KR101647415B1 - 키랄 촉매 및 이의 염의 제조 방법 - Google Patents

키랄 촉매 및 이의 염의 제조 방법 Download PDF

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Publication number
KR101647415B1
KR101647415B1 KR1020147017924A KR20147017924A KR101647415B1 KR 101647415 B1 KR101647415 B1 KR 101647415B1 KR 1020147017924 A KR1020147017924 A KR 1020147017924A KR 20147017924 A KR20147017924 A KR 20147017924A KR 101647415 B1 KR101647415 B1 KR 101647415B1
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South Korea
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compound
formula
group
alkyl
benzyl
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KR1020147017924A
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English (en)
Korean (ko)
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KR20140097517A (ko
Inventor
핑-유 우
율리안 파울 헨쉬키
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시노팜 타이완 리미티드
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D265/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
    • C07D265/28—1,4-Oxazines; Hydrogenated 1,4-oxazines
    • C07D265/30—1,4-Oxazines; Hydrogenated 1,4-oxazines not condensed with other rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B53/00—Asymmetric syntheses
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C303/00—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides
    • C07C303/36—Preparation of esters or amides of sulfuric acids; Preparation of sulfonic acids or of their esters, halides, anhydrides or amides of amides of sulfonic acids
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
    • C07D295/08—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms
    • C07D295/096—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms with the ring nitrogen atoms and the oxygen or sulfur atoms separated by carbocyclic rings or by carbon chains interrupted by carbocyclic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Catalysts (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
KR1020147017924A 2011-11-30 2012-11-29 키랄 촉매 및 이의 염의 제조 방법 Expired - Fee Related KR101647415B1 (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201161565449P 2011-11-30 2011-11-30
US61/565,449 2011-11-30
PCT/IB2012/002910 WO2013080049A2 (en) 2011-11-30 2012-11-29 A process for the manufacture of chiral catalysts and their salts

Publications (2)

Publication Number Publication Date
KR20140097517A KR20140097517A (ko) 2014-08-06
KR101647415B1 true KR101647415B1 (ko) 2016-08-10

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KR1020147017924A Expired - Fee Related KR101647415B1 (ko) 2011-11-30 2012-11-29 키랄 촉매 및 이의 염의 제조 방법

Country Status (11)

Country Link
US (1) US8859765B2 (enExample)
EP (1) EP2785688B1 (enExample)
JP (1) JP5918386B2 (enExample)
KR (1) KR101647415B1 (enExample)
CN (1) CN103974932B (enExample)
AU (1) AU2012346860B2 (enExample)
BR (1) BR112014013285A8 (enExample)
CA (1) CA2855751C (enExample)
IL (1) IL232574A (enExample)
TW (1) TWI483926B (enExample)
WO (1) WO2013080049A2 (enExample)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP6261111B2 (ja) * 2013-07-17 2018-01-17 国立大学法人名古屋大学 アレーンスルホンアミドの還元方法及びアレーンスルホン酸の製法
KR20160000989U (ko) 2014-09-18 2016-03-28 엘에스산전 주식회사 전기 커넥터
CN114436911B (zh) * 2022-03-17 2023-04-28 南京林业大学 一种樟脑磺酰苄胺类化合物的制备方法及其应用

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20110269955A1 (en) * 2010-04-30 2011-11-03 Uang Biin-Jiun Method for preparing 2-morpholinoisobornane- 10-thiol and intermediates formed therein

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8168835B2 (en) * 2010-05-26 2012-05-01 National Tsing Hua University Method for preparing propargylic alcohol catalyzed by 2-morpholinoisobornane-10-thiol

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20110269955A1 (en) * 2010-04-30 2011-11-03 Uang Biin-Jiun Method for preparing 2-morpholinoisobornane- 10-thiol and intermediates formed therein

Also Published As

Publication number Publication date
US8859765B2 (en) 2014-10-14
KR20140097517A (ko) 2014-08-06
BR112014013285A8 (pt) 2017-06-20
WO2013080049A2 (en) 2013-06-06
US20130150574A1 (en) 2013-06-13
TWI483926B (zh) 2015-05-11
AU2012346860A1 (en) 2014-05-29
CN103974932B (zh) 2016-05-18
IL232574A (en) 2017-02-28
AU2012346860B2 (en) 2015-09-24
JP2015505827A (ja) 2015-02-26
CA2855751A1 (en) 2013-06-06
EP2785688A4 (en) 2015-07-15
JP5918386B2 (ja) 2016-05-18
EP2785688B1 (en) 2017-09-13
EP2785688A2 (en) 2014-10-08
BR112014013285A2 (pt) 2017-06-13
CA2855751C (en) 2017-02-21
CN103974932A (zh) 2014-08-06
WO2013080049A3 (en) 2013-08-08
IL232574A0 (en) 2014-06-30
TW201335127A (zh) 2013-09-01

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