CN106456587B - 含有欧米茄-3和白藜芦醇的固体制剂 - Google Patents

含有欧米茄-3和白藜芦醇的固体制剂 Download PDF

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Publication number
CN106456587B
CN106456587B CN201580029892.0A CN201580029892A CN106456587B CN 106456587 B CN106456587 B CN 106456587B CN 201580029892 A CN201580029892 A CN 201580029892A CN 106456587 B CN106456587 B CN 106456587B
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omega
acid
polyunsaturated fatty
weight
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Expired - Fee Related
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CN106456587A (zh
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G·詹尼尼
M·圣阿涅洛
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Alpha Sigma Co ltd
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Alpha Sigmar Joint-Stock Co
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    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19—Carboxylic acids, e.g. valproic acid
    • A61K31/20—Carboxylic acids, e.g. valproic acid having a carboxyl group bound to a chain of seven or more carbon atoms, e.g. stearic, palmitic, arachidic acids
    • A61K31/202—Carboxylic acids, e.g. valproic acid having a carboxyl group bound to a chain of seven or more carbon atoms, e.g. stearic, palmitic, arachidic acids having three or more double bonds, e.g. linolenic
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605—Excipients; Inactive ingredients
    • A61K9/1611—Inorganic compounds
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    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/045—Hydroxy compounds, e.g. alcohols; Salts thereof, e.g. alcoholates
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    • A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/10—Alcohols; Phenols; Salts thereof, e.g. glycerol; Polyethylene glycols [PEG]; Poloxamers; PEG/POE alkyl ethers
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    • A61K9/167—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction with an outer layer or coating comprising drug; with chemically bound drugs or non-active substances on their surface
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    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
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    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841—Filling excipients; Inactive ingredients
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    • A61P9/00—Drugs for disorders of the cardiovascular system
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  • Pharmacology & Pharmacy (AREA)
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  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Inorganic Chemistry (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Nutrition Science (AREA)
  • Physiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Rheumatology (AREA)
  • Cardiology (AREA)
  • Pulmonology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Obesity (AREA)
  • Toxicology (AREA)
  • Oncology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Biochemistry (AREA)
  • Hospice & Palliative Care (AREA)
  • Vascular Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Psychiatry (AREA)
  • Emergency Medicine (AREA)
  • Pain & Pain Management (AREA)
  • Immunology (AREA)
CN201580029892.0A 2014-06-04 2015-03-26 含有欧米茄-3和白藜芦醇的固体制剂 Expired - Fee Related CN106456587B (zh)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP14001940.7 2014-06-04
EP14001940.7A EP2952180B1 (en) 2014-06-04 2014-06-04 Solid formulations containing resveratrol and omega-3 polyunsaturated fatty acids (n-3 PUFA)
PCT/EP2015/056530 WO2015185239A1 (en) 2014-06-04 2015-03-26 Solid formulations containing omega-3 and resveratrol

Publications (2)

Publication Number Publication Date
CN106456587A CN106456587A (zh) 2017-02-22
CN106456587B true CN106456587B (zh) 2020-03-20

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CN201580029892.0A Expired - Fee Related CN106456587B (zh) 2014-06-04 2015-03-26 含有欧米茄-3和白藜芦醇的固体制剂

Country Status (14)

Country Link
US (1) US20170112791A1 (enExample)
EP (1) EP2952180B1 (enExample)
JP (1) JP2017522278A (enExample)
CN (1) CN106456587B (enExample)
AU (1) AU2015271278A1 (enExample)
CA (1) CA2943021A1 (enExample)
EA (1) EA032762B1 (enExample)
ES (1) ES2615630T3 (enExample)
MX (1) MX369782B (enExample)
PL (1) PL2952180T3 (enExample)
PT (1) PT2952180T (enExample)
SI (1) SI2952180T1 (enExample)
UA (1) UA119174C2 (enExample)
WO (1) WO2015185239A1 (enExample)

Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2009034124A1 (en) * 2007-09-12 2009-03-19 Novozymes A/S Omega-3 stabilisation towards oxidation
US20100247632A1 (en) * 2009-03-24 2010-09-30 Dong Liang C Stabilized solubility-enhanced formulations for oral delivery
US20110244031A1 (en) * 2010-03-31 2011-10-06 Lifecycle Pharma A/S Porous tablets as carriers for liquid formulations

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2004026950A2 (en) * 2002-08-14 2004-04-01 E.I. Du Pont De Nemours And Company Solid flowable powder with high liquid loading
ITRM20020562A1 (it) 2002-11-06 2004-05-07 Sigma Tau Ind Farmaceuti Uso del resveratrolo per la preparazione di un medicamento utile per il trattamento delle infezioni da virus dell'influenza.
KR101100078B1 (ko) * 2008-03-27 2011-12-29 홉킨스바이오연구센터(주) 관절염 치료를 위한 약제학적 조성물
CN102665698A (zh) 2009-12-23 2012-09-12 迪菲安特制药有限责任公司 可用于治疗心血管疾病的联合组合物
IT1400695B1 (it) 2010-06-21 2013-06-28 Labomar S R L Composizioni farmaceutiche e/o nutraceutiche contenenti principi attivi insolubili in acqua e procedimento per ottenerle.
CA3142049C (en) * 2012-09-12 2023-08-29 Novaliq Gmbh Semifluorinated alkane compositions

Patent Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2009034124A1 (en) * 2007-09-12 2009-03-19 Novozymes A/S Omega-3 stabilisation towards oxidation
US20100247632A1 (en) * 2009-03-24 2010-09-30 Dong Liang C Stabilized solubility-enhanced formulations for oral delivery
US20110244031A1 (en) * 2010-03-31 2011-10-06 Lifecycle Pharma A/S Porous tablets as carriers for liquid formulations

Also Published As

Publication number Publication date
CN106456587A (zh) 2017-02-22
JP2017522278A (ja) 2017-08-10
ES2615630T3 (es) 2017-06-07
CA2943021A1 (en) 2015-12-10
PL2952180T3 (pl) 2017-05-31
SI2952180T1 (sl) 2017-05-31
EP2952180A1 (en) 2015-12-09
EA201692399A1 (ru) 2017-03-31
EA032762B1 (ru) 2019-07-31
WO2015185239A1 (en) 2015-12-10
PT2952180T (pt) 2017-03-02
AU2015271278A1 (en) 2016-11-10
MX369782B (es) 2019-11-21
US20170112791A1 (en) 2017-04-27
MX2016013189A (es) 2017-01-16
UA119174C2 (uk) 2019-05-10
EP2952180B1 (en) 2017-01-25

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