CN106860784A - 一种治疗角膜溃疡的药物及其制备方法 - Google Patents
一种治疗角膜溃疡的药物及其制备方法 Download PDFInfo
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Abstract
本发明公开了一种治疗角膜溃疡的药物及其制备方法,其主要是由金银花、柴胡、当归、决明子、瓜蒌子、虎杖、莱菔子、青葙子、防风、蔓荆子、知母、厚朴、枳壳、甘草、荆芥、枸杞子、钩藤、淡竹叶、薄荷、泽泻、车前子、连翘、川芎、羌活按一定重量配比制备而成,本发明药物具有清肝明目,疏风散热,滋阴降火的功能,用于治疗角膜溃疡见效快、疗效好,不复发。
Description
技术领域
本发明涉及一种治疗角膜溃疡的药物及其制备方法,属中药领域。
背景技术
角膜溃疡为常因异物等外伤,角膜异物剔除后损伤以及沙眼及其并发症、内翻倒睫刺伤角膜,细菌、病毒或真菌乘机而入,引起感染而发生角膜溃疡。中医则认为角膜溃疡与湿热蕴结,阴虚火旺,肝郁气滞有关。由于西药治疗副作用大,因此人们对有效治疗角膜溃疡的中药药物存在极大的需求,至今为止,还没有发现关于本发明的有关报道。
发明内容
本发明人依据中医理论的研究和临床试验的反复验证,终于找到了有效治疗角膜溃疡的药物,从而完成了本发明。
本发明的目的就是提供一种有效治疗角膜溃疡的中药组合药物。
本发明的另一目的就是提供了该中药组合药物的制备方法。
本发明药物是选择金银花、柴胡、当归、决明子、瓜蒌子、虎杖、莱菔子、青葙子、防风、蔓荆子、知母、厚朴、枳壳、甘草、荆芥、枸杞子、钩藤、淡竹叶、薄荷、泽泻、车前子、连翘、川芎、羌活、淡竹叶、苍术、山药进行组合制备的,将这些药物组合使得各药物功效产生协同作用,从而能够有效治疗角膜溃疡。其中选用金银花是因为其性味甘,寒,入肺、胃经,有清热,解毒的功能,治温病发热,热毒血痢,痈疡,肿毒,瘰疬,痔漏。选用柴胡是因为其性味苦,凉,入肝、胆经,有和解表里,疏肝,升阳的功能,治寒热往来,胸满胁痛,口苦耳聋,头痛目眩,疟疾,下利脱肛,月经不调,子宫下垂。选用当归是因为其性味甘辛,温,入心、肝、脾经,有补血和血,调经止痛,润燥滑肠的功能,治月经不调,经闭腹痛,癥瘕结聚,崩漏,血虚头痛,眩晕,痿痹,肠燥便难,赤痢后重,痈疽疮疡,跌扑损伤。选用决明子是因为其性味苦甘,凉,入肝、肾经,有清肝,明目,利水,通便的功能,治风热赤眼,青盲,雀目,高血压,肝炎,肝硬化腹化,习惯性便秘。选用瓜蒌子是因为其性味甘,寒,归肺、胃、大肠经,有润肺化痰,滑肠通便的功能,治燥咳痰黏,肠燥便秘。选用虎杖是因为其性味苦,平,有祛风,利湿,破瘀,通经的功能,治风湿筋骨疼痛,湿热黄疸,淋浊带下,妇女经闭,产后恶露不下,癥瘕积聚,痔漏下血,跌扑损伤,烫伤,恶疮癣疾。选用莱菔子是因为其性味辛甘,平,入肺、胃经,有下气定喘,消食化痰的功能,治咳嗽痰喘,食积气滞,胸闷腹胀,下痢后重。选用青葙子是因为其性味苦,凉,入肝经,有祛风热,清肝火的功能,治目赤肿痛,障翳,高血压,鼻衄,皮肤风热瘙痒,疥癞。选用防风是因为其性味辛甘,温,入膀胱、肺、脾经,有发表,祛风,胜湿,止痛的功能,治外感风寒,头痛,目眩,项强,风寒湿痹,骨节酸痛,四肢挛急,破伤风。选用蔓荆子是因为其性味苦辛,凉,入肝、胃,膀胱经,有疏散风热,清利头目的功能,治风热感冒,正、偏头痛,齿痛,目睛内痛。选用知母是因为其性味苦,寒,入肺、胃、肾经,有滋阴降火,润燥滑肠的功能,治烦热消渴,骨蒸劳热,肺热咳嗽,大便燥结,小便不利。选用厚朴是因为其性味苦辛,温,入脾、胃、大肠经,有温中,下气,燥湿,消痰的功能,治胸腹痞满胀痛,反胃、呕吐,宿食不消,痰饮喘咳,寒湿泻痢。选用枳壳是因为其性味苦辛,凉,入肺、脾、大肠经,有破气,行痰,消积的功能,治胸膈痰滞,胸痞,胁胀,食积,噫气,呕逆,下痢后重,脱肛,子宫脱垂。选用甘草是因为其性味甘平,归脾、胃肺经,有润肺,解毒的功能,炙用治脾胃虚弱,食少,腹痛,便溏,劳倦发热,肺痿咳嗽。选用荆芥是因为其性味辛,温,入肺、肝经,有发表,祛风,理血的功能,炒炭止血,治感冒发热,头痛,咽喉肿痛,中风口噤,吐血,衄血,便血,崩漏,产后血晕,痈肿,疮疥,瘰疬。选用枸杞子是因为其性味甘,平,有滋肾,润肺,补肝,明目的功能,治肝肾阴亏,腰膝酸软,头晕目眩,目昏多泪,虚劳咳嗽,消渴,遗清。钩藤是因为其性味苦,凉,入肝、心经,有清热平肝,熄风定惊的功能,治小儿惊癎瘈瘲,大人血压偏高,头晕、目眩,妇人子癎。选用淡竹叶是因为其性味甘淡,寒,入心肾二经,有清心火,除烦热,利小便的功能,治热病口渴,心烦,小便赤涩,淋浊,口糜舌疮,牙龈肿痛。选用薄荷是因为其性味辛,凉,入肺、肝经,有疏风,散热,辟秽,解毒的功能,治外感风热,头痛,目赤,咽喉肿痛,食滞气胀,口疮,牙痛,疮疥,瘾疹。选用泽泻是因为其性味甘,寒,入膀胱经,有利水,渗湿,泄热的功能,治小便不利,水肿肛满,呕吐,泻痢,痰饮,脚气,淋病,尿血。选用车前子是因为其性味甘,寒,入肾、膀胱经,有利水,清热,明目,祛痰的功能,治小便不通,淋浊,带下,尿血,暑湿泻痢,咳嗽多痰,湿痹,目赤障翳。选用连翘是因为其性味苦,凉,入心、肝、胆经,有清热,解毒,散结,消肿的功能,治温热,丹毒,斑疹,痈疡肿毒,瘰疬,小便淋闭。选用川芎是因为其性味辛,温,入肝、胆经,有行气开郁,祛风燥湿,活血止痛的功能,治风冷头痛旋晕,胁痛腹疼,寒痹筋挛,经闭,难产,产后瘀阻块痛,痈疽疮疡。选用羌活是因为其性味辛苦,温,入膀胱、肾经,有散表寒,祛风湿,利关节的功能,治感冒风寒,头痛无汗,风寒湿痹,项强筋急,骨节酸疼,风水浮肿,痈疽疮毒。选用淡竹叶是因为其性味甘淡,寒,入心肾二经,有清心火,除烦热,利小便的功能,治热病口渴,心烦,小便赤涩,淋浊,口糜舌疮,牙龈肿痛。选用苍术是因为其性味辛苦,温,入脾、胃经,有健脾,燥湿,解郁,辟秽的功能,治湿盛困脾,倦怠嗜卧,脘痞腹胀,食欲不振,呕吐,泄泻,痢疾,疟疾,痰饮,水肿,时气感冒,风寒湿痹,足痿,夜盲。选用山药是因为其性味甘,平,入肺、脾、肾经,有健脾,补肺,固肾,益精的功能,治脾虚泄泻,久痢,虚劳咳嗽,消渴,遗精、带下,小便频数。
具体实施方式
本发明组分的药物用量也是发明人经过大量摸索总结得出的,各组分的用量在下述重量范围内都具有较好的疗效:
金银花10-20克,柴胡5-15克,当归10-15克,决明子20-30克,瓜蒌子10-20克,虎杖5-10克,莱菔子5-15克,青葙子10-20克,防风5-15克,蔓荆子5-15克,知母5-15克,厚朴5-10克,枳壳5-15克,甘草5-10克,荆芥10-20克,枸杞子5-10克,钩藤10-15克,淡竹叶10-20克,薄荷5-15克,泽泻10-15克,车前子10-20克,连翘5-15克,川芎10-15克,羌活5-15克,淡竹叶10-15克,苍术10-20克,山药5-15克。
优选为:
金银花15克,柴胡10克,当归12克,决明子25克,瓜蒌子15克,虎杖8克,莱菔子10克,青葙子15克,防风10克,蔓荆子10克,知母10克,厚朴8克,枳壳10克,甘草8克,荆芥15克,枸杞子8克,钩藤12克,淡竹叶15克,薄荷10克,泽泻12克,车前子15克,连翘10克,川芎12克,羌活10克,淡竹叶12克,苍术15克,山药10克。
本发明药物的制备方法如下
一、备料
1、金银花:筛去泥沙,拣净杂质;
2、柴胡:拣去杂质,除去残茎,洗净泥沙,捞出,润透后及时切片,随即晒干;
3、当归:拣去杂质,洗净,闷润,稍晾,切片晒干;
4、决明子:取净决明子,置锅内炒至微有香气,取出,放凉;
5、瓜蒌子:取原药材,除去干瘪种子、杂质,用时捣碎;
6、虎杖:采得后,细锉,晒干;
7、莱菔子:簸去杂质,漂净泥土,捞出,晒干,用时捣碎;
8、青葙子:取原药材,除去杂质,筛去灰屑;
9、防风:除去残茎,用水浸泡,捞出,润透切片,晒干;
10、蔓荆子:筛净灰屑,除去残存萼片,置锅内用武火炒至焦黄色,略喷清水,放凉;
11、知母:拣净杂质,用水撞洗,捞出,润软,切片晒干;
12、厚朴:用水浸泡捞出,润透后刮去粗皮,洗净,切丝,晾干;
13、枳壳:除去瓤、核,冼净,稍浸,捞出,润软,以手能捏对折为止,切片,晾干;
14、甘草:拣去杂质,洗净,用水浸泡至八成透时,捞出,润透,切片,凉干;
15、荆芥:拣净杂质,用水略泡,捞出切段,晒干;
16、枸杞子:簸净杂质,摘去残留的梗和蒂;
17、钩藤:拣去老梗、杂质,洗净,晒干;
18、淡竹叶:拣去杂质及根,切段,晒干;
19、薄荷:拣净杂质,除去残根,先将叶抖下另放,然后将茎喷洒清水,润透后切段,晒干,再与叶和匀;
20、泽泻:拣去杂质,大小分档,用水浸泡至八成透,捞出,晒凉,闷润至内外湿度均匀,切片,晒干;
21、车前子:拣去杂质,筛去泥屑,空粒;
22、连翘:拣净杂质,搓开,除去枝梗;
23、川芎:拣去杂质,分开大、小个,用水浸泡,晒晾,闷润后切片,干燥;
24、羌活:拣去杂质,洗净,润透,切片,晾干;
25、淡竹叶:拣去杂质及根,切段,晒干;
26、苍术:拣去杂质,用水泡至七、八成透,捞出,润透后切片,晒干;
27、山药:拣净杂质,用水浸泡至山药中心部软化为度,捞出稍晾,切片晒干或烘干。
二、制备
1、将所述重量的金银花、柴胡、当归、决明子、瓜蒌子、虎杖、莱菔子、青葙子、防风、蔓荆子、知母、厚朴、枳壳、甘草、荆芥、枸杞子、钩藤、淡竹叶、薄荷、泽泻、车前子、连翘、川芎、羌活、淡竹叶、苍术、山药放入煎药容器内,第一次加水8倍量,浸泡100分钟后,武火煎煮沸腾,再用文火煎煮20分钟,过滤得第一次煎煮液,将第一次煎煮液倒入容器内;
2、将过滤的药渣加水5倍量,武火煮沸,再用文火煎煮20分钟,过滤得第二次煎煮液;
3、将两次煎煮液混合搅拌均匀,分为3剂服用。
组方中决明子有清肝,明目,利水,通便的功能为君药;青葙子祛风热,清肝火;知母有滋阴降火的功能,二者为臣药,三味药共同发挥清肝,明目,利水,通便,祛风热,滋阴降火的作用,治疗角膜溃疡效力全面,且以清肝,明目,利水,祛风热,滋阴降火为主可治本,蔓荆子有疏散风热,清利头目的功能为佐药,枸杞子有滋肾,润肺,补肝,明目的功能的功能为使药,与下余诸药是治标。
本发明药物具有清肝明目,疏风散热,滋阴降火的功能,用于治疗角膜溃疡,疗程短、见效快、治愈后不复发。
以下通过试验例来进一步阐述本发明所述药物的有益效果,这些试验例包括本发明药物的动物毒性试验报告和临床疗效观察资料。
[试验例1]本发明药物的动物毒性试验报告:
取家兔30只,雌雄兼用,体重2.0—2.5kg,分两组,每组15只,其中一组为超剂量试验组,另一组为正常量试验组。超常量组为20ml/kg,正常量为10ml/kg,给药方式为灌胃法给药,每天两次,连服7天,每天观察给药反应,结果表明二组家兔活动、饮食正常,药物无不良毒副作用。
[试验例2]本发明药物的临床疗效观察
1、一般资料
收治角膜溃疡门诊患者共13例。
2、诊断标准
典型症状为怕光、流泪、眼痛、角膜上出现灰白色小点或片状浸润;严重时上述症状更加明显,睁不开眼,眼痛难忍,视力减退。
3、治疗方法
选用上述药剂,给患者服用,每次服用1剂,每天早、晚各服1次,7天为一个疗程,连续服用3个疗程。
4、疗效评定标准
显效:角膜溃疡症状消失,恢复正常,痊愈;
好转:患者怕光、流泪、眼痛、视力减退的现象减轻,角膜溃疡症状明显好转,体质逐步恢复;
无效:达不到好转标准者。
5、治疗结果(见下表)
在上述治疗中,用本发明药物治疗角膜溃疡患者13例,结果显效10例,显效率为76.91%,好转2例,好转率为15.39%,无效1例,总有效率为92.3%。
Claims (3)
1.一种治疗角膜溃疡的药物,其特征在于:它是由下列重量范围内的原料药制成:
金银花10-20克,柴胡5-15克,当归10-15克,决明子20-30克,瓜蒌子10-20克,虎杖5-10克,莱菔子5-15克,青葙子10-20克,防风5-15克,蔓荆子5-15克,知母5-15克,厚朴5-10克,枳壳5-15克,甘草5-10克,荆芥10-20克,枸杞子5-10克,钩藤10-15克,淡竹叶10-20克,薄荷5-15克,泽泻10-15克,车前子10-20克,连翘5-15克,川芎10-15克,羌活5-15克,淡竹叶10-15克,苍术10-20克,山药5-15克。
2.根据权利要求1所述的药物,其中各原料药的用量为:
金银花15克,柴胡10克,当归12克,决明子25克,瓜蒌子15克,虎杖8克,莱菔子10克,青葙子15克,防风10克,蔓荆子10克,知母10克,厚朴8克,枳壳10克,甘草8克,荆芥15克,枸杞子8克,钩藤12克,淡竹叶15克,薄荷10克,泽泻12克,车前子15克,连翘10克,川芎12克,羌活10克,淡竹叶12克,苍术15克,山药10克。
3.根据权利要求1或2所述药物的制备方法,它包括下列步骤:
(一)备料
(1)金银花:筛去泥沙,拣净杂质;
(2)柴胡:拣去杂质,除去残茎,洗净泥沙,捞出,润透后及时切片,随即晒干;
(3)当归:拣去杂质,洗净,闷润,稍晾,切片晒干;
(4)决明子:取净决明子,置锅内炒至微有香气,取出,放凉;
(5)瓜蒌子:取原药材,除去干瘪种子、杂质,用时捣碎;
(6)虎杖:采得后,细锉,晒干;
(7)莱菔子:簸去杂质,漂净泥土,捞出,晒干,用时捣碎;
(8)青葙子:取原药材,除去杂质,筛去灰屑;
(9)防风:除去残茎,用水浸泡,捞出,润透切片,晒干;
(10)蔓荆子:筛净灰屑,除去残存萼片,置锅内用武火炒至焦黄色,略喷清水,放凉;
(11)知母:拣净杂质,用水撞洗,捞出,润软,切片晒干;
(12)厚朴:用水浸泡捞出,润透后刮去粗皮,洗净,切丝,晾干;
(13)枳壳:除去瓤、核,冼净,稍浸,捞出,润软,以手能捏对折为止,切片,晾干;
(14)甘草:拣去杂质,洗净,用水浸泡至八成透时,捞出,润透,切片,凉干;
(15)荆芥:拣净杂质,用水略泡,捞出切段,晒干;
(16)枸杞子:簸净杂质,摘去残留的梗和蒂;
(17)钩藤:拣去老梗、杂质,洗净,晒干;
(18)淡竹叶:拣去杂质及根,切段,晒干;
(19)薄荷:拣净杂质,除去残根,先将叶抖下另放,然后将茎喷洒清水,润透后切段,晒干,再与叶和匀;
(20)泽泻:拣去杂质,大小分档,用水浸泡至八成透,捞出,晒凉,闷润至内外湿度均匀,切片,晒干;
(21)车前子:拣去杂质,筛去泥屑,空粒;
(22)连翘:拣净杂质,搓开,除去枝梗;
(23)川芎:拣去杂质,分开大、小个,用水浸泡,晒晾,闷润后切片,干燥;
(24)羌活:拣去杂质,洗净,润透,切片,晾干;
(25)淡竹叶:拣去杂质及根,切段,晒干;
(26)苍术:拣去杂质,用水泡至七、八成透,捞出,润透后切片,晒干;
(27)山药:拣净杂质,用水浸泡至山药中心部软化为度,捞出稍晾,切片晒干或烘干;
(二)制备
(1)将所述重量的金银花、柴胡、当归、决明子、瓜蒌子、虎杖、莱菔子、青葙子、防风、蔓荆子、知母、厚朴、枳壳、甘草、荆芥、枸杞子、钩藤、淡竹叶、薄荷、泽泻、车前子、连翘、川芎、羌活、淡竹叶、苍术、山药放入煎药容器内,加水8倍量,浸泡100分钟后,武火煎煮沸腾,再用文火煎煮20分钟,过滤得第一次煎煮液,将第一次煎煮液倒入容器内;
(2)将过滤的药渣加水5倍量,武火煮沸,再用文火煎煮20分钟,过滤得第二次煎煮液;
(3)将两次煎煮液混合搅拌均匀,分为3剂服用。
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