022B (zh) 2017-03-28 2022-12-01 美商富曼西公司 新穎噠嗪酮類除草劑
BR112019028016B1 (pt) * 2017-06-30 2023-12-05 Fmc Corporation Composto, composições herbicidas, mistura herbicida e método para controlar o crescimento de vegetação indesejada
CA3113061A1 (en) 2018-09-27 2020-04-02 Fmc Corporation Intermediates for preparing herbicidal pyridazinones
MX2021003530A (es) 2018-09-27 2021-05-27 Fmc Corp Herbicidas de piridazinona e intermediarios de piridazinona usados para preparar un herbicida.
BR112022003039A2 (pt) 2019-09-25 2022-05-17 Nippon Soda Co Composto, herbicida, e, método para controlar ervas daninhas
UY39137A (es) 2020-04-01 2021-10-29 Fmc Corp Atropisómeros de derivados de piridazinona como herbicidas
CA3206162A1 (en) 2020-12-22 2022-06-30 Fmc Corporation Substituted pyridazinone herbicides

Citations (4)

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US20040225125A1 (en) * 2003-05-05 2004-11-11 New York University Solid phase synthesis of novel biaryl triazine library by suzuki cross coupling
WO2011045271A1 (de) * 2009-10-15 2011-04-21 Bayer Cropscience Ag Herbizid wirksame heterocyclylsubstituierte pyridazinone
WO2012091156A1 (en) * 2010-12-27 2012-07-05 Sumitomo Chemical Company, Limited Pyridazinone compound and herbicide and noxious arthropod controlling agent comprising it
CN103180300A (zh) * 2010-09-08 2013-06-26 住友化学株式会社 制备哒嗪酮化合物的方法和其中间体

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EP2042491A1 (de) 2007-09-14 2009-04-01 Bayer CropScience AG Pyridazine als Fungizide
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US20040225125A1 (en) * 2003-05-05 2004-11-11 New York University Solid phase synthesis of novel biaryl triazine library by suzuki cross coupling
WO2011045271A1 (de) * 2009-10-15 2011-04-21 Bayer Cropscience Ag Herbizid wirksame heterocyclylsubstituierte pyridazinone
CN103180300A (zh) * 2010-09-08 2013-06-26 住友化学株式会社 制备哒嗪酮化合物的方法和其中间体
WO2012091156A1 (en) * 2010-12-27 2012-07-05 Sumitomo Chemical Company, Limited Pyridazinone compound and herbicide and noxious arthropod controlling agent comprising it

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Also Published As

Publication number Publication date
US20180312467A1 (en) 2018-11-01
CA3003410A1 (en) 2017-05-04
AR106522A1 (es) 2018-01-24
JP6782774B2 (ja) 2020-11-11
WO2017074988A1 (en) 2017-05-04
HUE049157T2 (hu) 2020-09-28
ZA201803362B (en) 2019-08-28
KR20180075574A (ko) 2018-07-04
RU2018119134A3 (cg-RX-API-DMAC10.html) 2020-03-16
JP2018533580A (ja) 2018-11-15
MX2018005133A (es) 2019-01-10
EP3368531A1 (en) 2018-09-05
TWI739769B (zh) 2021-09-21
CN108779106A (zh) 2018-11-09
IL258765A (en) 2018-06-28
EP3368531B1 (en) 2020-01-15
AU2016346207B2 (en) 2020-06-04
US10913719B2 (en) 2021-02-09
RU2743561C2 (ru) 2021-02-19
TW201722917A (zh) 2017-07-01
SG11201803134VA (en) 2018-05-30
BR112018008616A2 (pt) 2019-11-26
AU2016346207A1 (en) 2018-05-10
BR112018008616B1 (pt) 2021-09-08
MX388612B (es) 2025-03-11
RU2018119134A (ru) 2019-11-28
IL258765B (en) 2021-01-31

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