CN102516086B - 胺的制备方法 - Google Patents

胺的制备方法 Download PDF

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Publication number
CN102516086B
CN102516086B CN201110318357.0A CN201110318357A CN102516086B CN 102516086 B CN102516086 B CN 102516086B CN 201110318357 A CN201110318357 A CN 201110318357A CN 102516086 B CN102516086 B CN 102516086B
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China
Prior art keywords
compound
general formula
formula
palladium
alkyl
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CN201110318357.0A
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English (en)
Chinese (zh)
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CN102516086A (zh
Inventor
H·托布勒
H·沃尔特
C·科尔西
J·埃伦弗罗因德
F·焦尔达诺
M·泽勒
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Syngenta Group Inc
Syngenta Participations AG
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Syngenta Participations AG
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C209/00—Preparation of compounds containing amino groups bound to a carbon skeleton
    • C07C209/62—Preparation of compounds containing amino groups bound to a carbon skeleton by cleaving carbon-to-nitrogen, sulfur-to-nitrogen, or phosphorus-to-nitrogen bonds, e.g. hydrolysis of amides, N-dealkylation of amines or quaternary ammonium compounds
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C209/00—Preparation of compounds containing amino groups bound to a carbon skeleton
    • C07C209/24—Preparation of compounds containing amino groups bound to a carbon skeleton by reductive alkylation of ammonia, amines or compounds having groups reducible to amino groups, with carbonyl compounds
    • C07C209/28—Preparation of compounds containing amino groups bound to a carbon skeleton by reductive alkylation of ammonia, amines or compounds having groups reducible to amino groups, with carbonyl compounds by reduction with other reducing agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C17/00—Preparation of halogenated hydrocarbons
    • C07C17/23—Preparation of halogenated hydrocarbons by dehalogenation
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C17/00—Preparation of halogenated hydrocarbons
    • C07C17/26—Preparation of halogenated hydrocarbons by reactions involving an increase in the number of carbon atoms in the skeleton
    • C07C17/30—Preparation of halogenated hydrocarbons by reactions involving an increase in the number of carbon atoms in the skeleton by a Diels-Alder synthesis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C17/00—Preparation of halogenated hydrocarbons
    • C07C17/35—Preparation of halogenated hydrocarbons by reactions not affecting the number of carbon or of halogen atoms in the reaction
    • C07C17/354—Preparation of halogenated hydrocarbons by reactions not affecting the number of carbon or of halogen atoms in the reaction by hydrogenation
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C209/00—Preparation of compounds containing amino groups bound to a carbon skeleton
    • C07C209/04—Preparation of compounds containing amino groups bound to a carbon skeleton by substitution of functional groups by amino groups
    • C07C209/06—Preparation of compounds containing amino groups bound to a carbon skeleton by substitution of functional groups by amino groups by substitution of halogen atoms
    • C07C209/10—Preparation of compounds containing amino groups bound to a carbon skeleton by substitution of functional groups by amino groups by substitution of halogen atoms with formation of amino groups bound to carbon atoms of six-membered aromatic rings or from amines having nitrogen atoms bound to carbon atoms of six-membered aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C209/00—Preparation of compounds containing amino groups bound to a carbon skeleton
    • C07C209/24—Preparation of compounds containing amino groups bound to a carbon skeleton by reductive alkylation of ammonia, amines or compounds having groups reducible to amino groups, with carbonyl compounds
    • C07C209/26—Preparation of compounds containing amino groups bound to a carbon skeleton by reductive alkylation of ammonia, amines or compounds having groups reducible to amino groups, with carbonyl compounds by reduction with hydrogen
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C209/00—Preparation of compounds containing amino groups bound to a carbon skeleton
    • C07C209/68—Preparation of compounds containing amino groups bound to a carbon skeleton from amines, by reactions not involving amino groups, e.g. reduction of unsaturated amines, aromatisation, or substitution of the carbon skeleton
    • C07C209/70—Preparation of compounds containing amino groups bound to a carbon skeleton from amines, by reactions not involving amino groups, e.g. reduction of unsaturated amines, aromatisation, or substitution of the carbon skeleton by reduction of unsaturated amines
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C211/00—Compounds containing amino groups bound to a carbon skeleton
    • C07C211/43—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton
    • C07C211/57—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton having amino groups bound to carbon atoms of six-membered aromatic rings being part of condensed ring systems of the carbon skeleton
    • C07C211/60—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton having amino groups bound to carbon atoms of six-membered aromatic rings being part of condensed ring systems of the carbon skeleton containing a ring other than a six-membered aromatic ring forming part of at least one of the condensed ring systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C211/00—Compounds containing amino groups bound to a carbon skeleton
    • C07C211/43—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton
    • C07C211/57—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton having amino groups bound to carbon atoms of six-membered aromatic rings being part of condensed ring systems of the carbon skeleton
    • C07C211/61—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton having amino groups bound to carbon atoms of six-membered aromatic rings being part of condensed ring systems of the carbon skeleton with at least one of the condensed ring systems formed by three or more rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C25/00—Compounds containing at least one halogen atom bound to a six-membered aromatic ring
    • C07C25/18—Polycyclic aromatic halogenated hydrocarbons
    • C07C25/22—Polycyclic aromatic halogenated hydrocarbons with condensed rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C25/00—Compounds containing at least one halogen atom bound to a six-membered aromatic ring
    • C07C25/24—Halogenated aromatic hydrocarbons with unsaturated side chains
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/09—Geometrical isomers
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2603/00—Systems containing at least three condensed rings
    • C07C2603/56—Ring systems containing bridged rings
    • C07C2603/58—Ring systems containing bridged rings containing three rings
    • C07C2603/60—Ring systems containing bridged rings containing three rings containing at least one ring with less than six members
    • C07C2603/66—Ring systems containing bridged rings containing three rings containing at least one ring with less than six members containing five-membered rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Catalysts (AREA)
CN201110318357.0A 2005-12-12 2006-12-11 胺的制备方法 Active CN102516086B (zh)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
EP05027072 2005-12-12
EP05027072.7 2005-12-12
EP06008248 2006-04-21
EP06008248.4 2006-04-21

Related Parent Applications (1)

Application Number Title Priority Date Filing Date
CN200680051127XA Division CN101360703B (zh) 2005-12-12 2006-12-11 胺的制备方法

Publications (2)

Publication Number Publication Date
CN102516086A CN102516086A (zh) 2012-06-27
CN102516086B true CN102516086B (zh) 2014-10-22

Family

ID=37946810

Family Applications (3)

Application Number Title Priority Date Filing Date
CN201110318357.0A Active CN102516086B (zh) 2005-12-12 2006-12-11 胺的制备方法
CN200680051127XA Active CN101360703B (zh) 2005-12-12 2006-12-11 胺的制备方法
CN201410401736.XA Active CN104151132B (zh) 2005-12-12 2006-12-11 胺的制备方法

Family Applications After (2)

Application Number Title Priority Date Filing Date
CN200680051127XA Active CN101360703B (zh) 2005-12-12 2006-12-11 胺的制备方法
CN201410401736.XA Active CN104151132B (zh) 2005-12-12 2006-12-11 胺的制备方法

Country Status (21)

Country Link
US (1) US7781615B2 (enExample)
EP (5) EP2316814A1 (enExample)
JP (1) JP5144533B2 (enExample)
KR (1) KR101364220B1 (enExample)
CN (3) CN102516086B (enExample)
AR (1) AR058302A1 (enExample)
AU (1) AU2006326289B2 (enExample)
BR (1) BRPI0619629B1 (enExample)
CA (1) CA2631973C (enExample)
CL (2) CL2010000015A1 (enExample)
CR (1) CR10052A (enExample)
DK (1) DK1963251T3 (enExample)
EA (1) EA014275B1 (enExample)
EC (1) ECSP088525A (enExample)
EG (1) EG25547A (enExample)
ES (1) ES2391904T3 (enExample)
IL (3) IL191760A (enExample)
IN (1) IN2015DN00818A (enExample)
PL (1) PL1963251T3 (enExample)
TW (1) TWI396676B (enExample)
WO (1) WO2007068417A2 (enExample)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PL1963251T3 (pl) * 2005-12-12 2013-01-31 Syngenta Participations Ag Proces wytwarzania amin
UA109173C2 (uk) 2007-09-20 2015-07-27 Склад, що містить фунгіцидний штам і хімічну сполуку
UA101382C2 (ru) 2008-07-04 2013-03-25 Басф Се Фунгицидные смеси, содержащие замещенные 1-метилпиразол-4-илкарбоксанилиды
EA019039B1 (ru) 2008-10-27 2013-12-30 Зингента Партисипейшнс Аг Способ получения бензонорборненов
BRPI0923401B1 (pt) 2008-12-24 2021-11-23 Syngenta Limited Método para o preparo de aril amidas e composto
JP6153864B2 (ja) * 2010-04-20 2017-06-28 シンジェンタ パーティシペーションズ アクチェンゲゼルシャフト ピラゾールカルボン酸アミドの調製方法
JP5833663B2 (ja) 2010-11-15 2015-12-16 バイエル・インテレクチュアル・プロパティ・ゲゼルシャフト・ミット・ベシュレンクテル・ハフツングＢａｙｅｒ Ｉｎｔｅｌｌｅｃｔｕａｌ Ｐｒｏｐｅｒｔｙ ＧｍｂＨ ５−ハロゲノピラゾールカルボキサミド類
RU2493145C1 (ru) * 2012-10-02 2013-09-20 Федеральное государственное бюджетное образовательное учреждение высшего профессионального образования "Волгоградский государственный технический университет" (ВолгГТУ) Способ получения 2-(аминоалкил)-3-(аминофенил)бицикло[2.2.1]гептанов
RU2657017C2 (ru) 2013-03-14 2018-06-08 ДАУ АГРОСАЙЕНСИЗ ЭлЭлСи Контроль широколиственных культур с помощью 6-арилпиколинкарбоновых кислот, 2-арилпиримидинкарбоновых кислот или их солей или сложных эфиров
US11560384B2 (en) 2017-05-04 2023-01-24 University Of Utah Research Foundation Benzonorbornadiene derivatives and reactions thereof

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN1705668A (zh) * 2002-10-18 2005-12-07 辛根塔参与股份公司 杂环甲酰胺衍生物

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1086978A (en) * 1965-09-21 1967-10-11 Shionogi & Co Improvements in or relating to the preparation of 7-oxobenzonorbornene derivatives
JPH075487B2 (ja) 1985-11-14 1995-01-25 住友化学工業株式会社 １―ブロモ―２―クロロ―４―フルオロベンゼンの製造法
US7223879B2 (en) 1998-07-10 2007-05-29 Massachusetts Institute Of Technology Ligands for metals and improved metal-catalyzed processes based thereon
KR20030093240A (ko) * 2001-03-16 2003-12-06 이데미쓰 고산 가부시키가이샤 방향족 아미노 화합물의 제조방법
JP4219622B2 (ja) * 2002-06-11 2009-02-04 独立行政法人科学技術振興機構 ベンザイン化合物の新規製造法
EP1539717B1 (en) * 2002-08-22 2011-07-13 Syngenta Participations AG Microbiocidal (e.g fungicidal) 1,2,3-triazole derivatives
PL1963251T3 (pl) * 2005-12-12 2013-01-31 Syngenta Participations Ag Proces wytwarzania amin

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN1705668A (zh) * 2002-10-18 2005-12-07 辛根塔参与股份公司 杂环甲酰胺衍生物

Also Published As

Publication number Publication date
KR20080077011A (ko) 2008-08-20
EP2316813A1 (en) 2011-05-04
IL218350A0 (en) 2012-04-30
CN101360703B (zh) 2012-07-18
EP2316813B1 (en) 2013-04-03
ES2391904T3 (es) 2012-11-30
TW200800854A (en) 2008-01-01
US20090221856A1 (en) 2009-09-03
WO2007068417A3 (en) 2007-10-04
EG25547A (en) 2012-02-15
CN102516086A (zh) 2012-06-27
BRPI0619629A2 (pt) 2011-10-04
KR101364220B1 (ko) 2014-02-21
CA2631973A1 (en) 2007-06-21
DK1963251T3 (da) 2012-11-26
CN104151132B (zh) 2016-07-06
CN104151132A (zh) 2014-11-19
JP2009518346A (ja) 2009-05-07
EP2316809B1 (en) 2014-06-18
AR058302A1 (es) 2008-01-30
IL191760A0 (en) 2008-12-29
CR10052A (es) 2008-09-17
JP5144533B2 (ja) 2013-02-13
IN2015DN00818A (enExample) 2015-07-10
US7781615B2 (en) 2010-08-24
CA2631973C (en) 2015-02-03
EP2316815A1 (en) 2011-05-04
CL2010000015A1 (es) 2010-07-02
BRPI0619629B1 (pt) 2016-03-01
IL218351A0 (en) 2012-04-30
ECSP088525A (es) 2008-07-30
AU2006326289A1 (en) 2007-06-21
IL191760A (en) 2014-05-28
PL1963251T3 (pl) 2013-01-31
IL218351A (en) 2014-05-28
EA014275B1 (ru) 2010-10-29
EP2316814A1 (en) 2011-05-04
TWI396676B (zh) 2013-05-21
AU2006326289B2 (en) 2011-12-22
EA200870038A1 (ru) 2008-10-30
EP1963251B1 (en) 2012-08-15
EP2316809A1 (en) 2011-05-04
WO2007068417A2 (en) 2007-06-21
CL2012000114A1 (es) 2012-08-31
CN101360703A (zh) 2009-02-04
EP1963251A2 (en) 2008-09-03

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GR01 Patent grant
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Effective date of registration: 20221102

Address after: Basel, SUI

Patentee after: SYNGENTA PARTICIPATIONS AG

Patentee after: Syngenta Group Inc.

Address before: Basel, SUI

Patentee before: SYNGENTA PARTICIPATIONS AG

TR01 Transfer of patent right