CN1073554C - 邻氯甲基苯基二羟乙酸衍生物的制备方法 - Google Patents

邻氯甲基苯基二羟乙酸衍生物的制备方法 Download PDF

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Publication number
CN1073554C
CN1073554C CN96123428A CN96123428A CN1073554C CN 1073554 C CN1073554 C CN 1073554C CN 96123428 A CN96123428 A CN 96123428A CN 96123428 A CN96123428 A CN 96123428A CN 1073554 C CN1073554 C CN 1073554C
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CN
China
Prior art keywords
formula
compound
atoms
nitrogen
yuans
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Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
CN96123428A
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English (en)
Chinese (zh)
Other versions
CN1167756A (zh
Inventor
J-M·阿瑟克
H-D·施奈德
A·普菲弗纳
W·普法夫
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Bayer CropScience AG
Original Assignee
Novartis AG
Bayer AG
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Application filed by Novartis AG, Bayer AG filed Critical Novartis AG
Publication of CN1167756A publication Critical patent/CN1167756A/zh
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C251/00—Compounds containing nitrogen atoms doubly-bound to a carbon skeleton
    • C07C251/32—Oximes
    • C07C251/50—Oximes having oxygen atoms of oxyimino groups bound to carbon atoms of substituted hydrocarbon radicals
    • C07C251/52—Oximes having oxygen atoms of oxyimino groups bound to carbon atoms of substituted hydrocarbon radicals of hydrocarbon radicals substituted by halogen atoms or by nitro or nitroso groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
    • C07D295/14—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D295/155—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals with the ring nitrogen atoms and the carbon atoms with three bonds to hetero atoms separated by carbocyclic rings or by carbon chains interrupted by carbocyclic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C229/00—Compounds containing amino and carboxyl groups bound to the same carbon skeleton
    • C07C229/02—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton
    • C07C229/34—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton containing six-membered aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C249/00—Preparation of compounds containing nitrogen atoms doubly-bound to a carbon skeleton
    • C07C249/04—Preparation of compounds containing nitrogen atoms doubly-bound to a carbon skeleton of oximes
    • C07C249/08—Preparation of compounds containing nitrogen atoms doubly-bound to a carbon skeleton of oximes by reaction of hydroxylamines with carbonyl compounds
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C251/00—Compounds containing nitrogen atoms doubly-bound to a carbon skeleton
    • C07C251/32—Oximes
    • C07C251/34—Oximes with oxygen atoms of oxyimino groups bound to hydrogen atoms or to carbon atoms of unsubstituted hydrocarbon radicals
    • C07C251/48—Oximes with oxygen atoms of oxyimino groups bound to hydrogen atoms or to carbon atoms of unsubstituted hydrocarbon radicals with the carbon atom of at least one of the oxyimino groups bound to a carbon atom of a six-membered aromatic ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C251/00—Compounds containing nitrogen atoms doubly-bound to a carbon skeleton
    • C07C251/32—Oximes
    • C07C251/50—Oximes having oxygen atoms of oxyimino groups bound to carbon atoms of substituted hydrocarbon radicals
    • C07C251/60—Oximes having oxygen atoms of oxyimino groups bound to carbon atoms of substituted hydrocarbon radicals of hydrocarbon radicals substituted by carboxyl groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C69/00—Esters of carboxylic acids; Esters of carbonic or haloformic acids
    • C07C69/66—Esters of carboxylic acids having esterified carboxylic groups bound to acyclic carbon atoms and having any of the groups OH, O—metal, —CHO, keto, ether, acyloxy, groups, groups, or in the acid moiety
    • C07C69/73—Esters of carboxylic acids having esterified carboxylic groups bound to acyclic carbon atoms and having any of the groups OH, O—metal, —CHO, keto, ether, acyloxy, groups, groups, or in the acid moiety of unsaturated acids
    • C07C69/738—Esters of keto-carboxylic acids or aldehydo-carboxylic acids
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C69/00—Esters of carboxylic acids; Esters of carbonic or haloformic acids
    • C07C69/76—Esters of carboxylic acids having a carboxyl group bound to a carbon atom of a six-membered aromatic ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2601/00—Systems containing only non-condensed rings
    • C07C2601/02—Systems containing only non-condensed rings with a three-membered ring

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Steroid Compounds (AREA)
CN96123428A 1996-01-03 1996-12-30 邻氯甲基苯基二羟乙酸衍生物的制备方法 Expired - Lifetime CN1073554C (zh)

Applications Claiming Priority (8)

Application Number Priority Date Filing Date Title
CH196 1996-01-03
CH1/96 1996-01-03
CH1112/1996 1996-05-02
CH1112/96 1996-05-02
CH111296 1996-05-02
CH1874/96 1996-07-26
CH1874/1996 1996-07-26
CH187496 1996-07-26

Related Child Applications (2)

Application Number Title Priority Date Filing Date
CNB011174870A Division CN1185208C (zh) 1996-01-03 2001-04-29 邻氯甲基苯基二羟乙酸衍生物的制备方法
CNB011174889A Division CN1185209C (zh) 1996-01-03 2001-04-29 邻氯甲基苯基二羟乙酸衍生物的制备方法

Publications (2)

Publication Number Publication Date
CN1167756A CN1167756A (zh) 1997-12-17
CN1073554C true CN1073554C (zh) 2001-10-24

Family

ID=27171705

Family Applications (3)

Application Number Title Priority Date Filing Date
CN96123428A Expired - Lifetime CN1073554C (zh) 1996-01-03 1996-12-30 邻氯甲基苯基二羟乙酸衍生物的制备方法
CNB011174870A Expired - Lifetime CN1185208C (zh) 1996-01-03 2001-04-29 邻氯甲基苯基二羟乙酸衍生物的制备方法
CNB011174889A Expired - Lifetime CN1185209C (zh) 1996-01-03 2001-04-29 邻氯甲基苯基二羟乙酸衍生物的制备方法

Family Applications After (2)

Application Number Title Priority Date Filing Date
CNB011174870A Expired - Lifetime CN1185208C (zh) 1996-01-03 2001-04-29 邻氯甲基苯基二羟乙酸衍生物的制备方法
CNB011174889A Expired - Lifetime CN1185209C (zh) 1996-01-03 2001-04-29 邻氯甲基苯基二羟乙酸衍生物的制备方法

Country Status (23)

Country Link
US (2) US5756811A (enExample)
EP (1) EP0782982B1 (enExample)
JP (1) JP4621308B2 (enExample)
KR (2) KR100540153B1 (enExample)
CN (3) CN1073554C (enExample)
AR (1) AR005362A1 (enExample)
AT (1) ATE193010T1 (enExample)
AU (1) AU714429B2 (enExample)
BR (1) BR9700009A (enExample)
CA (1) CA2194203C (enExample)
CZ (1) CZ290146B6 (enExample)
DE (1) DE59605241D1 (enExample)
DK (1) DK0782982T3 (enExample)
ES (1) ES2147357T3 (enExample)
GR (1) GR3033714T3 (enExample)
HK (2) HK1048982A1 (enExample)
HU (1) HUP9603547A1 (enExample)
IL (1) IL119922A (enExample)
MX (1) MX9700003A (enExample)
PL (1) PL184464B1 (enExample)
PT (1) PT782982E (enExample)
SK (1) SK168996A3 (enExample)
TW (1) TW477785B (enExample)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR19990036612A (ko) * 1997-10-08 1999-05-25 고사이 아끼오 벤질 브로마이드 유도체의 제조 방법
GB9908530D0 (en) 1999-04-14 1999-06-09 Novartis Ag Organic compounds
US20100113778A1 (en) * 2007-04-12 2010-05-06 John-Matthias Wiegand Process for preparing o-chloromethylphenylglyoxylic esters, improved process for preparing (e)-2-(2-chloromethylphenyl)-2-alkoximinoacetic esters, and novel intermediates for their preparation
WO2009037230A2 (en) * 2007-09-17 2009-03-26 Dsm Fine Chemicals Austria Nfg Gmbh & Co Kg Improved process for preparing (e)-2-(2-chloromethylphenyl)-2-alkoximinoacetic esters
CN108358797A (zh) * 2018-04-20 2018-08-03 南京农业大学 一种烷基甘氨酸的合成方法

Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0420091A1 (de) * 1989-09-29 1991-04-03 BASF Aktiengesellschaft Neue Anilinderivate und diese enthaltende Fungizide
EP0585751A1 (de) * 1992-08-29 1994-03-09 BASF Aktiengesellschaft N-Methylamide, Verfahren und Zwischenprodukte zu ihrer Herstellung sowie Verfahren zur Bekämpfung von Schädlingen
DE4305502A1 (de) * 1993-02-23 1994-08-25 Basf Ag Ortho-substituierte 2-Methoxyiminophenylessigsäuremethylamide

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NZ213630A (en) * 1984-10-19 1990-02-26 Ici Plc Acrylic acid derivatives and fungicidal compositions
GB8617648D0 (en) 1986-07-18 1986-08-28 Ici Plc Fungicides
DE3835028A1 (de) * 1988-10-14 1990-04-19 Basf Ag Oximether-derivate, verfahren zu ihrer herstellung und diese enthaltende fungizide
DE3843439A1 (de) * 1988-12-23 1990-06-28 Basf Ag Schwefelhaltige oximether und diese enthaltende fungizide
HU219157B (hu) * 1994-01-05 2001-02-28 Novartis Ag. Peszticid hatású [dioxa-diaza/vagy oxa-triaza/-heptadienil-fenil]-akrilsav- és glioxilsav-származékok, előállításuk és alkalmazásuk
AU691863B2 (en) 1994-02-04 1998-05-28 Basf Aktiengesellschaft Phenyl acetic acid derivatives, process and intermediate products for their production and agents containing them
RU2146247C1 (ru) * 1994-06-10 2000-03-10 Басф Акциенгезельшафт СПОСОБЫ И ПРОМЕЖУТОЧНЫЕ ПРОДУКТЫ ДЛЯ ПОЛУЧЕНИЯ МЕТИЛАМИДОВ α-МЕТОКСИИМИНОКАРБОНОВЫХ КИСЛОТ
US5583249A (en) * 1994-08-19 1996-12-10 Ciba-Geigy Corporation Pesticides

Patent Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0420091A1 (de) * 1989-09-29 1991-04-03 BASF Aktiengesellschaft Neue Anilinderivate und diese enthaltende Fungizide
EP0585751A1 (de) * 1992-08-29 1994-03-09 BASF Aktiengesellschaft N-Methylamide, Verfahren und Zwischenprodukte zu ihrer Herstellung sowie Verfahren zur Bekämpfung von Schädlingen
DE4305502A1 (de) * 1993-02-23 1994-08-25 Basf Ag Ortho-substituierte 2-Methoxyiminophenylessigsäuremethylamide

Also Published As

Publication number Publication date
IL119922A (en) 2004-07-25
CN1368498A (zh) 2002-09-11
JPH09227486A (ja) 1997-09-02
CN1185208C (zh) 2005-01-19
ATE193010T1 (de) 2000-06-15
EP0782982A1 (de) 1997-07-09
CA2194203C (en) 2005-04-26
US5756811A (en) 1998-05-26
BR9700009A (pt) 1998-11-10
TW477785B (en) 2002-03-01
HUP9603547A1 (hu) 1998-01-28
HK1048983A1 (zh) 2003-04-25
ES2147357T3 (es) 2000-09-01
CN1185209C (zh) 2005-01-19
DK0782982T3 (da) 2000-10-09
MX9700003A (es) 1997-12-31
AR005362A1 (es) 1999-04-28
PL184464B1 (pl) 2002-11-29
CZ397A3 (cs) 1998-07-15
KR970059162A (ko) 1997-08-12
DE59605241D1 (de) 2000-06-21
HU9603547D0 (en) 1997-02-28
JP4621308B2 (ja) 2011-01-26
SK168996A3 (en) 1998-02-04
PL317751A1 (en) 1997-07-07
GR3033714T3 (en) 2000-10-31
CN1167756A (zh) 1997-12-17
EP0782982B1 (de) 2000-05-17
HK1048982A1 (zh) 2003-04-25
PT782982E (pt) 2000-10-31
US6124493A (en) 2000-09-26
KR100540148B1 (ko) 2005-12-29
KR100540153B1 (ko) 2006-04-20
CN1368497A (zh) 2002-09-11
CA2194203A1 (en) 1997-07-04
AU714429B2 (en) 2000-01-06
CZ290146B6 (cs) 2002-06-12
AU1000397A (en) 1997-07-10
IL119922A0 (en) 1997-03-18

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EXPY Termination of patent right or utility model