CN103228643B - 作为组胺h4受体配体的苯并唑衍生物 - Google Patents

作为组胺h4受体配体的苯并唑衍生物 Download PDF

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CN103228643B
CN103228643B CN201180057036.8A CN201180057036A CN103228643B CN 103228643 B CN103228643 B CN 103228643B CN 201180057036 A CN201180057036 A CN 201180057036A CN 103228643 B CN103228643 B CN 103228643B
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methyl
methylpiperidin
yloxy
benzimidazol
phenyl
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CN103228643A (zh
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伊莎贝尔·贝雷比-伯特兰
泽维尔·比洛
蒂埃里·卡尔梅斯
马克·卡佩特
丹尼斯·丹维
史蒂芬·科瑞夫
奥利维尔·拉比奥
珍妮-玛丽·勒孔特
尼古拉斯·列沃因
泽维尔·利尼奥
菲利普·罗伯特
让-查尔斯·施瓦茨
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Bioprojet SC
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CN201180057036.8A 2010-09-27 2011-09-27 作为组胺h4受体配体的苯并唑衍生物 Active CN103228643B (zh)

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Application Number Priority Date Filing Date Title
EP20100306038 EP2447263A1 (en) 2010-09-27 2010-09-27 Benzazole derivatives as histamine H4 receptor ligands
EP10306038.0 2010-09-27
PCT/EP2011/066782 WO2012041860A1 (en) 2010-09-27 2011-09-27 Benzazole derivatives as histamine h4 receptor ligands

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CN103228643A CN103228643A (zh) 2013-07-31
CN103228643B true CN103228643B (zh) 2015-11-25

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CN106800524A (zh) * 2015-02-13 2017-06-06 佛山市赛维斯医药科技有限公司 一类含双酰肼和萘基结构的化合物、制备方法及其用途
JP7447002B2 (ja) * 2017-09-11 2024-03-11 クルーゾン・ファーマシューティカルズ・インコーポレイテッド ＳＨＰ２のオクタヒドロシクロペンタ［ｃ］ピロールのアロステリック阻害剤
RS60320B1 (sr) * 2017-11-15 2020-07-31 Bioprojet Soc Civ Derivati benzimidazola kao dvostruki ligandi histaminskog h1 i histaminskog h4 receptora
CN113278409B (zh) * 2021-06-22 2022-04-29 西南石油大学 一种高温酸化缓蚀剂
CN119086786B (zh) * 2024-11-08 2025-02-14 南京恒远科技开发有限公司 叔丁基-(s)-[2-(2-氰基-4,4-二氟吡咯烷-1-基)-2-氧乙基]氨基甲酸酯光学异构体的检测方法

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CN103228643A (zh) 2013-07-31
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EP2621916A1 (en) 2013-08-07
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