CN105705161A - 赖谷胰岛素的稳定制剂 - Google Patents
赖谷胰岛素的稳定制剂 Download PDFInfo
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- CN105705161A CN105705161A CN201480058603.5A CN201480058603A CN105705161A CN 105705161 A CN105705161 A CN 105705161A CN 201480058603 A CN201480058603 A CN 201480058603A CN 105705161 A CN105705161 A CN 105705161A
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- China
- Prior art keywords
- aqueous pharmaceutical
- pharmaceutical preparations
- insulin
- diabetes
- glulisine
- Prior art date
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- A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- A61K38/22—Hormones
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- A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- A61K38/22—Hormones
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- A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
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- A61K47/20—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing sulfur, e.g. dimethyl sulfoxide [DMSO], docusate, sodium lauryl sulfate or aminosulfonic acids
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Landscapes
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- Emergency Medicine (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Medicinal Preparation (AREA)
Applications Claiming Priority (3)
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| EP13306475.8 | 2013-10-25 | ||
| EP13306475 | 2013-10-25 | ||
| PCT/EP2014/072915 WO2015059302A1 (en) | 2013-10-25 | 2014-10-24 | Stable formulation of insulin glulisine |
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| CN105705161A true CN105705161A (zh) | 2016-06-22 |
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| KR (1) | KR20160074562A (enExample) |
| CN (1) | CN105705161A (enExample) |
| AR (1) | AR098168A1 (enExample) |
| AU (1) | AU2014338863A1 (enExample) |
| BR (1) | BR112016008736A2 (enExample) |
| CA (1) | CA2928320A1 (enExample) |
| CL (1) | CL2016000950A1 (enExample) |
| HK (1) | HK1225613A1 (enExample) |
| IL (1) | IL245109A0 (enExample) |
| MX (1) | MX2016005395A (enExample) |
| PH (1) | PH12016500720A1 (enExample) |
| RU (1) | RU2691059C2 (enExample) |
| SG (2) | SG11201602939QA (enExample) |
| TW (1) | TW201605489A (enExample) |
| WO (1) | WO2015059302A1 (enExample) |
Families Citing this family (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP5694779B2 (ja) | 2008-01-09 | 2015-04-01 | サノフィ−アベンティス・ドイチュラント・ゲゼルシャフト・ミット・ベシュレンクテル・ハフツング | 極度に遅延した時間作用プロファイルを有する新規なインスリン誘導体 |
| LT3228320T (lt) | 2008-10-17 | 2020-03-10 | Sanofi-Aventis Deutschland Gmbh | Insulino ir glp-1 agonisto derinys |
| PL2498802T3 (pl) | 2009-11-13 | 2015-06-30 | Sanofi Aventis Deutschland | Kompozycja farmaceutyczna zawierająca agonistę GLP-1, insulinę i metioninę |
| EP2498801B1 (de) | 2009-11-13 | 2018-01-24 | Sanofi-Aventis Deutschland GmbH | HARMAZEUTISCHE ZUSAMMENSETZUNG UMFASSEND desPro36Exendin-4(1-39)-Lys6-NH2 UND METHIONIN |
| SI2611458T1 (sl) | 2010-08-30 | 2017-01-31 | Sanofi-Aventis Deutschland Gmbh | Uporaba AVE0010 za izdelavo zdravila za zdravljenje sladkorne bolezni tipa 2 |
| US9821032B2 (en) | 2011-05-13 | 2017-11-21 | Sanofi-Aventis Deutschland Gmbh | Pharmaceutical combination for improving glycemic control as add-on therapy to basal insulin |
| AR087744A1 (es) | 2011-09-01 | 2014-04-16 | Sanofi Aventis Deutschland | Composicion farmaceutica para uso en el tratamiento de una enfermedad neurodegenerativa |
| CA2970200A1 (en) | 2014-12-12 | 2016-06-16 | Sanofi-Aventis Deutschland Gmbh | Insulin glargine/lixisenatide fixed ratio formulation |
| TWI748945B (zh) | 2015-03-13 | 2021-12-11 | 德商賽諾菲阿凡提斯德意志有限公司 | 第２型糖尿病病患治療 |
| TW201705975A (zh) | 2015-03-18 | 2017-02-16 | 賽諾菲阿凡提斯德意志有限公司 | 第２型糖尿病病患之治療 |
| GB201607918D0 (en) * | 2016-05-06 | 2016-06-22 | Arecor Ltd | Novel formulations |
| IL277721B2 (en) | 2018-04-04 | 2024-03-01 | Arecor Ltd | Medical infusion pump system for the delivery of an insulin compound |
| FR3083700B1 (fr) * | 2018-07-13 | 2021-03-12 | Adocia | Formulation thermostable d'insuline humaine a21g |
| AR131148A1 (es) * | 2022-11-26 | 2025-02-19 | Obshchestvo S Ogranichennoy Otvetstvennostyu «Geropharm» | Composiciones de insulina de acción rápida (variantes de las mismas) |
Citations (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN1498113A (zh) * | 2001-03-23 | 2004-05-19 | ������ҽҩ�¹�����˾ | 稳定性提高的无锌或低锌胰岛素制剂 |
| WO2011085393A1 (en) * | 2010-01-11 | 2011-07-14 | Genecopoeia, Inc. | Stable insulin formulations and methods of making and using thereof |
| CN102596175A (zh) * | 2009-07-06 | 2012-07-18 | 赛诺菲-安万特德国有限公司 | 含有甲硫氨酸的水性胰岛素制备物 |
| WO2012174478A2 (en) * | 2011-06-17 | 2012-12-20 | Halozyme, Inc. | Stable formulations of a hyaluronan-degrading enzyme |
Family Cites Families (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5474978A (en) | 1994-06-16 | 1995-12-12 | Eli Lilly And Company | Insulin analog formulations |
| US5866538A (en) | 1996-06-20 | 1999-02-02 | Novo Nordisk A/S | Insulin preparations containing NaCl |
| US5948751A (en) | 1996-06-20 | 1999-09-07 | Novo Nordisk A/S | X14-mannitol |
| AR012894A1 (es) | 1997-06-13 | 2000-11-22 | Lilly Co Eli | Formulacion de insulina en solucion estable, su uso para preparar un medicamento y proceso para la preparacion de la misma. |
| TWI394580B (zh) * | 2008-04-28 | 2013-05-01 | Halozyme Inc | 超快起作用胰島素組成物 |
| EP2308473A4 (en) * | 2008-07-01 | 2013-01-09 | Nitto Denko Corp | PHARMACEUTICAL COMPOSITION CONTAINING MICROPARTICLES WITH SURFACE COATING |
| MA33467B1 (fr) * | 2009-07-31 | 2012-07-03 | Sanofi Aventis Deutschland | Promédicaments comprenant un conjugué insuline-lieur |
| PL2498802T3 (pl) * | 2009-11-13 | 2015-06-30 | Sanofi Aventis Deutschland | Kompozycja farmaceutyczna zawierająca agonistę GLP-1, insulinę i metioninę |
| US20130011378A1 (en) * | 2011-06-17 | 2013-01-10 | Tzung-Horng Yang | Stable formulations of a hyaluronan-degrading enzyme |
| CN104902922B (zh) * | 2012-11-13 | 2017-12-12 | 阿道恰公司 | 包含经取代阴离子化合物的速效胰岛素制剂 |
| AU2015205620A1 (en) * | 2014-01-09 | 2016-07-14 | Sanofi | Stabilized pharmaceutical formulations of insulin aspart |
-
2014
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- 2014-10-24 RU RU2016119746A patent/RU2691059C2/ru not_active IP Right Cessation
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- 2014-10-24 SG SG10201803430SA patent/SG10201803430SA/en unknown
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- 2014-10-24 EP EP14789560.1A patent/EP3060240A1/en not_active Withdrawn
- 2014-10-24 JP JP2016524503A patent/JP6525987B2/ja not_active Expired - Fee Related
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|---|---|---|---|---|
| CN1498113A (zh) * | 2001-03-23 | 2004-05-19 | ������ҽҩ�¹�����˾ | 稳定性提高的无锌或低锌胰岛素制剂 |
| CN102596175A (zh) * | 2009-07-06 | 2012-07-18 | 赛诺菲-安万特德国有限公司 | 含有甲硫氨酸的水性胰岛素制备物 |
| WO2011085393A1 (en) * | 2010-01-11 | 2011-07-14 | Genecopoeia, Inc. | Stable insulin formulations and methods of making and using thereof |
| WO2012174478A2 (en) * | 2011-06-17 | 2012-12-20 | Halozyme, Inc. | Stable formulations of a hyaluronan-degrading enzyme |
Also Published As
| Publication number | Publication date |
|---|---|
| JP6525987B2 (ja) | 2019-06-05 |
| KR20160074562A (ko) | 2016-06-28 |
| IL245109A0 (en) | 2016-06-30 |
| RU2016119746A3 (enExample) | 2018-06-04 |
| AU2014338863A1 (en) | 2016-05-19 |
| CA2928320A1 (en) | 2015-04-30 |
| SG10201803430SA (en) | 2018-06-28 |
| TW201605489A (zh) | 2016-02-16 |
| HK1225613A1 (zh) | 2017-09-15 |
| US20180036411A1 (en) | 2018-02-08 |
| PH12016500720A1 (en) | 2016-05-30 |
| EP3060240A1 (en) | 2016-08-31 |
| AR098168A1 (es) | 2016-05-04 |
| SG11201602939QA (en) | 2016-05-30 |
| CL2016000950A1 (es) | 2016-11-04 |
| RU2691059C2 (ru) | 2019-06-10 |
| US20150119323A1 (en) | 2015-04-30 |
| MX2016005395A (es) | 2017-02-28 |
| WO2015059302A1 (en) | 2015-04-30 |
| RU2016119746A (ru) | 2017-11-30 |
| JP2016539921A (ja) | 2016-12-22 |
| BR112016008736A2 (pt) | 2017-09-12 |
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