CN103974932B - 手性催化剂及其盐的制备方法 - Google Patents
手性催化剂及其盐的制备方法 Download PDFInfo
- Publication number
- CN103974932B CN103974932B CN201280059398.5A CN201280059398A CN103974932B CN 103974932 B CN103974932 B CN 103974932B CN 201280059398 A CN201280059398 A CN 201280059398A CN 103974932 B CN103974932 B CN 103974932B
- Authority
- CN
- China
- Prior art keywords
- compound
- formula
- benzyl
- group
- alkyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Fee Related
Links
- 0 CC(C)(C(C1)C2)C1(C*SCC1(C3)C(C)(C)C3CC1N1CCOCC1)C2N1CCOCC1 Chemical compound CC(C)(C(C1)C2)C1(C*SCC1(C3)C(C)(C)C3CC1N1CCOCC1)C2N1CCOCC1 0.000 description 7
- URDRZHXRBLBOLE-UHFFFAOYSA-N CC(C)(C(C1)C2)C1(CS)C2N1CCOCC1 Chemical compound CC(C)(C(C1)C2)C1(CS)C2N1CCOCC1 URDRZHXRBLBOLE-UHFFFAOYSA-N 0.000 description 1
- FYCFSHHHAPEDIS-UHFFFAOYSA-N CC(C)(C1CC2)C1=C2SSC Chemical compound CC(C)(C1CC2)C1=C2SSC FYCFSHHHAPEDIS-UHFFFAOYSA-N 0.000 description 1
- OYILJRPBZMOPNM-UHFFFAOYSA-N CCC1(C2)C(C)(C)C2CC1N1CCOCC1 Chemical compound CCC1(C2)C(C)(C)C2CC1N1CCOCC1 OYILJRPBZMOPNM-UHFFFAOYSA-N 0.000 description 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D265/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
- C07D265/28—1,4-Oxazines; Hydrogenated 1,4-oxazines
- C07D265/30—1,4-Oxazines; Hydrogenated 1,4-oxazines not condensed with other rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B53/00—Asymmetric syntheses
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C303/00—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides
- C07C303/36—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides of amides of sulfonic acids
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
- C07D295/08—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms
- C07D295/096—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms with the ring nitrogen atoms and the oxygen or sulfur atoms separated by carbocyclic rings or by carbon chains interrupted by carbocyclic rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Catalysts (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201161565449P | 2011-11-30 | 2011-11-30 | |
| US61/565,449 | 2011-11-30 | ||
| PCT/IB2012/002910 WO2013080049A2 (en) | 2011-11-30 | 2012-11-29 | A process for the manufacture of chiral catalysts and their salts |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| CN103974932A CN103974932A (zh) | 2014-08-06 |
| CN103974932B true CN103974932B (zh) | 2016-05-18 |
Family
ID=48536192
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CN201280059398.5A Expired - Fee Related CN103974932B (zh) | 2011-11-30 | 2012-11-29 | 手性催化剂及其盐的制备方法 |
Country Status (11)
| Country | Link |
|---|---|
| US (1) | US8859765B2 (enExample) |
| EP (1) | EP2785688B1 (enExample) |
| JP (1) | JP5918386B2 (enExample) |
| KR (1) | KR101647415B1 (enExample) |
| CN (1) | CN103974932B (enExample) |
| AU (1) | AU2012346860B2 (enExample) |
| BR (1) | BR112014013285A8 (enExample) |
| CA (1) | CA2855751C (enExample) |
| IL (1) | IL232574A (enExample) |
| TW (1) | TWI483926B (enExample) |
| WO (1) | WO2013080049A2 (enExample) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP6261111B2 (ja) * | 2013-07-17 | 2018-01-17 | 国立大学法人名古屋大学 | アレーンスルホンアミドの還元方法及びアレーンスルホン酸の製法 |
| KR20160000989U (ko) | 2014-09-18 | 2016-03-28 | 엘에스산전 주식회사 | 전기 커넥터 |
| CN114436911B (zh) * | 2022-03-17 | 2023-04-28 | 南京林业大学 | 一种樟脑磺酰苄胺类化合物的制备方法及其应用 |
Citations (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20110269955A1 (en) * | 2010-04-30 | 2011-11-03 | Uang Biin-Jiun | Method for preparing 2-morpholinoisobornane- 10-thiol and intermediates formed therein |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US8168835B2 (en) * | 2010-05-26 | 2012-05-01 | National Tsing Hua University | Method for preparing propargylic alcohol catalyzed by 2-morpholinoisobornane-10-thiol |
-
2012
- 2012-11-29 JP JP2014543996A patent/JP5918386B2/ja not_active Expired - Fee Related
- 2012-11-29 AU AU2012346860A patent/AU2012346860B2/en not_active Ceased
- 2012-11-29 KR KR1020147017924A patent/KR101647415B1/ko not_active Expired - Fee Related
- 2012-11-29 BR BR112014013285A patent/BR112014013285A8/pt not_active IP Right Cessation
- 2012-11-29 CN CN201280059398.5A patent/CN103974932B/zh not_active Expired - Fee Related
- 2012-11-29 WO PCT/IB2012/002910 patent/WO2013080049A2/en not_active Ceased
- 2012-11-29 EP EP12853125.8A patent/EP2785688B1/en active Active
- 2012-11-29 US US13/689,703 patent/US8859765B2/en not_active Expired - Fee Related
- 2012-11-29 CA CA2855751A patent/CA2855751C/en not_active Expired - Fee Related
- 2012-11-30 TW TW101145127A patent/TWI483926B/zh not_active IP Right Cessation
-
2014
- 2014-05-12 IL IL232574A patent/IL232574A/en not_active IP Right Cessation
Patent Citations (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20110269955A1 (en) * | 2010-04-30 | 2011-11-03 | Uang Biin-Jiun | Method for preparing 2-morpholinoisobornane- 10-thiol and intermediates formed therein |
Non-Patent Citations (3)
| Title |
|---|
| Asymmetric Addition of Dimethylzinc to a-Ketoesters Catalyzed by (-)-MITH;Hsyueh-Liang Wu, et al.;《J. Org. Chem.》;20080723;第73卷;6445-6447 * |
| Asymmetric Synthesis of Functionalized Diarylmethanols Catalyzed by a New γ-Amino Thiol;Ping-Yu Wu, et al.;《J. Org. Chem.》;20051206;第71卷;833-835 * |
| Asymmetric synthesis of propargylic alcohols catalyzed by (-)-MITH;Ping-Yu Wu, et al.;《Tetrahedron: Asymmetry》;20090902;第20卷;1837-1841 * |
Also Published As
| Publication number | Publication date |
|---|---|
| US8859765B2 (en) | 2014-10-14 |
| KR20140097517A (ko) | 2014-08-06 |
| BR112014013285A8 (pt) | 2017-06-20 |
| WO2013080049A2 (en) | 2013-06-06 |
| US20130150574A1 (en) | 2013-06-13 |
| TWI483926B (zh) | 2015-05-11 |
| AU2012346860A1 (en) | 2014-05-29 |
| IL232574A (en) | 2017-02-28 |
| AU2012346860B2 (en) | 2015-09-24 |
| JP2015505827A (ja) | 2015-02-26 |
| CA2855751A1 (en) | 2013-06-06 |
| EP2785688A4 (en) | 2015-07-15 |
| JP5918386B2 (ja) | 2016-05-18 |
| EP2785688B1 (en) | 2017-09-13 |
| EP2785688A2 (en) | 2014-10-08 |
| BR112014013285A2 (pt) | 2017-06-13 |
| CA2855751C (en) | 2017-02-21 |
| CN103974932A (zh) | 2014-08-06 |
| WO2013080049A3 (en) | 2013-08-08 |
| KR101647415B1 (ko) | 2016-08-10 |
| IL232574A0 (en) | 2014-06-30 |
| TW201335127A (zh) | 2013-09-01 |
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| C06 | Publication | ||
| PB01 | Publication | ||
| C10 | Entry into substantive examination | ||
| SE01 | Entry into force of request for substantive examination | ||
| C14 | Grant of patent or utility model | ||
| GR01 | Patent grant | ||
| CF01 | Termination of patent right due to non-payment of annual fee |
Granted publication date: 20160518 Termination date: 20181129 |
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| CF01 | Termination of patent right due to non-payment of annual fee |