CN104321048B - 抑制神经元胞吐的化合物(ii) - Google Patents

抑制神经元胞吐的化合物(ii) Download PDF

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Publication number
CN104321048B
CN104321048B CN201380026300.0A CN201380026300A CN104321048B CN 104321048 B CN104321048 B CN 104321048B CN 201380026300 A CN201380026300 A CN 201380026300A CN 104321048 B CN104321048 B CN 104321048B
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agent
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reagent
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English (en)
Chinese (zh)
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CN104321048A (zh
Inventor
A·菲尔勒蒙蒂埃尔
G·费尔南德兹巴勒斯特尔
J·M·加西亚安东
C·卡雷诺塞尔莱马
N·阿尔米尼亚纳多梅内奇
R·德尔加多冈萨雷斯
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Lubrizol Advanced Materials Inc
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Lubrizol Advanced Materials Inc
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Priority claimed from EP12382144.9A external-priority patent/EP2649983A1/en
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/04—Linear peptides containing only normal peptide links
    • C07K7/06—Linear peptides containing only normal peptide links having 5 to 11 amino acids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00—Cosmetics or similar toiletry preparations
    • A61K8/02—Cosmetics or similar toiletry preparations characterised by special physical form
    • A61K8/11—Encapsulated compositions
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00—Cosmetics or similar toiletry preparations
    • A61K8/02—Cosmetics or similar toiletry preparations characterised by special physical form
    • A61K8/14—Liposomes; Vesicles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00—Cosmetics or similar toiletry preparations
    • A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/30—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
    • A61K8/64—Proteins; Peptides; Derivatives or degradation products thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/06—Antipsoriatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/10—Anti-acne agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/12—Keratolytics, e.g. wart or anti-corn preparations
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/14—Drugs for dermatological disorders for baldness or alopecia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/16—Emollients or protectives, e.g. against radiation
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61Q—SPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
    • A61Q19/00—Preparations for care of the skin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61Q—SPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
    • A61Q15/00—Anti-perspirants or body deodorants
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

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  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • Dermatology (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Birds (AREA)
  • Epidemiology (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Toxicology (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Cosmetics (AREA)
  • Peptides Or Proteins (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
CN201380026300.0A 2012-04-13 2013-04-12 抑制神经元胞吐的化合物(ii) Active CN104321048B (zh)

Applications Claiming Priority (9)

Application Number Priority Date Filing Date Title
EP12382144.9A EP2649983A1 (en) 2012-04-13 2012-04-13 Compounds which inhibit neuronal exocytosis (II)
EP12382144.9 2012-04-13
US201261652647P 2012-05-29 2012-05-29
US61/652,647 2012-05-29
EP12382303 2012-07-27
EP12382303.1 2012-07-27
US201261746888P 2012-12-28 2012-12-28
US61/746,888 2012-12-28
PCT/EP2013/057656 WO2013153191A1 (en) 2012-04-13 2013-04-12 Compounds which inhibit neuronal exocytosis (ii)

Publications (2)

Publication Number Publication Date
CN104321048A CN104321048A (zh) 2015-01-28
CN104321048B true CN104321048B (zh) 2019-01-11

Family

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Family Applications (1)

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CN201380026300.0A Active CN104321048B (zh) 2012-04-13 2013-04-12 抑制神经元胞吐的化合物(ii)

Country Status (11)

Country Link
US (1) US10035820B2 (enExample)
EP (1) EP2836193B1 (enExample)
JP (1) JP6470678B2 (enExample)
KR (1) KR102113994B1 (enExample)
CN (1) CN104321048B (enExample)
AU (1) AU2013246882B2 (enExample)
BR (1) BR112014025396B1 (enExample)
CA (1) CA2869599C (enExample)
ES (1) ES2660901T3 (enExample)
MX (1) MX356343B (enExample)
WO (1) WO2013153191A1 (enExample)

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US10154958B1 (en) 2017-07-20 2018-12-18 King Abdulaziz University Composition containing essential oils and plant extracts for treating vaginal infection and inflammation
JP7523358B2 (ja) * 2018-06-13 2024-07-26 アジェンデ・キミケ・リウニテ・アンジェリニ・フランチェスコ・ア・チ・エレ・ア・エフェ・ソシエタ・ペル・アチオニ ムスカリン受容体ｍ３に対して阻害活性を有するペプチド
US12274731B1 (en) 2018-07-12 2025-04-15 Washington University Polybasic antimalarial agents and methods of use thereof
WO2020142211A1 (en) 2019-01-02 2020-07-09 The Procter & Gamble Company Skin care compositions containing peptide compound and aphanothece sacrum exopolysaccharide extract
MY205382A (en) * 2019-05-21 2024-10-18 Eyebio Korea Novel peptide compound or pharmaceutically acceptable salt thereof
US12246024B2 (en) 2019-12-13 2025-03-11 Free State Pharma Inc Compositions and methods for controlling cerumen production
CN111345293B (zh) * 2020-04-08 2021-08-27 江门海关技术中心 一种虫类标本用防蛀剂及其制备方法
KR102584000B1 (ko) 2021-01-19 2023-10-06 김기연 신경전달물질을 조절하는 펩타이드를 포함하는 스포츠 로션 조성물
US11571378B2 (en) 2021-01-22 2023-02-07 The Procter & Gamble Company Skin care composition and method of using the same
US11771637B2 (en) 2021-01-22 2023-10-03 The Procter & Gamble Company Skin care composition and method of using the same
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Also Published As

Publication number Publication date
CA2869599C (en) 2021-07-27
CN104321048A (zh) 2015-01-28
BR112014025396B1 (pt) 2020-03-17
EP2836193B1 (en) 2018-01-31
KR20150002800A (ko) 2015-01-07
AU2013246882B2 (en) 2017-10-19
CA2869599A1 (en) 2013-10-17
EP2836193A1 (en) 2015-02-18
AU2013246882A1 (en) 2014-10-09
JP6470678B2 (ja) 2019-02-13
KR102113994B1 (ko) 2020-05-25
US10035820B2 (en) 2018-07-31
WO2013153191A1 (en) 2013-10-17
US20150098989A1 (en) 2015-04-09
MX2014012223A (es) 2014-11-25
ES2660901T3 (es) 2018-03-26
JP2015514124A (ja) 2015-05-18
MX356343B (es) 2018-05-23

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